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Design and optimization of renin inhibitors: Orally bioavailable alkyl amines. [electronic resource] by
- Tice, Colin M
- Xu, Zhenrong
- Yuan, Jing
- Simpson, Robert D
- Cacatian, Salvacion T
- Flaherty, Patrick T
- Zhao, Wei
- Guo, Joan
- Ishchenko, Alexey
- Singh, Suresh B
- Wu, Zhongren
- Scott, Boyd B
- Bukhtiyarov, Yuri
- Berbaum, Jennifer
- Mason, Jennifer
- Panemangalore, Reshma
- Cappiello, Maria Grazia
- Müller, Dominik
- Harrison, Richard K
- McGeehan, Gerard M
- Dillard, Lawrence W
- Baldwin, John J
- Claremon, David A
Producer: 20090901
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
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5.
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Spirocyclic ureas: orally bioavailable 11 beta-HSD1 inhibitors identified by computer-aided drug design. [electronic resource] by
- Tice, Colin M
- Zhao, Wei
- Xu, Zhenrong
- Cacatian, Salvacion T
- Simpson, Robert D
- Ye, Yuan-Jie
- Singh, Suresh B
- McKeever, Brian M
- Lindblom, Peter
- Guo, Joan
- Krosky, Paula M
- Kruk, Barbara A
- Berbaum, Jennifer
- Harrison, Richard K
- Johnson, Judith J
- Bukhtiyarov, Yuri
- Panemangalore, Reshma
- Scott, Boyd B
- Zhao, Yi
- Bruno, Joseph G
- Zhuang, Linghang
- McGeehan, Gerard M
- He, Wei
- Claremon, David A
Producer: 20100920
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
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6.
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Biphenyl/diphenyl ether renin inhibitors: filling the S1 pocket of renin via the S3 pocket. [electronic resource] by
- Yuan, Jing
- Simpson, Robert D
- Zhao, Wei
- Tice, Colin M
- Xu, Zhenrong
- Cacatian, Salvacion
- Jia, Lanqi
- Flaherty, Patrick T
- Guo, Joan
- Ishchenko, Alexey
- Wu, Zhongren
- McKeever, Brian M
- Scott, Boyd B
- Bukhtiyarov, Yuri
- Berbaum, Jennifer
- Panemangalore, Reshma
- Bentley, Ross
- Doe, Christopher P
- Harrison, Richard K
- McGeehan, Gerard M
- Singh, Suresh B
- Dillard, Lawrence W
- Baldwin, John J
- Claremon, David A
Producer: 20111122
In:
Bioorganic & medicinal chemistry letters vol. 21
Availability: No items available.
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7.
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Structure-based design and synthesis of 1,3-oxazinan-2-one inhibitors of 11β-hydroxysteroid dehydrogenase type 1. [electronic resource] by
- Xu, Zhenrong
- Tice, Colin M
- Zhao, Wei
- Cacatian, Salvacion
- Ye, Yuan-Jie
- Singh, Suresh B
- Lindblom, Peter
- McKeever, Brian M
- Krosky, Paula M
- Kruk, Barbara A
- Berbaum, Jennifer
- Harrison, Richard K
- Johnson, Judith A
- Bukhtiyarov, Yuri
- Panemangalore, Reshma
- Scott, Boyd B
- Zhao, Yi
- Bruno, Joseph G
- Togias, Jennifer
- Guo, Joan
- Guo, Rong
- Carroll, Patrick J
- McGeehan, Gerard M
- Zhuang, Linghang
- He, Wei
- Claremon, David A
Producer: 20111031
In:
Journal of medicinal chemistry vol. 54
Availability: No items available.
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8.
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Optimization of orally bioavailable alkyl amine renin inhibitors. [electronic resource] by
- Xu, Zhenrong
- Cacatian, Salvacion
- Yuan, Jing
- Simpson, Robert D
- Jia, Lanqi
- Zhao, Wei
- Tice, Colin M
- Flaherty, Patrick T
- Guo, Joan
- Ishchenko, Alexey
- Singh, Suresh B
- Wu, Zhongren
- McKeever, Brian M
- Scott, Boyd B
- Bukhtiyarov, Yuri
- Berbaum, Jennifer
- Mason, Jennifer
- Panemangalore, Reshma
- Cappiello, Maria Grazia
- Bentley, Ross
- Doe, Christopher P
- Harrison, Richard K
- McGeehan, Gerard M
- Dillard, Lawrence W
- Baldwin, John J
- Claremon, David A
Producer: 20100420
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
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9.
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Discovery and optimization of adamantyl carbamate inhibitors of 11β-HSD1. [electronic resource] by
- Tice, Colin M
- Zhao, Wei
- Krosky, Paula M
- Kruk, Barbara A
- Berbaum, Jennifer
- Johnson, Judith A
- Bukhtiyarov, Yuri
- Panemangalore, Reshma
- Scott, Boyd B
- Zhao, Yi
- Bruno, Joseph G
- Howard, Lamont
- Togias, Jennifer
- Ye, Yuan-Jie
- Singh, Suresh B
- McKeever, Brian M
- Lindblom, Peter R
- Guo, Joan
- Guo, Rong
- Nar, Herbert
- Schuler-Metz, Annette
- Gregg, Richard E
- Leftheris, Katerina
- Harrison, Richard K
- McGeehan, Gerard M
- Zhuang, Linghang
- Claremon, David A
Producer: 20110329
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
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