Results
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Thermodynamic and kinetic characterization of hydroxyethylamine β-secretase-1 inhibitors. [electronic resource] by
- Mondal, Kalyani
- Regnstrom, Karin
- Morishige, Winse
- Barbour, Robin
- Probst, Gary
- Xu, Ying-Zi
- Artis, Dean R
- Yao, Nanhua
- Beroza, Paul
- Bova, Michael P
Producer: 20140117
In:
Biochemical and biophysical research communications vol. 441
Availability: No items available.
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5.
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Triazolopyridazine LRRK2 kinase inhibitors. [electronic resource] by
- Franzini, Maurizio
- Ye, Xiaocong M
- Adler, Marc
- Aubele, Danielle L
- Garofalo, Albert W
- Gauby, Shawn
- Goldbach, Erich
- Probst, Gary D
- Quinn, Kevin P
- Santiago, Pam
- Sham, Hing L
- Tam, Danny
- Truong, Anh
- Ren, Zhao
Producer: 20130930
In:
Bioorganic & medicinal chemistry letters vol. 23
Availability: No items available.
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6.
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Novel cinnoline-based inhibitors of LRRK2 kinase activity. [electronic resource] by
- Garofalo, Albert W
- Adler, Marc
- Aubele, Danielle L
- Bowers, Simeon
- Franzini, Maurizio
- Goldbach, Erich
- Lorentzen, Colin
- Neitz, R Jeffrey
- Probst, Gary D
- Quinn, Kevin P
- Santiago, Pam
- Sham, Hing L
- Tam, Danny
- Truong, Anh P
- Ye, Xiaocong M
- Ren, Zhao
Producer: 20130528
In:
Bioorganic & medicinal chemistry letters vol. 23
Availability: No items available.
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7.
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N-Bridged bicyclic sulfonamides as inhibitors of gamma-secretase. [electronic resource] by
- Bowers, Simeon
- Probst, Gary D
- Truong, Anh P
- Hom, Roy K
- Konradi, Andrei W
- Sham, Hing L
- Garofalo, Albert W
- Wong, Karina
- Goldbach, Erich
- Quinn, Kevin P
- Sauer, John-Michael
- Wallace, William
- Nguyen, Lan
- Hemphill, Susanna S
- Bova, Michael P
- Basi, Guriqbal S
Producer: 20100209
In:
Bioorganic & medicinal chemistry letters vol. 19
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8.
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Discovery of 4-alkylamino-7-aryl-3-cyanoquinoline LRRK2 kinase inhibitors. [electronic resource] by
- Garofalo, Albert W
- Adler, Marc
- Aubele, Danielle L
- Brigham, Elizabeth F
- Chian, David
- Franzini, Maurizio
- Goldbach, Erich
- Kwong, Grace T
- Motter, Ruth
- Probst, Gary D
- Quinn, Kevin P
- Ruslim, Lany
- Sham, Hing L
- Tam, Danny
- Tanaka, Pearl
- Truong, Anh P
- Ye, Xiaocong M
- Ren, Zhao
Producer: 20130930
In:
Bioorganic & medicinal chemistry letters vol. 23
Availability: No items available.
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Structure-based design of novel dihydroisoquinoline BACE-1 inhibitors that do not engage the catalytic aspartates. [electronic resource] by
- Bowers, Simeon
- Xu, Ying-zi
- Yuan, Shendong
- Probst, Gary D
- Hom, Roy K
- Chan, Wayman
- Konradi, Andrei W
- Sham, Hing L
- Zhu, Yong L
- Beroza, Paul
- Pan, Hu
- Brecht, Eric
- Yao, Nanhua
- Lougheed, Julie
- Tam, Danny
- Ren, Zhao
- Ruslim, Lany
- Bova, Michael P
- Artis, Dean R
Producer: 20130930
In:
Bioorganic & medicinal chemistry letters vol. 23
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10.
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Antibody-Drug Conjugates (ADCs) Derived from Interchain Cysteine Cross-Linking Demonstrate Improved Homogeneity and Other Pharmacological Properties over Conventional Heterogeneous ADCs. [electronic resource] by
- Behrens, Christopher R
- Ha, Edward H
- Chinn, Lawrence L
- Bowers, Simeon
- Probst, Gary
- Fitch-Bruhns, Maureen
- Monteon, Jorge
- Valdiosera, Amanda
- Bermudez, Abel
- Liao-Chan, Sindy
- Wong, Tiffany
- Melnick, Jonathan
- Theunissen, Jan-Willem
- Flory, Mark R
- Houser, Derrick
- Venstrom, Kristy
- Levashova, Zoia
- Sauer, Paul
- Migone, Thi-Sau
- van der Horst, Edward H
- Halcomb, Randall L
- Jackson, David Y
Producer: 20160915
In:
Molecular pharmaceutics vol. 12
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11.
