Results
|
81.
|
Investigating the spectrum of biological activity of ring-substituted salicylanilides and carbamoylphenylcarbamates. [electronic resource] by
- Otevrel, Jan
- Mandelova, Zuzana
- Pesko, Matus
- Guo, Jiahui
- Kralova, Katarina
- Sersen, Frantisek
- Vejsova, Marcela
- Kalinowski, Danuta S
- Kovacevic, Zaklina
- Coffey, Aidan
- Csollei, Jozef
- Richardson, Des R
- Jampilek, Josef
Producer: 20110211
In:
Molecules (Basel, Switzerland) vol. 15
Availability: No items available.
|
|
82.
|
Iron chelators of the di-2-pyridylketone thiosemicarbazone and 2-benzoylpyridine thiosemicarbazone series inhibit HIV-1 transcription: identification of novel cellular targets--iron, cyclin-dependent kinase (CDK) 2, and CDK9. [electronic resource] by
- Debebe, Zufan
- Ammosova, Tatyana
- Breuer, Denitra
- Lovejoy, David B
- Kalinowski, Danuta S
- Kumar, Krishna
- Jerebtsova, Marina
- Ray, Patricio
- Kashanchi, Fatah
- Gordeuk, Victor R
- Richardson, Des R
- Nekhai, Sergei
Producer: 20110113
In:
Molecular pharmacology vol. 79
Availability: No items available.
|
|
83.
|
Simultaneous determination of the novel thiosemicarbazone anti-cancer agent, Bp4eT, and its main phase I metabolites in plasma: application to a pilot pharmacokinetic study in rats. [electronic resource] by
- Stariat, Ján
- Suprunová, Vlasta
- Roh, Jaroslav
- Šesták, Vít
- Eisner, Tomáš
- Filipský, Tomáš
- Mladěnka, Přemysl
- Nobilis, Milan
- Šimůnek, Tomáš
- Klimeš, Jiří
- Kalinowski, Danuta S
- Richardson, Des R
- Kovaříková, Petra
Producer: 20141128
In:
Biomedical chromatography : BMC vol. 28
Availability: No items available.
|
|
84.
|
The iron chelator, deferasirox, as a novel strategy for cancer treatment: oral activity against human lung tumor xenografts and molecular mechanism of action. [electronic resource] by
- Lui, Goldie Y L
- Obeidy, Peyman
- Ford, Samuel J
- Tselepis, Chris
- Sharp, Danae M
- Jansson, Patric J
- Kalinowski, Danuta S
- Kovacevic, Zaklina
- Lovejoy, David B
- Richardson, Des R
Producer: 20130409
In:
Molecular pharmacology vol. 83
Availability: No items available.
|
|
85.
|
In Vitro Characterization of the Pharmacological Properties of the Anti-Cancer Chelator, Bp4eT, and Its Phase I Metabolites. [electronic resource] by
- Potůčková, Eliška
- Roh, Jaroslav
- Macháček, Miloslav
- Sahni, Sumit
- Stariat, Ján
- Šesták, Vít
- Jansová, Hana
- Hašková, Pavlína
- Jirkovská, Anna
- Vávrová, Kateřina
- Kovaříková, Petra
- Kalinowski, Danuta S
- Richardson, Des R
- Šimůnek, Tomáš
Producer: 20160706
In:
PloS one vol. 10
Availability: No items available.
|
|
86.
|
The novel iron chelator, 2-pyridylcarboxaldehyde 2-thiophenecarboxyl hydrazone, reduces catecholamine-mediated myocardial toxicity. [electronic resource] by
- Mladĕnka, Premysl
- Kalinowski, Danuta S
- Haskova, Pavlína
- Bobrovová, Zuzana
- Hrdina, Radomír
- Simůnek, Tomás
- Nachtigal, Petr
- Semecký, Vladimĺr
- Vávrová, Jaroslava
- Holeckova, Magdaléna
- Palicka, Vladimir
- Mazurová, Yvona
- Jansson, Patric J
- Richardson, Des R
Producer: 20090330
In:
Chemical research in toxicology vol. 22
Availability: No items available.
|
|
87.
|
The proto-oncogene c-Src and its downstream signaling pathways are inhibited by the metastasis suppressor, NDRG1. [electronic resource] by
- Liu, Wensheng
- Yue, Fei
- Zheng, Minhua
- Merlot, Angelica
- Bae, Dong-Hun
- Huang, Michael
- Lane, Darius
- Jansson, Patric
- Lui, Goldie Yuan Lam
- Richardson, Vera
- Sahni, Sumit
- Kalinowski, Danuta
- Kovacevic, Zaklina
- Richardson, Des R
Producer: 20160307
In:
Oncotarget vol. 6
Availability: No items available.
