Results
|
1.
|
Preclinical disposition of GDC-0973 and prospective and retrospective analysis of human dose and efficacy predictions. [electronic resource] by
- Choo, Edna F
- Belvin, Marcia
- Boggs, Jason
- Deng, Yuzhong
- Hoeflich, Klaus P
- Ly, Justin
- Merchant, Mark
- Orr, Christine
- Plise, Emile
- Robarge, Kirk
- Martini, Jean F
- Kassees, Robert
- Aoyama, Ron G
- Ramaiya, Atulkumar
- Johnston, Stuart H
Producer: 20120823
In:
Drug metabolism and disposition: the biological fate of chemicals vol. 40
Availability: No items available.
|
|
2.
|
Bridging the gap between preclinical and clinical studies using pharmacokinetic-pharmacodynamic modeling: an analysis of GDC-0973, a MEK inhibitor. [electronic resource] by
- Wong, Harvey
- Vernillet, Laurent
- Peterson, Amy
- Ware, Joseph A
- Lee, Lillian
- Martini, Jean-Francois
- Yu, Peiwen
- Li, Congfen
- Del Rosario, Geoffrey
- Choo, Edna F
- Hoeflich, Klaus P
- Shi, Yongchang
- Aftab, Blake T
- Aoyama, Ron
- Lam, Sanh Tan
- Belvin, Marcia
- Prescott, John
Producer: 20120815
In:
Clinical cancer research : an official journal of the American Association for Cancer Research vol. 18
Availability: No items available.
|
|
3.
|
Discovery of potent and selective inhibitors of calmodulin-dependent kinase II (CaMKII). [electronic resource] by
- Koltun, Dmitry O
- Parkhill, Eric Q
- Kalla, Rao
- Perry, Thao D
- Elzein, Elfatih
- Li, Xiaofen
- Simonovich, Scott P
- Ziebenhaus, Christopher
- Hansen, Timothy R
- Marchand, Bruno
- Hung, WaiLok K
- Lagpacan, Leanna
- Hung, Magdeleine
- Aoyama, Ron G
- Murray, Bernard P
- Perry, Jason K
- Somoza, John R
- Villaseñor, Armando G
- Pagratis, Nikos
- Zablocki, Jeff A
Producer: 20190530
In:
Bioorganic & medicinal chemistry letters vol. 28
Availability: No items available.
|
|
4.
|
Discovery and characterization of an inhibitor of glucosylceramide synthase. [electronic resource] by
- Richards, Steven
- Larson, Christopher J
- Koltun, Elena S
- Hanel, Art
- Chan, Vicky
- Nachtigall, Jason
- Harrison, Amanda
- Aay, Naing
- Du, Hongwang
- Arcalas, Arlyn
- Galan, Adam
- Zhang, Jeff
- Zhang, Wentao
- Won, Kwang-Ai
- Tam, Danny
- Qian, Fawn
- Wang, Tao
- Finn, Patricia
- Ogilvie, Kathy
- Rosen, Jon
- Aoyama, Ron
- Plonowski, Artur
- Cancilla, Belinda
- Bentzien, Frauke
- Yakes, Michael
- Mohan, Raju
- Lamb, Peter
- Nuss, John
- Kearney, Patrick
Producer: 20120912
In:
Journal of medicinal chemistry vol. 55
Availability: No items available.
|
|
5.
|
Discovery of a novel class of highly potent, selective, ATP-competitive, and orally bioavailable inhibitors of the mammalian target of rapamycin (mTOR). [electronic resource] by
- Takeuchi, Craig S
- Kim, Byung Gyu
- Blazey, Charles M
- Ma, Sunghoon
- Johnson, Henry W B
- Anand, Neel K
- Arcalas, Arlyn
- Baik, Tae Gon
- Buhr, Chris A
- Cannoy, Jonah
- Epshteyn, Sergey
- Joshi, Anagha
- Lara, Katherine
- Lee, Matthew S
- Wang, Longcheng
- Leahy, James W
- Nuss, John M
- Aay, Naing
- Aoyama, Ron
- Foster, Paul
- Lee, Jae
- Lehoux, Isabelle
- Munagala, Narsimha
- Plonowski, Arthur
- Rajan, Sharmila
- Woolfrey, John
- Yamaguchi, Kyoko
- Lamb, Peter
- Miller, Nicole
Producer: 20130523
In:
Journal of medicinal chemistry vol. 56
Availability: No items available.
|
|
6.
|
SAR and in vivo evaluation of 4-aryl-2-aminoalkylpyrimidines as potent and selective Janus kinase 2 (JAK2) inhibitors. [electronic resource] by
- Forsyth, Timothy
- Kearney, Patrick C
- Kim, Byung Gyu
- Johnson, Henry W B
- Aay, Naing
- Arcalas, Arlyn
- Brown, David S
- Chan, Vicky
- Chen, Jeff
- Du, Hongwang
- Epshteyn, Sergey
- Galan, Adam A
- Huynh, Tai P
- Ibrahim, Mohamed A
- Kane, Brian
- Koltun, Elena S
- Mann, Grace
- Meyr, Lisa E
- Lee, Matthew S
- Lewis, Gary L
- Noguchi, Robin T
- Pack, Michael
- Ridgway, Brian H
- Shi, Xian
- Takeuchi, Craig S
- Zu, Peiwen
- Leahy, James W
- Nuss, John M
- Aoyama, Ron
- Engst, Stefan
- Gendreau, Steven B
- Kassees, Robert
- Li, Jia
- Lin, Shwu-Hwa
- Martini, Jean-Francois
- Stout, Thomas
- Tong, Philip
- Woolfrey, John
- Zhang, Wentao
- Yu, Peiwen
Producer: 20130520
In:
Bioorganic & medicinal chemistry letters vol. 22
Availability: No items available.
|