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Design and synthesis of a novel, orally active, brain penetrant, tri-substituted thiophene based JNK inhibitor. [electronic resource] by
- Bowers, Simeon
- Truong, Anh P
- Neitz, R Jeffrey
- Neitzel, Martin
- Probst, Gary D
- Hom, Roy K
- Peterson, Brian
- Galemmo, Robert A
- Konradi, Andrei W
- Sham, Hing L
- Tóth, Gergley
- Pan, Hu
- Yao, Nanhua
- Artis, Dean R
- Brigham, Elizabeth F
- Quinn, Kevin P
- Sauer, John-Michael
- Powell, Kyle
- Ruslim, Lany
- Ren, Zhao
- Bard, Frédérique
- Yednock, Ted A
- Griswold-Prenner, Irene
Producer: 20110705
In:
Bioorganic & medicinal chemistry letters vol. 21
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12.
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Design and synthesis of disubstituted thiophene and thiazole based inhibitors of JNK. [electronic resource] by
- Hom, Roy K
- Bowers, Simeon
- Sealy, Jennifer M
- Truong, Anh P
- Probst, Gary D
- Neitzel, Martin L
- Neitz, R Jeffrey
- Fang, Larry
- Brogley, Louis
- Wu, Jing
- Konradi, Andrei W
- Sham, Hing L
- Tóth, Gergely
- Pan, Hu
- Yao, Nanhua
- Artis, Dean R
- Quinn, Kevin
- Sauer, John-Michael
- Powell, Kyle
- Ren, Zhao
- Bard, Frédérique
- Yednock, Ted A
- Griswold-Prenner, Irene
Producer: 20110314
In:
Bioorganic & medicinal chemistry letters vol. 20
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13.
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Design, synthesis and structure-activity relationship of novel [3.3.1] bicyclic sulfonamide-pyrazoles as potent γ-secretase inhibitors. [electronic resource] by
- Aubele, Danielle L
- Truong, Anh P
- Dressen, Darren B
- Probst, Gary D
- Bowers, Simeon
- Mattson, Matthew N
- Semko, Chris M
- Sun, Minghua
- Garofalo, Albert W
- Konradi, Andrei W
- Sham, Hing L
- Zmolek, Wes
- Wong, Karina
- Goldbach, Erich
- Quinn, Kevin P
- Sauer, John-Michael
- Brigham, Elizabeth F
- Wallace, William
- Nguyen, Lan
- Bova, Michael P
- Hemphill, Susanna S
- Basi, Guriqbal
Producer: 20120416
In:
Bioorganic & medicinal chemistry letters vol. 21
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14.
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Discovery of a novel [3.2.1] benzo fused bicyclic sulfonamide-pyrazoles as potent, selective and efficacious γ-secretase inhibitors. [electronic resource] by
- Ye, Xiaocong M
- Konradi, Andrei W
- Sun, Minghua
- Yuan, Shendong
- Aubele, Danielle L
- Dappen, Michael
- Dressen, Darren
- Garofalo, Albert W
- Jagodzinski, Jacek J
- Latimer, Lee
- Probst, Gary D
- Sham, Hing L
- Wone, David
- Xu, Ying-zi
- Ness, Daniel
- Brigham, Elizabeth
- Kwong, Grace T
- Willtis, Chris
- Tonn, George
- Goldbach, Erich
- Quinn, Kevin P
- Zhang, Hongbin H
- Sauer, John-Michael
- Bova, Michael
- Basi, Guriqbal S
Producer: 20131031
In:
Bioorganic & medicinal chemistry letters vol. 23
Availability: No items available.
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15.
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Design and synthesis of cell potent BACE-1 inhibitors: structure-activity relationship of P1' substituents. [electronic resource] by
- Sealy, Jennifer M
- Truong, Anh P
- Tso, Luke
- Probst, Gary D
- Aquino, Jose
- Hom, Roy K
- Jagodzinska, Barbara M
- Dressen, Darren
- Wone, David W G
- Brogley, Louis
- John, Varghese
- Tung, Jay S
- Pleiss, Michael A
- Tucker, John A
- Konradi, Andrei W
- Dappen, Michael S
- Toth, Gergely
- Pan, Hu
- Ruslim, Lany
- Miller, Jim
- Bova, Michael P
- Sinha, Sukanto
- Quinn, Kevin P
- Sauer, John-Michael
Producer: 20100127
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
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16.
