Assay Conditions Influence Affinities of Rat Organic Cation Transporter 1: Analysis of Mutagenesis in the Modeled Outward-Facing Cleft by Measuring Effects of Substrates and Inhibitors on Initial Uptake. [electronic resource]
Producer: 20190411Description: 402-415 p. digitalISSN:- 1521-0111
- 1-Methyl-4-phenylpyridinium -- metabolism
- Animals
- Catecholamine Plasma Membrane Transport Proteins -- antagonists & inhibitors
- Dose-Response Relationship, Drug
- Female
- HEK293 Cells
- Humans
- Mutagenesis -- drug effects
- Quaternary Ammonium Compounds -- metabolism
- Rats
- Substrate Specificity -- drug effects
- Xenopus laevis
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't
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