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Fragment-based discovery of potent inhibitors of the anti-apoptotic MCL-1 protein. [electronic resource] by
- Petros, Andrew M
- Swann, Steven L
- Song, Danying
- Swinger, Kerren
- Park, Chang
- Zhang, Haichao
- Wendt, Michael D
- Kunzer, Aaron R
- Souers, Andrew J
- Sun, Chaohong
Producer: 20141104
In:
Bioorganic & medicinal chemistry letters vol. 24
Availability: No items available.
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MCL-1 Is a Key Determinant of Breast Cancer Cell Survival: Validation of MCL-1 Dependency Utilizing a Highly Selective Small Molecule Inhibitor. [electronic resource] by
- Xiao, Yu
- Nimmer, Paul
- Sheppard, George S
- Bruncko, Milan
- Hessler, Paul
- Lu, Xin
- Roberts-Rapp, Lisa
- Pappano, William N
- Elmore, Steven W
- Souers, Andrew J
- Leverson, Joel D
- Phillips, Darren C
Producer: 20160505
In:
Molecular cancer therapeutics vol. 14
Availability: No items available.
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15.
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In vivo efficacy of acyl CoA: diacylglycerol acyltransferase (DGAT) 1 inhibition in rodent models of postprandial hyperlipidemia. [electronic resource] by
- King, Andrew J
- Segreti, Jason A
- Larson, Kelly J
- Souers, Andrew J
- Kym, Philip R
- Reilly, Regina M
- Collins, Christine A
- Voorbach, Martin J
- Zhao, Gang
- Mittelstadt, Scott W
- Cox, Bryan F
Producer: 20100907
In:
European journal of pharmacology vol. 637
Availability: No items available.
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Synthesis and evaluation of 2-amino-8-alkoxy quinolines as MCHr1 antagonists. Part 2. [electronic resource] by
- Vasudevan, Anil
- Wodka, Dariusz
- Verzal, Mary K
- Souers, Andrew J
- Gao, Ju
- Brodjian, Sevan
- Fry, Dennis
- Dayton, Brian
- Marsh, Kennan C
- Hernandez, Lisa E
- Ogiela, Christopher A
- Collins, Christine A
- Kym, Philip R
Producer: 20050324
In:
Bioorganic & medicinal chemistry letters vol. 14
Availability: No items available.
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Synthesis and evaluation of 2-amino-8-alkoxy quinolines as MCHr1 antagonists. Part 3. [electronic resource] by
- Souers, Andrew J
- Wodka, Dariusz
- Gao, Ju
- Lewis, Jared C
- Vasudevan, Anil
- Brodjian, Sevan
- Dayton, Brian
- Ogiela, Christopher A
- Fry, Dennis
- Hernandez, Lisa E
- Marsh, Kennan C
- Collins, Christine A
- Kym, Philip R
Producer: 20050324
In:
Bioorganic & medicinal chemistry letters vol. 14
Availability: No items available.
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18.
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Synthesis and evaluation of 2-amino-8-alkoxy quinolines as MCHr1 antagonists. Part 1. [electronic resource] by
- Souers, Andrew J
- Wodka, Dariusz
- Gao, Ju
- Lewis, Jared C
- Vasudevan, Anil
- Gentles, Robert
- Brodjian, Sevan
- Dayton, Brian
- Ogiela, Christopher A
- Fry, Dennis
- Hernandez, Lisa E
- Marsh, Kennan C
- Collins, Christine A
- Kym, Philip R
Producer: 20050324
In:
Bioorganic & medicinal chemistry letters vol. 14
Availability: No items available.
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19.
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Clearance of systemic hematologic tumors by venetoclax (Abt-199) and navitoclax. [electronic resource] by
- Ackler, Scott
- Oleksijew, Anatol
- Chen, Jun
- Chyla, Brenda J
- Clarin, Jerry
- Foster, Kelly
- McGonigal, Thomas
- Mishra, Sasmita
- Schlessinger, Sally
- Smith, Morey L
- Tahir, Stephen K
- Leverson, Joel D
- Souers, Andrew J
- Boghaert, Erwin R
- Hickson, Jonathan
Producer: 20151030
In:
Pharmacology research & perspectives vol. 3
Availability: No items available.
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Identification of 2-(4-benzyloxyphenyl)-N- [1-(2-pyrrolidin-1-yl-ethyl)-1H-indazol-6-yl]acetamide, an orally efficacious melanin-concentrating hormone receptor 1 antagonist for the treatment of obesity. [electronic resource] by
- Souers, Andrew J
- Gao, Ju
- Brune, Michael
- Bush, Eugene
- Wodka, Dariusz
- Vasudevan, Anil
- Judd, Andrew S
- Mulhern, Mathew
- Brodjian, Sevan
- Dayton, Brian
- Shapiro, Robin
- Hernandez, Lisa E
- Marsh, Kennan C
- Sham, Hing L
- Collins, Christine A
- Kym, Philip R
Producer: 20050411
In:
Journal of medicinal chemistry vol. 48
Availability: No items available.
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