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Discovery of the imidazo[1,5-a][1,2,4]-triazolo[1,5-d][1,4]benzodiazepine scaffold as a novel, potent and selective GABA(A) alpha5 inverse agonist series. [electronic resource] by
- Achermann, Guido
- Ballard, Theresa M
- Blasco, Francesca
- Broutin, Pierre-Emmanuel
- Büttelmann, Bernd
- Fischer, Holger
- Graf, Martin
- Hernandez, Maria-Clemencia
- Hilty, Peter
- Knoflach, Frédéric
- Koblet, Andreas
- Knust, Henner
- Kurt, Anke
- Martin, James R
- Masciadri, Raffaello
- Porter, Richard H P
- Stadler, Heinz
- Thomas, Andrew W
- Trube, Gerhard
- Wichmann, Jürgen
Producer: 20091130
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
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96.
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Optimizing a Weakly Binding Fragment into a Potent RORγt Inverse Agonist with Efficacy in an in Vivo Inflammation Model. [electronic resource] by
- Carcache, David A
- Vulpetti, Anna
- Kallen, Joerg
- Mattes, Henri
- Orain, David
- Stringer, Rowan
- Vangrevelinghe, Eric
- Wolf, Romain M
- Kaupmann, Klemens
- Ottl, Johannes
- Dawson, Janet
- Cooke, Nigel G
- Hoegenauer, Klemens
- Billich, Andreas
- Wagner, Juergen
- Guntermann, Christine
- Hintermann, Samuel
Producer: 20190618
In:
Journal of medicinal chemistry vol. 61
Availability: No items available.
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