Results
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2.
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Assessment of the integrity of compounds stored in assay-ready plates using a kinase sentinel assay. [electronic resource] by
- Chen, Ada
- Zhao, Xiaoning
- Mercer, Laina
- Su, Cheng
- Zalameda, Leeanne
- Liu, Yichin
- Lembke, Amanda
- Eastwood, Heather
- Dang, Son
- Oung, Thim
- Xia, Xiaoyang
- Young, Stephen W
- Xiao, Shouhua
- McCarter, John D
Producer: 20140310
In:
Combinatorial chemistry & high throughput screening vol. 16
Availability: No items available.
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3.
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The MDM2 Inhibitor AMG 232 Demonstrates Robust Antitumor Efficacy and Potentiates the Activity of p53-Inducing Cytotoxic Agents. [electronic resource] by
- Canon, Jude
- Osgood, Tao
- Olson, Steven H
- Saiki, Anne Y
- Robertson, Rebecca
- Yu, Dongyin
- Eksterowicz, John
- Ye, Qiuping
- Jin, Lixia
- Chen, Ada
- Zhou, Jing
- Cordover, David
- Kaufman, Stephen
- Kendall, Richard
- Oliner, Jonathan D
- Coxon, Angela
- Radinsky, Robert
Producer: 20160316
In:
Molecular cancer therapeutics vol. 14
Availability: No items available.
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4.
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Optimization beyond AMG 232: discovery and SAR of sulfonamides on a piperidinone scaffold as potent inhibitors of the MDM2-p53 protein-protein interaction. [electronic resource] by
- Wang, Yingcai
- Zhu, Jiang
- Liu, Jiwen Jim
- Chen, Xiaoqi
- Mihalic, Jeff
- Deignan, Jeffrey
- Yu, Ming
- Sun, Daqing
- Kayser, Frank
- McGee, Lawrence R
- Lo, Mei-Chu
- Chen, Ada
- Zhou, Jing
- Ye, Qiuping
- Huang, Xin
- Long, Alexander M
- Yakowec, Peter
- Oliner, Jonathan D
- Olson, Steven H
- Medina, Julio C
Producer: 20150306
In:
Bioorganic & medicinal chemistry letters vol. 24
Availability: No items available.
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5.
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Preclinical evaluation of AMG 925, a FLT3/CDK4 dual kinase inhibitor for treating acute myeloid leukemia. [electronic resource] by
- Keegan, Kathleen
- Li, Cong
- Li, Zhihong
- Ma, Ji
- Ragains, Mark
- Coberly, Suzanne
- Hollenback, David
- Eksterowicz, John
- Liang, Lingming
- Weidner, Margaret
- Huard, Justin
- Wang, Xianghong
- Alba, Grace
- Orf, Jessica
- Lo, Mei-Chu
- Zhao, Sharon
- Ngo, Rachel
- Chen, Ada
- Liu, Lily
- Carlson, Timothy
- Quéva, Christophe
- McGee, Lawrence R
- Medina, Julio
- Kamb, Alexander
- Wickramasinghe, Dineli
- Dai, Kang
Producer: 20141209
In:
Molecular cancer therapeutics vol. 13
Availability: No items available.
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6.
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Discovery of Potent and Selective Non-Nucleotide Small Molecule Inhibitors of CD73. [electronic resource] by
- Beatty, Joel W
- Lindsey, Erick A
- Thomas-Tran, Rhiannon
- Debien, Laurent
- Mandal, Debashis
- Jeffrey, Jenna L
- Tran, Anh T
- Fournier, Jeremy
- Jacob, Steven D
- Yan, Xuelei
- Drew, Samuel L
- Ginn, Elaine
- Chen, Ada
- Pham, Amber T
- Zhao, Sharon
- Jin, Lixia
- Young, Stephen W
- Walker, Nigel P
- Leleti, Manmohan Reddy
- Moschütz, Susanne
- Sträter, Norbert
- Powers, Jay P
- Lawson, Kenneth V
Producer: 20200924
In:
Journal of medicinal chemistry vol. 63
Availability: No items available.
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7.
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AMG 580: a novel small molecule phosphodiesterase 10A (PDE10A) positron emission tomography tracer. [electronic resource] by
- Chen, Hang
- Lester-Zeiner, Dianna
- Shi, Jianxia
- Miller, Silke
- Glaus, Charlie
- Hu, Essa
- Chen, Ning
- Able, Jessica
- Biorn, Christopher
- Wong, Jamie
- Ma, Ji
- Michelsen, Klaus
- Hill Della Puppa, Geraldine
- Kazules, Tim
- Dou, Hui Hannah
- Talreja, Santosh
- Zhao, Xiaoning
- Chen, Ada
- Rumfelt, Shannon
- Kunz, Roxanne K
- Ye, Hu
- Thiel, Oliver R
- Williamson, Toni
- Davis, Carl
- Porter, Amy
- Immke, David
- Allen, Jennifer R
- Treanor, James
Producer: 20150708
In:
The Journal of pharmacology and experimental therapeutics vol. 352
Availability: No items available.
