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Synthesis and SAR studies of imidazo-[1,2-a]-pyrazine Aurora kinase inhibitors with improved off-target kinase selectivity. [electronic resource] by
- Voss, Matthew E
- Rainka, Matthew P
- Fleming, Mike
- Peterson, Lisa H
- Belanger, David B
- Siddiqui, M Arshad
- Hruza, Alan
- Voigt, Johannes
- Gray, Kimberly
- Basso, Andrea D
Producer: 20120910
In:
Bioorganic & medicinal chemistry letters vol. 22
Availability: No items available.
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7.
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Discovery of a highly potent orally bioavailable imidazo-[1, 2-a]pyrazine Aurora inhibitor. [electronic resource] by
- Yu, Tao
- Zhang, Yonglian
- Kerekes, Angela D
- Tagat, Jayaram R
- Doll, Ronald J
- Xiao, Yushi
- Esposite, Sara
- Hruza, Alan
- Belanger, David B
- Voss, Matthew
- Rainka, Matthew P
- Basso, Andrea
- Liu, Ming
- Liang, Lianzhu
- Sui, Ning
- Prelusky, Daniel
- Rindgen, Diane
- Zhang, Likang
Producer: 20190227
In:
Bioorganic & medicinal chemistry letters vol. 28
Availability: No items available.
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8.
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Heterobiaryl purine derivatives as potent antiproliferative agents: inhibitors of cyclin dependent kinases. Part II. [electronic resource] by
- Trova, Michael P
- Barnes, Keith D
- Alicea, Luis
- Benanti, Travis
- Bielaska, Mark
- Bilotta, Joseph
- Bliss, Brian
- Duong, Thuy Nguyen
- Haydar, Simon
- Herr, R Jason
- Hui, Yu
- Johnson, Matthew
- Lehman, John M
- Peace, Denise
- Rainka, Matthew
- Snider, Patricia
- Salamone, Susan
- Tregay, Steven
- Zheng, Xiaozhang
- Friedrich, Thomas D
Producer: 20100119
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
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Discovery of orally bioavailable imidazo[1,2-a]pyrazine-based Aurora kinase inhibitors. [electronic resource] by
- Belanger, David B
- Williams, Michael J
- Curran, Patrick J
- Mandal, Amit K
- Meng, Zhaoyang
- Rainka, Matthew P
- Yu, Tao
- Shih, Neng-Yang
- Siddiqui, M Arshad
- Liu, Ming
- Tevar, Seema
- Lee, Suining
- Liang, Lianzhu
- Gray, Kimberly
- Yaremko, Bohdan
- Jones, Jennifer
- Smith, Elizabeth B
- Prelusky, Dan B
- Basso, Andrea D
Producer: 20110329
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
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