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A combined spectroscopic and crystallographic approach to probing drug-human serum albumin interactions. [electronic resource] by
- Buttar, David
- Colclough, Nicola
- Gerhardt, Stefan
- MacFaul, Philip A
- Phillips, Scott D
- Plowright, Alleyn
- Whittamore, Paul
- Tam, Kin
- Maskos, Klaus
- Steinbacher, Stefan
- Steuber, Holger
Producer: 20110209
In:
Bioorganic & medicinal chemistry vol. 18
Availability: No items available.
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Optimisation of pharmacokinetic properties in a neutral series of 11β-HSD1 inhibitors. [electronic resource] by
- Scott, James S
- Gill, Adrian L
- Godfrey, Linda
- Groombridge, Sam D
- Rees, Amanda
- Revill, John
- Schofield, Paul
- Sörme, Pernilla
- Stocker, Andrew
- Swales, John G
- Whittamore, Paul R O
Producer: 20130320
In:
Bioorganic & medicinal chemistry letters vol. 22
Availability: No items available.
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Discovery of a series of indan carboxylic acid glycogen phosphorylase inhibitors. [electronic resource] by
- Bennett, Stuart N L
- Campbell, Andrew D
- Hancock, Andrew
- Johnstone, Craig
- Kenny, Peter W
- Pickup, Adrian
- Plowright, Alleyn T
- Selmi, Nidhal
- Simpson, Iain
- Stocker, Andy
- Whalley, David P
- Whittamore, Paul R O
Producer: 20100913
In:
Bioorganic & medicinal chemistry letters vol. 20
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6.
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Novel acidic 11β-hydroxysteroid dehydrogenase type 1 (11β-HSD1) inhibitor with reduced acyl glucuronide liability: the discovery of 4-[4-(2-adamantylcarbamoyl)-5-tert-butyl-pyrazol-1-yl]benzoic acid (AZD8329). [electronic resource] by
- Scott, James S
- deSchoolmeester, Joanne
- Kilgour, Elaine
- Mayers, Rachel M
- Packer, Martin J
- Hargreaves, David
- Gerhardt, Stefan
- Ogg, Derek J
- Rees, Amanda
- Selmi, Nidhal
- Stocker, Andrew
- Swales, John G
- Whittamore, Paul R O
Producer: 20130205
In:
Journal of medicinal chemistry vol. 55
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Discovery of a potent, selective, and orally bioavailable acidic 11β-hydroxysteroid dehydrogenase type 1 (11β-HSD1) inhibitor: discovery of 2-[(3S)-1-[5-(cyclohexylcarbamoyl)-6-propylsulfanylpyridin-2-yl]-3-piperidyl]acetic acid (AZD4017). [electronic resource] by
- Scott, James S
- Bowker, Suzanne S
- Deschoolmeester, Joanne
- Gerhardt, Stefan
- Hargreaves, David
- Kilgour, Elaine
- Lloyd, Adele
- Mayers, Rachel M
- McCoull, William
- Newcombe, Nicholas J
- Ogg, Derek
- Packer, Martin J
- Rees, Amanda
- Revill, John
- Schofield, Paul
- Selmi, Nidhal
- Swales, John G
- Whittamore, Paul R O
Producer: 20120907
In:
Journal of medicinal chemistry vol. 55
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Making medicinal chemistry more effective--application of Lean Sigma to improve processes, speed and quality. [electronic resource] by
- Andersson, Shalini
- Armstrong, Alan
- Björe, Annika
- Bowker, Sue
- Chapman, Steve
- Davies, Rob
- Donald, Craig
- Egner, Bryan
- Elebring, Thomas
- Holmqvist, Sara
- Inghardt, Tord
- Johannesson, Petra
- Johansson, Magnus
- Johnstone, Craig
- Kemmitt, Paul
- Kihlberg, Jan
- Korsgren, Pernilla
- Lemurell, Malin
- Moore, Jane
- Pettersson, Jonas A
- Pointon, Helen
- Pontén, Fritiof
- Schofield, Paul
- Selmi, Nidhal
- Whittamore, Paul
Producer: 20110803
In:
Drug discovery today vol. 14
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Novel thienopyrrole glycogen phosphorylase inhibitors: synthesis, in vitro SAR and crystallographic studies. [electronic resource] by
- Whittamore, Paul R O
- Addie, Matthew S
- Bennett, Stuart N L
- Birch, Alan M
- Butters, Michael
- Godfrey, Linda
- Kenny, Peter W
- Morley, Andrew D
- Murray, Paul M
- Oikonomakos, Nikos G
- Otterbein, Ludovic R
- Pannifer, Andrew D
- Parker, Jeremy S
- Readman, Kristy
- Siedlecki, Pawel S
- Schofield, Paul
- Stocker, Andy
- Taylor, Melvyn J
- Townsend, Linda A
- Whalley, David P
- Whitehouse, Jennifer
Producer: 20061222
In:
Bioorganic & medicinal chemistry letters vol. 16
Availability: No items available.
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