The novel compound (+/-)-1-[10-((E)-3-Phenyl-allyl)-3,10-diaza-bicyclo[4.3.1]dec-3-yl]-propan-1-one (NS7051) attenuates nociceptive transmission in animal models of experimental pain; a pharmacological comparison with the combined mu-opioid receptor agonist and monoamine reuptake inhibitor tramadol. [electronic resource]
Producer: 20080512Description: 331-43 p. digitalISSN:- 0028-3908
- Analgesics, Opioid -- pharmacology
- Animals
- Azabicyclo Compounds -- pharmacology
- Behavior, Animal -- drug effects
- Brain -- metabolism
- Dose-Response Relationship, Drug
- Formaldehyde
- Freund's Adjuvant
- Inflammation -- chemically induced
- Male
- Microdialysis
- Neurotransmitter Uptake Inhibitors -- pharmacology
- Nociceptors -- drug effects
- Pain -- drug therapy
- Pain Measurement -- drug effects
- Postural Balance -- drug effects
- Rats
- Rats, Sprague-Dawley
- Reaction Time
- Receptors, Opioid, delta -- drug effects
- Receptors, Opioid, mu -- agonists
- Synaptic Transmission -- drug effects
- Tramadol -- pharmacology
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Publication Type: Comparative Study; Journal Article
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