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Thermodynamic and kinetic characterization of hydroxyethylamine β-secretase-1 inhibitors. [electronic resource] by
- Mondal, Kalyani
- Regnstrom, Karin
- Morishige, Winse
- Barbour, Robin
- Probst, Gary
- Xu, Ying-Zi
- Artis, Dean R
- Yao, Nanhua
- Beroza, Paul
- Bova, Michael P
Producer: 20140117
In:
Biochemical and biophysical research communications vol. 441
Availability: No items available.
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6.
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Development of a novel β-secretase binding assay using the AlphaScreen platform. [electronic resource] by
- Ren, Zhao
- Tam, Danny
- Xu, Ying-Zi
- Wone, David
- Yuan, Shendong
- Sham, Hing L
- Cheung, Harry
- Regnstrom, Karin
- Chen, Xiaohua
- Rudolph, Donald
- Jobling, Michael F
- Artis, Dean R
- Bova, Michael P
Producer: 20140220
In:
Journal of biomolecular screening vol. 18
Availability: No items available.
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7.
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Selective alpha4beta7 integrin antagonists and their potential as antiinflammatory agents. [electronic resource] by
- Dubree, Nathan J P
- Artis, Dean R
- Castanedo, Georgette
- Marsters, James
- Sutherlin, Daniel
- Caris, Lisa
- Clark, Kevin
- Keating, Susan M
- Beresini, Maureen H
- Chiu, Henry
- Fong, Sherman
- Lowman, Henry B
- Skelton, Nicholas J
- Jackson, David Y
Producer: 20020819
In:
Journal of medicinal chemistry vol. 45
Availability: No items available.
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8.
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A family of phosphodiesterase inhibitors discovered by cocrystallography and scaffold-based drug design. [electronic resource] by
- Card, Graeme L
- Blasdel, Landy
- England, Bruce P
- Zhang, Chao
- Suzuki, Yoshihisa
- Gillette, Sam
- Fong, Daniel
- Ibrahim, Prabha N
- Artis, Dean R
- Bollag, Gideon
- Milburn, Michael V
- Kim, Sung-Hou
- Schlessinger, Joseph
- Zhang, Kam Y J
Producer: 20050531
In:
Nature biotechnology vol. 23
Availability: No items available.
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9.
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Structural basis for the activity of drugs that inhibit phosphodiesterases. [electronic resource] by
- Card, Graeme L
- England, Bruce P
- Suzuki, Yoshihisa
- Fong, Daniel
- Powell, Ben
- Lee, Byunghun
- Luu, Catherine
- Tabrizizad, Maryam
- Gillette, Sam
- Ibrahim, Prabha N
- Artis, Dean R
- Bollag, Gideon
- Milburn, Michael V
- Kim, Sung-Hou
- Schlessinger, Joseph
- Zhang, Kam Y J
Producer: 20050531
In:
Structure (London, England : 1993) vol. 12
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10.
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Label free fragment screening using surface plasmon resonance as a tool for fragment finding - analyzing parkin, a difficult CNS target. [electronic resource] by
- Regnström, Karin
- Yan, Jiangli
- Nguyen, Lan
- Callaway, Kari
- Yang, Yanli
- Diep, Linnea
- Xing, Weimei
- Adhikari, Anirban
- Beroza, Paul
- Hom, Roy K
- Riley, Brigit
- Rudolph, Don
- Jobling, Michael F
- Baker, Jeanne
- Johnston, Jennifer
- Konradi, Andrei
- Bova, Michael P
- Artis, Dean R
- Artis, Rick D
Producer: 20140213
In:
PloS one vol. 8
Availability: No items available.
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11.
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Design and synthesis of thiophene dihydroisoquinolines as novel BACE1 inhibitors. [electronic resource] by
- Xu, Ying-Zi
- Yuan, Shendong
- Bowers, Simeon
- Hom, Roy K
- Chan, Wayman
- Sham, Hing L
- Zhu, Yong L
- Beroza, Paul
- Pan, Hu
- Brecht, Eric
- Yao, Nanhua
- Lougheed, Julie
- Yan, Jiangli
- Tam, Danny
- Ren, Zhao
- Ruslim, Lany
- Bova, Michael P
- Artis, Dean R
Producer: 20131126
In:
Bioorganic & medicinal chemistry letters vol. 23
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12.
