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Synthesis and activity of analogues of the isoleucyl tRNA synthetase inhibitor SB-203207. [electronic resource] by
- Crasto, Curtis F
- Forrest, Andrew K
- Karoli, Tomislav
- March, Darren R
- Mensah, Lucy
- O'Hanlon, Peter J
- Nairn, Michael R
- Oldham, Mark D
- Yue, Weimin
- Banwell, Martin G
- Easton, Christopher J
Producer: 20040406
In:
Bioorganic & medicinal chemistry vol. 11
Availability: No items available.
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Optimisation of aryl substitution leading to potent methionyl tRNA synthetase inhibitors with excellent gram-positive antibacterial activity. [electronic resource] by
- Jarvest, Richard L
- Berge, John M
- Brown, Murray J
- Brown, Pamela
- Elder, John S
- Forrest, Andrew K
- Houge-Frydrych, C S V
- O'Hanlon, Peter J
- McNair, David J
- Rittenhouse, Stephen
- Sheppard, Robert J
Producer: 20031120
In:
Bioorganic & medicinal chemistry letters vol. 13
Availability: No items available.
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Design of Selective Benzoxazepin PI3Kδ Inhibitors Through Control of Dihedral Angles. [electronic resource] by
- Safina, Brian S
- Elliott, Richard L
- Forrest, Andrew K
- Heald, Robert A
- Murray, Jeremy M
- Nonomiya, Jim
- Pang, Jodie
- Salphati, Laurent
- Seward, Eileen M
- Staben, Steven T
- Ultsch, Mark
- Wei, Binqing
- Yang, Wenqian
- Sutherlin, Daniel P
Publication details: ACS medicinal chemistry letters Sep 2017
In:
ACS medicinal chemistry letters vol. 8
Availability: No items available.
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7.
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Definition of the heterocyclic pharmacophore of bacterial methionyl tRNA synthetase inhibitors: potent antibacterially active non-quinolone analogues. [electronic resource] by
- Jarvest, Richard L
- Armstrong, Sula A
- Berge, John M
- Brown, Pamela
- Elder, John S
- Brown, Murray J
- Copley, Royston C B
- Forrest, Andrew K
- Hamprecht, Dieter W
- O'Hanlon, Peter J
- Mitchell, Darren J
- Rittenhouse, Stephen
- Witty, David R
Producer: 20050412
In:
Bioorganic & medicinal chemistry letters vol. 14
Availability: No items available.
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Synthesis and properties of macrolones characterized by two ether bonds in the linker. [electronic resource] by
- Jakopović, Ivana Palej
- Kragol, Goran
- Forrest, Andrew K
- Frydrych, Catherine S V
- Stimac, Vlado
- Kapić, Samra
- Skugor, Maja Matanović
- Ilijas, Marina
- Paljetak, Hana Cipcić
- Jelić, Dubravko
- Holmes, David J
- Hickey, Deirdre M B
- Verbanac, Donatella
- Eraković Haber, Vesna
- Alihodzić, Sulejman
Producer: 20110208
In:
Bioorganic & medicinal chemistry vol. 18
Availability: No items available.
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Nanomolar inhibitors of Staphylococcus aureus methionyl tRNA synthetase with potent antibacterial activity against gram-positive pathogens. [electronic resource] by
- Jarvest, Richard L
- Berge, John M
- Berry, Valerie
- Boyd, Helen F
- Brown, Murray J
- Elder, John S
- Forrest, Andrew K
- Fosberry, Andrew P
- Gentry, Daniel R
- Hibbs, Martin J
- Jaworski, Deborah D
- O'Hanlon, Peter J
- Pope, Andrew J
- Rittenhouse, Stephen
- Sheppard, Robert J
- Slater-Radosti, Courtney
- Worby, Angela
Producer: 20020531
In:
Journal of medicinal chemistry vol. 45
Availability: No items available.
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