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Proline-based hydroxamates targeting the zinc-dependent deacetylase LpxC: Synthesis, antibacterial properties, and docking studies. [electronic resource] by
- Kalinin, Dmitrii V
- Agoglitta, Oriana
- Van de Vyver, Hélène
- Melesina, Jelena
- Wagner, Stefan
- Riemann, Burkhard
- Schäfers, Michael
- Sippl, Wolfgang
- Löffler, Bettina
- Holl, Ralph
Producer: 20200220
In:
Bioorganic & medicinal chemistry vol. 27
Availability: No items available.
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10.
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Structure-Based Design, Synthesis, and Biological Evaluation of Triazole-Based smHDAC8 Inhibitors. [electronic resource] by
- Kalinin, Dmitrii V
- Jana, Sunit K
- Pfafenrot, Maxim
- Chakrabarti, Alokta
- Melesina, Jelena
- Shaik, Tajith B
- Lancelot, Julien
- Pierce, Raymond J
- Sippl, Wolfgang
- Romier, Christophe
- Jung, Manfred
- Holl, Ralph
Producer: 20210407
In:
ChemMedChem vol. 15
Availability: No items available.
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11.
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Characterization of Histone Deacetylase 8 (HDAC8) Selective Inhibition Reveals Specific Active Site Structural and Functional Determinants. [electronic resource] by
- Marek, Martin
- Shaik, Tajith B
- Heimburg, Tino
- Chakrabarti, Alokta
- Lancelot, Julien
- Ramos-Morales, Elizabeth
- Da Veiga, Cyrielle
- Kalinin, Dmitrii
- Melesina, Jelena
- Robaa, Dina
- Schmidtkunz, Karin
- Suzuki, Takayoshi
- Holl, Ralph
- Ennifar, Eric
- Pierce, Raymond J
- Jung, Manfred
- Sippl, Wolfgang
- Romier, Christophe
Producer: 20190930
In:
Journal of medicinal chemistry vol. 61
Availability: No items available.
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