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Functional and toxicological consequences of metabolic bioactivation of methapyrilene via thiophene S-oxidation: Induction of cell defence, apoptosis and hepatic necrosis. [electronic resource] by
- Mercer, Amy E
- Regan, Sophie L
- Hirst, Charlotte M
- Graham, Emma E
- Antoine, Daniel J
- Benson, Craig A
- Williams, Dominic P
- Foster, John
- Kenna, J Gerry
- Park, B Kevin
Producer: 20090918
In:
Toxicology and applied pharmacology vol. 239
Availability: No items available.
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Synthesis, in vitro and in vivo antimalarial assessment of sulfide, sulfone and vinyl amide-substituted 1,2,4-trioxanes prepared via thiol-olefin co-oxygenation (TOCO) of allylic alcohols. [electronic resource] by
- Amewu, Richard
- Gibbons, Peter
- Mukhtar, Amira
- Stachulski, Andrew V
- Ward, Stephen A
- Hall, Charlotte
- Rimmer, Karen
- Davies, Jill
- Vivas, Livia
- Bacsa, John
- Mercer, Amy E
- Nixon, Gemma
- Stocks, Paul A
- O'Neill, Paul M
Producer: 20100715
In:
Organic & biomolecular chemistry vol. 8
Availability: No items available.
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Antimalarial and antitumor evaluation of novel C-10 non-acetal dimers of 10beta-(2-hydroxyethyl)deoxoartemisinin. [electronic resource] by
- Jeyadevan, J Prince
- Bray, Patrick G
- Chadwick, James
- Mercer, Amy E
- Byrne, Aoife
- Ward, Stephen A
- Park, B Kevin
- Williams, Dominic P
- Cosstick, Rick
- Davies, Jill
- Higson, Adrian P
- Irving, Ed
- Posner, Gary H
- O'Neill, Paul M
Producer: 20040413
In:
Journal of medicinal chemistry vol. 47
Availability: No items available.
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Examination of the cytotoxic and embryotoxic potential and underlying mechanisms of next-generation synthetic trioxolane and tetraoxane antimalarials. [electronic resource] by
- Copple, Ian M
- Mercer, Amy E
- Firman, James
- Donegan, Gail
- Herpers, Bram
- Wong, Michael Hl
- Chadwick, James
- Bringela, Andreia D
- Cristiano, Maria L S
- van de Water, Bob
- Ward, Stephen A
- O'Neill, Paul M
- Park, B Kevin
Producer: 20130206
In:
Molecular medicine (Cambridge, Mass.) vol. 18
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11.
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Evidence for a common non-heme chelatable-iron-dependent activation mechanism for semisynthetic and synthetic endoperoxide antimalarial drugs. [electronic resource] by
- Stocks, Paul A
- Bray, Patrick G
- Barton, Victoria E
- Al-Helal, Mohammed
- Jones, Michael
- Araujo, Nuna C
- Gibbons, Peter
- Ward, Stephen A
- Hughes, Ruth H
- Biagini, Giancarlo A
- Davies, Jill
- Amewu, Richard
- Mercer, Amy E
- Ellis, Gemma
- O'Neill, Paul M
Producer: 20071024
In:
Angewandte Chemie (International ed. in English) vol. 46
Availability: No items available.
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12.
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Antitumour and antimalarial activity of artemisinin-acridine hybrids. [electronic resource] by
- Jones, Michael
- Mercer, Amy E
- Stocks, Paul A
- La Pensée, Louise J I
- Cosstick, Rick
- Park, B Kevin
- Kennedy, Miriam E
- Piantanida, Ivo
- Ward, Stephen A
- Davies, Jill
- Bray, Patrick G
- Rawe, Sarah L
- Baird, Jonathan
- Charidza, Tafadzwa
- Janneh, Omar
- O'Neill, Paul M
Producer: 20090615
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
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13.
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A tetraoxane-based antimalarial drug candidate that overcomes PfK13-C580Y dependent artemisinin resistance. [electronic resource] by
- O'Neill, Paul M
- Amewu, Richard K
- Charman, Susan A
- Sabbani, Sunil
- Gnädig, Nina F
- Straimer, Judith
- Fidock, David A
- Shore, Emma R
- Roberts, Natalie L
- Wong, Michael H-L
- Hong, W David
- Pidathala, Chandrakala
- Riley, Chris
- Murphy, Ben
- Aljayyoussi, Ghaith
- Gamo, Francisco Javier
- Sanz, Laura
- Rodrigues, Janneth
- Cortes, Carolina Gonzalez
- Herreros, Esperanza
- Angulo-Barturén, Iñigo
- Jiménez-Díaz, María Belén
- Bazaga, Santiago Ferrer
- Martínez-Martínez, María Santos
- Campo, Brice
- Sharma, Raman
- Ryan, Eileen
- Shackleford, David M
- Campbell, Simon
- Smith, Dennis A
- Wirjanata, Grennady
- Noviyanti, Rintis
- Price, Ric N
- Marfurt, Jutta
- Palmer, Michael J
- Copple, Ian M
- Mercer, Amy E
- Ruecker, Andrea
- Delves, Michael J
- Sinden, Robert E
- Siegl, Peter
- Davies, Jill
- Rochford, Rosemary
- Kocken, Clemens H M
- Zeeman, Anne-Marie
- Nixon, Gemma L
- Biagini, Giancarlo A
- Ward, Stephen A
Producer: 20181211
In:
Nature communications vol. 8
Availability: No items available.
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