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Pharmacophore Identification and Scaffold Exploration to Discover Novel, Potent, and Chemically Stable Inhibitors of Acid Ceramidase in Melanoma Cells. [electronic resource] by
- Ortega, Jose Antonio
- Arencibia, Jose M
- La Sala, Giuseppina
- Borgogno, Marco
- Bauer, Inga
- Bono, Luca
- Braccia, Clarissa
- Armirotti, Andrea
- Girotto, Stefania
- Ganesan, Anand
- De Vivo, Marco
Producer: 20170801
In:
Journal of medicinal chemistry vol. 60
Availability: No items available.
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Design, Synthesis, Dynamic Docking, Biochemical Characterization, and [electronic resource] by
- Arencibia, Jose M
- Brindani, Nicoletta
- Franco-Ulloa, Sebastian
- Nigro, Michela
- Kuriappan, Jissy Akkarapattiakal
- Ottonello, Giuliana
- Bertozzi, Sine Mandrup
- Summa, Maria
- Girotto, Stefania
- Bertorelli, Rosalia
- Armirotti, Andrea
- De Vivo, Marco
Producer: 20201007
In:
Journal of medicinal chemistry vol. 63
Availability: No items available.
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Substrate-selective inhibition of protein kinase PDK1 by small compounds that bind to the PIF-pocket allosteric docking site. [electronic resource] by
- Busschots, Katrien
- Lopez-Garcia, Laura A
- Lammi, Carmen
- Stroba, Adriana
- Zeuzem, Stefan
- Piiper, Albrecht
- Alzari, Pedro M
- Neimanis, Sonja
- Arencibia, Jose M
- Engel, Matthias
- Schulze, Jörg O
- Biondi, Ricardo M
Producer: 20140710
In:
Chemistry & biology vol. 19
Availability: No items available.
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An Allosteric Inhibitor Scaffold Targeting the PIF-Pocket of Atypical Protein Kinase C Isoforms. [electronic resource] by
- Arencibia, Jose M
- Fröhner, Wolfgang
- Krupa, Magdalena
- Pastor-Flores, Daniel
- Merker, Piotr
- Oellerich, Thomas
- Neimanis, Sonja
- Schmithals, Christian
- Köberle, Verena
- Süß, Evelyn
- Zeuzem, Stefan
- Stark, Holger
- Piiper, Albrecht
- Odadzic, Dalibor
- Schulze, Jörg O
- Biondi, Ricardo M
Producer: 20170711
In:
ACS chemical biology vol. 12
Availability: No items available.
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Improving Drug Penetrability with iRGD Leverages the Therapeutic Response to Sorafenib and Doxorubicin in Hepatocellular Carcinoma. [electronic resource] by
- Schmithals, Christian
- Köberle, Verena
- Korkusuz, Hüdayi
- Pleli, Thomas
- Kakoschky, Bianca
- Augusto, Eduardo Alonso
- Ibrahim, Ahmed Atef
- Arencibia, Jose M
- Vafaizadeh, Vida
- Groner, Bernd
- Korf, Horst-Werner
- Kronenberger, Bernd
- Zeuzem, Stefan
- Vogl, Thomas J
- Waidmann, Oliver
- Piiper, Albrecht
Producer: 20151026
In:
Cancer research vol. 75
Availability: No items available.
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12.
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Molecular mechanism of regulation of the atypical protein kinase C by N-terminal domains and an allosteric small compound. [electronic resource] by
- Zhang, Hua
- Neimanis, Sonja
- Lopez-Garcia, Laura A
- Arencibia, José M
- Amon, Sabine
- Stroba, Adriana
- Zeuzem, Stefan
- Proschak, Ewgen
- Stark, Holger
- Bauer, Angelika F
- Busschots, Katrien
- Jørgensen, Thomas J D
- Engel, Matthias
- Schulze, Jörg O
- Biondi, Ricardo M
Producer: 20150331
In:
Chemistry & biology vol. 21
Availability: No items available.
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