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8.
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Discovery of Potent and Simplified Piperidinone-Based Inhibitors of the MDM2-p53 Interaction. [electronic resource] by
- Yu, Ming
- Wang, Yingcai
- Zhu, Jiang
- Bartberger, Michael D
- Canon, Jude
- Chen, Ada
- Chow, David
- Eksterowicz, John
- Fox, Brian
- Fu, Jiasheng
- Gribble, Michael
- Huang, Xin
- Li, Zhihong
- Liu, Jiwen Jim
- Lo, Mei-Chu
- McMinn, Dustin
- Oliner, Jonathan D
- Osgood, Tao
- Rew, Yosup
- Saiki, Anne Y
- Shaffer, Paul
- Yan, Xuelei
- Ye, Qiuping
- Yu, Dongyin
- Zhao, Xiaoning
- Zhou, Jing
- Olson, Steven H
- Medina, Julio C
- Sun, Daqing
Producer: 20140822
In:
ACS medicinal chemistry letters vol. 5
Availability: No items available.
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9.
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Rational design and binding mode duality of MDM2-p53 inhibitors. [electronic resource] by
- Gonzalez-Lopez de Turiso, Felix
- Sun, Daqing
- Rew, Yosup
- Bartberger, Michael D
- Beck, Hilary P
- Canon, Jude
- Chen, Ada
- Chow, David
- Correll, Tiffany L
- Huang, Xin
- Julian, Lisa D
- Kayser, Frank
- Lo, Mei-Chu
- Long, Alexander M
- McMinn, Dustin
- Oliner, Jonathan D
- Osgood, Tao
- Powers, Jay P
- Saiki, Anne Y
- Schneider, Steve
- Shaffer, Paul
- Xiao, Shou-Hua
- Yakowec, Peter
- Yan, Xuelei
- Ye, Qiuping
- Yu, Dongyin
- Zhao, Xiaoning
- Zhou, Jing
- Medina, Julio C
- Olson, Steven H
Producer: 20130723
In:
Journal of medicinal chemistry vol. 56
Availability: No items available.
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10.
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Novel inhibitors of the MDM2-p53 interaction featuring hydrogen bond acceptors as carboxylic acid isosteres. [electronic resource] by
- Gonzalez, Ana Z
- Li, Zhihong
- Beck, Hilary P
- Canon, Jude
- Chen, Ada
- Chow, David
- Duquette, Jason
- Eksterowicz, John
- Fox, Brian M
- Fu, Jiasheng
- Huang, Xin
- Houze, Jonathan
- Jin, Lixia
- Li, Yihong
- Ling, Yun
- Lo, Mei-Chu
- Long, Alexander M
- McGee, Lawrence R
- McIntosh, Joel
- Oliner, Jonathan D
- Osgood, Tao
- Rew, Yosup
- Saiki, Anne Y
- Shaffer, Paul
- Wortman, Sarah
- Yakowec, Peter
- Yan, Xuelei
- Ye, Qiuping
- Yu, Dongyin
- Zhao, Xiaoning
- Zhou, Jing
- Olson, Steven H
- Sun, Daqing
- Medina, Julio C
Producer: 20140708
In:
Journal of medicinal chemistry vol. 57
Availability: No items available.
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11.
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Structure-based design of novel inhibitors of the MDM2-p53 interaction. [electronic resource] by
- Rew, Yosup
- Sun, Daqing
- Gonzalez-Lopez De Turiso, Felix
- Bartberger, Michael D
- Beck, Hilary P
- Canon, Jude
- Chen, Ada
- Chow, David
- Deignan, Jeffrey
- Fox, Brian M
- Gustin, Darin
- Huang, Xin
- Jiang, Min
- Jiao, Xianyun
- Jin, Lixia
- Kayser, Frank
- Kopecky, David J
- Li, Yihong
- Lo, Mei-Chu
- Long, Alexander M
- Michelsen, Klaus
- Oliner, Jonathan D
- Osgood, Tao
- Ragains, Mark
- Saiki, Anne Y
- Schneider, Steve
- Toteva, Maria
- Yakowec, Peter
- Yan, Xuelei
- Ye, Qiuping
- Yu, Dongyin
- Zhao, Xiaoning
- Zhou, Jing
- Medina, Julio C
- Olson, Steven H
Producer: 20121001
In:
Journal of medicinal chemistry vol. 55
Availability: No items available.
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12.
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Discovery of AM-7209, a potent and selective 4-amidobenzoic acid inhibitor of the MDM2-p53 interaction. [electronic resource] by
- Rew, Yosup
- Sun, Daqing
- Yan, Xuelei
- Beck, Hilary P
- Canon, Jude
- Chen, Ada
- Duquette, Jason
- Eksterowicz, John
- Fox, Brian M
- Fu, Jiasheng
- Gonzalez, Ana Z
- Houze, Jonathan
- Huang, Xin
- Jiang, Min
- Jin, Lixia
- Li, Yihong
- Li, Zhihong
- Ling, Yun
- Lo, Mei-Chu
- Long, Alexander M
- McGee, Lawrence R
- McIntosh, Joel
- Oliner, Jonathan D
- Osgood, Tao
- Saiki, Anne Y
- Shaffer, Paul
- Wang, Yu Chung
- Wortman, Sarah
- Yakowec, Peter
- Ye, Qiuping
- Yu, Dongyin
- Zhao, Xiaoning
- Zhou, Jing
- Medina, Julio C
- Olson, Steven H
Producer: 20150310
In:
Journal of medicinal chemistry vol. 57
Availability: No items available.