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A selective, slow binding inhibitor of factor VIIa binds to a nonstandard active site conformation and attenuates thrombus formation in vivo. [electronic resource] by
- Olivero, Alan G
- Eigenbrot, Charles
- Goldsmith, Richard
- Robarge, Kirk
- Artis, Dean R
- Flygare, John
- Rawson, Thomas
- Sutherlin, Daniel P
- Kadkhodayan, Saloumeh
- Beresini, Maureen
- Elliott, Linda O
- DeGuzman, Geralyn G
- Banner, David W
- Ultsch, Mark
- Marzec, Ulla
- Hanson, Stephen R
- Refino, Canio
- Bunting, Stuart
- Kirchhofer, Daniel
Producer: 20050419
In:
The Journal of biological chemistry vol. 280
Availability: No items available.
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13.
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Structure-based design of novel dihydroisoquinoline BACE-1 inhibitors that do not engage the catalytic aspartates. [electronic resource] by
- Bowers, Simeon
- Xu, Ying-zi
- Yuan, Shendong
- Probst, Gary D
- Hom, Roy K
- Chan, Wayman
- Konradi, Andrei W
- Sham, Hing L
- Zhu, Yong L
- Beroza, Paul
- Pan, Hu
- Brecht, Eric
- Yao, Nanhua
- Lougheed, Julie
- Tam, Danny
- Ren, Zhao
- Ruslim, Lany
- Bova, Michael P
- Artis, Dean R
Producer: 20130930
In:
Bioorganic & medicinal chemistry letters vol. 23
Availability: No items available.
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14.
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Design and synthesis of disubstituted thiophene and thiazole based inhibitors of JNK. [electronic resource] by
- Hom, Roy K
- Bowers, Simeon
- Sealy, Jennifer M
- Truong, Anh P
- Probst, Gary D
- Neitzel, Martin L
- Neitz, R Jeffrey
- Fang, Larry
- Brogley, Louis
- Wu, Jing
- Konradi, Andrei W
- Sham, Hing L
- Tóth, Gergely
- Pan, Hu
- Yao, Nanhua
- Artis, Dean R
- Quinn, Kevin
- Sauer, John-Michael
- Powell, Kyle
- Ren, Zhao
- Bard, Frédérique
- Yednock, Ted A
- Griswold-Prenner, Irene
Producer: 20110314
In:
Bioorganic & medicinal chemistry letters vol. 20
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15.
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Design and synthesis of a novel, orally active, brain penetrant, tri-substituted thiophene based JNK inhibitor. [electronic resource] by
- Bowers, Simeon
- Truong, Anh P
- Neitz, R Jeffrey
- Neitzel, Martin
- Probst, Gary D
- Hom, Roy K
- Peterson, Brian
- Galemmo, Robert A
- Konradi, Andrei W
- Sham, Hing L
- Tóth, Gergley
- Pan, Hu
- Yao, Nanhua
- Artis, Dean R
- Brigham, Elizabeth F
- Quinn, Kevin P
- Sauer, John-Michael
- Powell, Kyle
- Ruslim, Lany
- Ren, Zhao
- Bard, Frédérique
- Yednock, Ted A
- Griswold-Prenner, Irene
Producer: 20110705
In:
Bioorganic & medicinal chemistry letters vol. 21
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16.
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Design and pharmacology of a highly specific dual FMS and KIT kinase inhibitor. [electronic resource] by
- Zhang, Chao
- Ibrahim, Prabha N
- Zhang, Jiazhong
- Burton, Elizabeth A
- Habets, Gaston
- Zhang, Ying
- Powell, Ben
- West, Brian L
- Matusow, Bernice
- Tsang, Garson
- Shellooe, Rafe
- Carias, Heidi
- Nguyen, Hoa
- Marimuthu, Adhirai
- Zhang, Kam Y J
- Oh, Angela
- Bremer, Ryan
- Hurt, Clarence R
- Artis, Dean R
- Wu, Guoxian
- Nespi, Marika
- Spevak, Wayne
- Lin, Paul
- Nolop, Keith
- Hirth, Peter
- Tesch, Greg H
- Bollag, Gideon
Producer: 20130611
In:
Proceedings of the National Academy of Sciences of the United States of America vol. 110
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17.