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Discovery of betrixaban (PRT054021), N-(5-chloropyridin-2-yl)-2-(4-(N,N-dimethylcarbamimidoyl)benzamido)-5-methoxybenzamide, a highly potent, selective, and orally efficacious factor Xa inhibitor. [electronic resource] by
- Zhang, Penglie
- Huang, Wenrong
- Wang, Lingyan
- Bao, Liang
- Jia, Zhaozhong J
- Bauer, Shawn M
- Goldman, Erick A
- Probst, Gary D
- Song, Yonghong
- Su, Ting
- Fan, Jingmei
- Wu, Yanhong
- Li, Wenhao
- Woolfrey, John
- Sinha, Uma
- Wong, Paul W
- Edwards, Susan T
- Arfsten, Ann E
- Clizbe, Lane A
- Kanter, James
- Pandey, Anjali
- Park, Gary
- Hutchaleelaha, Athiwat
- Lambing, Joseph L
- Hollenbach, Stanley J
- Scarborough, Robert M
- Zhu, Bing-Yan
Producer: 20090826
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
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17.
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Improving the permeability of the hydroxyethylamine BACE-1 inhibitors: structure-activity relationship of P2' substituents. [electronic resource] by
- Truong, Anh P
- Probst, Gary D
- Aquino, Jose
- Fang, Larry
- Brogley, Louis
- Sealy, Jennifer M
- Hom, Roy K
- Tucker, John A
- John, Varghese
- Tung, Jay S
- Pleiss, Michael A
- Konradi, Andrei W
- Sham, Hing L
- Dappen, Michael S
- Tóth, Gergley
- Yao, Nanhua
- Brecht, Eric
- Pan, Hu
- Artis, Dean R
- Ruslim, Lany
- Bova, Michael P
- Sinha, Sukanto
- Yednock, Ted A
- Zmolek, Wes
- Quinn, Kevin P
- Sauer, John-Michael
Producer: 20101110
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
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18.
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Design and synthesis of hydroxyethylamine (HEA) BACE-1 inhibitors: prime side chromane-containing inhibitors. [electronic resource] by
- Ng, Raymond A
- Sun, Minghua
- Bowers, Simeon
- Hom, Roy K
- Probst, Gary D
- John, Varghese
- Fang, Lawrence Y
- Maillard, Michel
- Gailunas, Andrea
- Brogley, Louis
- Neitz, R Jeffrey
- Tung, Jay S
- Pleiss, Michael A
- Konradi, Andrei W
- Sham, Hing L
- Dappen, Michael S
- Adler, Marc
- Yao, Nanhua
- Zmolek, Wes
- Nakamura, David
- Quinn, Kevin P
- Sauer, John-Michael
- Bova, Michael P
- Ruslim, Lany
- Artis, Dean R
- Yednock, Ted A
Producer: 20140130
In:
Bioorganic & medicinal chemistry letters vol. 23
Availability: No items available.
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19.
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Design, synthesis, and structure-activity relationship of novel orally efficacious pyrazole/sulfonamide based dihydroquinoline gamma-secretase inhibitors. [electronic resource] by
- Truong, Anh P
- Aubele, Danielle L
- Probst, Gary D
- Neitzel, Martin L
- Semko, Chris M
- Bowers, Simeon
- Dressen, Darren
- Hom, Roy K
- Konradi, Andrei W
- Sham, Hing L
- Garofalo, Albert W
- Keim, Pamela S
- Wu, Jing
- Dappen, Michael S
- Wong, Karina
- Goldbach, Erich
- Quinn, Kevin P
- Sauer, John-Michael
- Brigham, Elizabeth F
- Wallace, William
- Nguyen, Lan
- Hemphill, Susanna S
- Bova, Michael P
- Bard, Frédérique
- Yednock, Ted A
- Basi, Guriqbal
Producer: 20091124
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
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20.
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Highly selective c-Jun N-terminal kinase (JNK) 2 and 3 inhibitors with in vitro CNS-like pharmacokinetic properties prevent neurodegeneration. [electronic resource] by
- Probst, Gary D
- Bowers, Simeon
- Sealy, Jennifer M
- Truong, Anh P
- Hom, Roy K
- Galemmo, Robert A
- Konradi, Andrei W
- Sham, Hing L
- Quincy, David A
- Pan, Hu
- Yao, Nanhua
- Lin, May
- Tóth, Gergley
- Artis, Dean R
- Zmolek, Wes
- Wong, Karina
- Qin, Ann
- Lorentzen, Colin
- Nakamura, David F
- Quinn, Kevin P
- Sauer, John-Michael
- Powell, Kyle
- Ruslim, Lany
- Wright, Sarah
- Chereau, David
- Ren, Zhao
- Anderson, John P
- Bard, Frédérique
- Yednock, Ted A
- Griswold-Prenner, Irene
Producer: 20110414
In:
Bioorganic & medicinal chemistry letters vol. 21
Availability: No items available.
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