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13.
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Selective and potent morpholinone inhibitors of the MDM2-p53 protein-protein interaction. [electronic resource] by
- Gonzalez, Ana Z
- Eksterowicz, John
- Bartberger, Michael D
- Beck, Hilary P
- Canon, Jude
- Chen, Ada
- Chow, David
- Duquette, Jason
- Fox, Brian M
- Fu, Jiasheng
- Huang, Xin
- Houze, Jonathan B
- Jin, Lixia
- Li, Yihong
- Li, Zhihong
- Ling, Yun
- Lo, Mei-Chu
- Long, Alexander M
- McGee, Lawrence R
- McIntosh, Joel
- McMinn, Dustin L
- Oliner, Jonathan D
- Osgood, Tao
- Rew, Yosup
- Saiki, Anne Y
- Shaffer, Paul
- Wortman, Sarah
- Yakowec, Peter
- Yan, Xuelei
- Ye, Qiuping
- Yu, Dongyin
- Zhao, Xiaoning
- Zhou, Jing
- Olson, Steven H
- Medina, Julio C
- Sun, Daqing
Producer: 20140527
In:
Journal of medicinal chemistry vol. 57
Availability: No items available.
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14.
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Discovery of AMG 232, a potent, selective, and orally bioavailable MDM2-p53 inhibitor in clinical development. [electronic resource] by
- Sun, Daqing
- Li, Zhihong
- Rew, Yosup
- Gribble, Michael
- Bartberger, Michael D
- Beck, Hilary P
- Canon, Jude
- Chen, Ada
- Chen, Xiaoqi
- Chow, David
- Deignan, Jeffrey
- Duquette, Jason
- Eksterowicz, John
- Fisher, Benjamin
- Fox, Brian M
- Fu, Jiasheng
- Gonzalez, Ana Z
- Gonzalez-Lopez De Turiso, Felix
- Houze, Jonathan B
- Huang, Xin
- Jiang, Min
- Jin, Lixia
- Kayser, Frank
- Liu, Jiwen Jim
- Lo, Mei-Chu
- Long, Alexander M
- Lucas, Brian
- McGee, Lawrence R
- McIntosh, Joel
- Mihalic, Jeff
- Oliner, Jonathan D
- Osgood, Tao
- Peterson, Matthew L
- Roveto, Philip
- Saiki, Anne Y
- Shaffer, Paul
- Toteva, Maria
- Wang, Yingcai
- Wang, Yu Chung
- Wortman, Sarah
- Yakowec, Peter
- Yan, Xuelei
- Ye, Qiuping
- Yu, Dongyin
- Yu, Ming
- Zhao, Xiaoning
- Zhou, Jing
- Zhu, Jiang
- Olson, Steven H
- Medina, Julio C
Producer: 20140429
In:
Journal of medicinal chemistry vol. 57
Availability: No items available.
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15.
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Discovery of AMG 925, a FLT3 and CDK4 dual kinase inhibitor with preferential affinity for the activated state of FLT3. [electronic resource] by
- Li, Zhihong
- Wang, Xianghong
- Eksterowicz, John
- Gribble, Michael W
- Alba, Grace Q
- Ayres, Merrill
- Carlson, Timothy J
- Chen, Ada
- Chen, Xiaoqi
- Cho, Robert
- Connors, Richard V
- DeGraffenreid, Michael
- Deignan, Jeffrey T
- Duquette, Jason
- Fan, Pingchen
- Fisher, Benjamin
- Fu, Jiasheng
- Huard, Justin N
- Kaizerman, Jacob
- Keegan, Kathleen S
- Li, Cong
- Li, Kexue
- Li, Yunxiao
- Liang, Lingming
- Liu, Wen
- Lively, Sarah E
- Lo, Mei-Chu
- Ma, Ji
- McMinn, Dustin L
- Mihalic, Jeffrey T
- Modi, Kriti
- Ngo, Rachel
- Pattabiraman, Kanaka
- Piper, Derek E
- Queva, Christophe
- Ragains, Mark L
- Suchomel, Julia
- Thibault, Steve
- Walker, Nigel
- Wang, Xiaodong
- Wang, Zhulun
- Wanska, Malgorzata
- Wehn, Paul M
- Weidner, Margaret F
- Zhang, Alex J
- Zhao, Xiaoning
- Kamb, Alexander
- Wickramasinghe, Dineli
- Dai, Kang
- McGee, Lawrence R
- Medina, Julio C
Producer: 20140706
In:
Journal of medicinal chemistry vol. 57
Availability: No items available.
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