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Improving the permeability of the hydroxyethylamine BACE-1 inhibitors: structure-activity relationship of P2' substituents. [electronic resource] by
- Truong, Anh P
- Probst, Gary D
- Aquino, Jose
- Fang, Larry
- Brogley, Louis
- Sealy, Jennifer M
- Hom, Roy K
- Tucker, John A
- John, Varghese
- Tung, Jay S
- Pleiss, Michael A
- Konradi, Andrei W
- Sham, Hing L
- Dappen, Michael S
- Tóth, Gergley
- Yao, Nanhua
- Brecht, Eric
- Pan, Hu
- Artis, Dean R
- Ruslim, Lany
- Bova, Michael P
- Sinha, Sukanto
- Yednock, Ted A
- Zmolek, Wes
- Quinn, Kevin P
- Sauer, John-Michael
Producer: 20101110
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
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18.
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Design and synthesis of hydroxyethylamine (HEA) BACE-1 inhibitors: prime side chromane-containing inhibitors. [electronic resource] by
- Ng, Raymond A
- Sun, Minghua
- Bowers, Simeon
- Hom, Roy K
- Probst, Gary D
- John, Varghese
- Fang, Lawrence Y
- Maillard, Michel
- Gailunas, Andrea
- Brogley, Louis
- Neitz, R Jeffrey
- Tung, Jay S
- Pleiss, Michael A
- Konradi, Andrei W
- Sham, Hing L
- Dappen, Michael S
- Adler, Marc
- Yao, Nanhua
- Zmolek, Wes
- Nakamura, David
- Quinn, Kevin P
- Sauer, John-Michael
- Bova, Michael P
- Ruslim, Lany
- Artis, Dean R
- Yednock, Ted A
Producer: 20140130
In:
Bioorganic & medicinal chemistry letters vol. 23
Availability: No items available.
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19.
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Design and synthesis of highly selective, orally active Polo-like kinase-2 (Plk-2) inhibitors. [electronic resource] by
- Bowers, Simeon
- Truong, Anh P
- Ye, Michael
- Aubele, Danielle L
- Sealy, Jennifer M
- Neitz, R Jeffrey
- Hom, Roy K
- Chan, Wayman
- Dappen, Michael S
- Galemmo, Robert A
- Konradi, Andrei W
- Sham, Hing L
- Zhu, Yong L
- Beroza, Paul
- Tonn, George
- Zhang, Heather
- Hoffman, Jennifer
- Motter, Ruth
- Fauss, Donald
- Tanaka, Pearl
- Bova, Michael P
- Ren, Zhao
- Tam, Danny
- Ruslim, Lany
- Baker, Jeanne
- Pandya, Deepal
- Diep, Linnea
- Fitzgerald, Kent
- Artis, Dean R
- Anderson, John P
- Bergeron, Marcelle
Producer: 20131108
In:
Bioorganic & medicinal chemistry letters vol. 23
Availability: No items available.
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20.
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Highly selective c-Jun N-terminal kinase (JNK) 2 and 3 inhibitors with in vitro CNS-like pharmacokinetic properties prevent neurodegeneration. [electronic resource] by
- Probst, Gary D
- Bowers, Simeon
- Sealy, Jennifer M
- Truong, Anh P
- Hom, Roy K
- Galemmo, Robert A
- Konradi, Andrei W
- Sham, Hing L
- Quincy, David A
- Pan, Hu
- Yao, Nanhua
- Lin, May
- Tóth, Gergley
- Artis, Dean R
- Zmolek, Wes
- Wong, Karina
- Qin, Ann
- Lorentzen, Colin
- Nakamura, David F
- Quinn, Kevin P
- Sauer, John-Michael
- Powell, Kyle
- Ruslim, Lany
- Wright, Sarah
- Chereau, David
- Ren, Zhao
- Anderson, John P
- Bard, Frédérique
- Yednock, Ted A
- Griswold-Prenner, Irene
Producer: 20110414
In:
Bioorganic & medicinal chemistry letters vol. 21
Availability: No items available.
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