|
|
88.
|
Lysosomal membrane stability plays a major role in the cytotoxic activity of the anti-proliferative agent, di-2-pyridylketone 4,4-dimethyl-3-thiosemicarbazone (Dp44mT). [electronic resource] by
- Gutierrez, Elaine M
- Seebacher, Nicole A
- Arzuman, Laila
- Kovacevic, Zaklina
- Lane, Darius J R
- Richardson, Vera
- Merlot, Angelica M
- Lok, Hiu
- Kalinowski, Danuta S
- Sahni, Sumit
- Jansson, Patric J
- Richardson, Des R
Producer: 20160908
In:
Biochimica et biophysica acta vol. 1863
Availability: No items available.
|
|
89.
|
Exploring the anti-cancer activity of novel thiosemicarbazones generated through the combination of retro-fragments: dissection of critical structure-activity relationships. [electronic resource] by
- Serda, Maciej
- Kalinowski, Danuta S
- Rasko, Nathalie
- Potůčková, Eliška
- Mrozek-Wilczkiewicz, Anna
- Musiol, Robert
- Małecki, Jan G
- Sajewicz, Mieczysław
- Ratuszna, Alicja
- Muchowicz, Angelika
- Gołąb, Jakub
- Simůnek, Tomáš
- Richardson, Des R
- Polanski, Jaroslaw
Producer: 20151008
In:
PloS one vol. 9
Availability: No items available.
|
|
90.
|
Novel and potent anti-tumor and anti-metastatic di-2-pyridylketone thiosemicarbazones demonstrate marked differences in pharmacology between the first and second generation lead agents. [electronic resource] by
- Sestak, Vit
- Stariat, Jan
- Cermanova, Jolana
- Potuckova, Eliska
- Chladek, Jaroslav
- Roh, Jaroslav
- Bures, Jan
- Jansova, Hana
- Prusa, Petr
- Sterba, Martin
- Micuda, Stanislav
- Simunek, Tomas
- Kalinowski, Danuta S
- Richardson, Des R
- Kovarikova, Petra
Producer: 20161007
In:
Oncotarget vol. 6
Availability: No items available.
|
|
91.
|
Novel second-generation di-2-pyridylketone thiosemicarbazones show synergism with standard chemotherapeutics and demonstrate potent activity against lung cancer xenografts after oral and intravenous administration in vivo. [electronic resource] by
- Lovejoy, David B
- Sharp, Danae M
- Seebacher, Nicole
- Obeidy, Peyman
- Prichard, Thomas
- Stefani, Christian
- Basha, Maram T
- Sharpe, Philip C
- Jansson, Patric J
- Kalinowski, Danuta S
- Bernhardt, Paul V
- Richardson, Des R
Producer: 20121126
In:
Journal of medicinal chemistry vol. 55
Availability: No items available.
|
|
92.
|
Copper and conquer: copper complexes of di-2-pyridylketone thiosemicarbazones as novel anti-cancer therapeutics. [electronic resource] by
- Park, Kyung Chan
- Fouani, Leyla
- Jansson, Patric J
- Wooi, Danson
- Sahni, Sumit
- Lane, Darius J R
- Palanimuthu, Duraippandi
- Lok, Hiu Chuen
- Kovačević, Zaklina
- Huang, Michael L H
- Kalinowski, Danuta S
- Richardson, Des R
Producer: 20171211
In:
Metallomics : integrated biometal science vol. 8
Availability: No items available.
|
|
93.
|
Investigating the anti-proliferative activity of styrylazanaphthalenes and azanaphthalenediones. [electronic resource] by
- Mrozek-Wilczkiewicz, Anna
- Kalinowski, Danuta S
- Musiol, Robert
- Finster, Jacek
- Szurko, Agnieszka
- Serafin, Katarzyna
- Knas, Magdalena
- Kamalapuram, Sishir K
- Kovacevic, Zaklina
- Jampilek, Josef
- Ratuszna, Alicja
- Rzeszowska-Wolny, Joanna
- Richardson, Des R
- Polanski, Jaroslaw
Producer: 20100702
In:
Bioorganic & medicinal chemistry vol. 18
Availability: No items available.
|
|
94.
|
Potentiating the cellular targeting and anti-tumor activity of Dp44mT via binding to human serum albumin: two saturable mechanisms of Dp44mT uptake by cells. [electronic resource] by
- Merlot, Angelica M
- Sahni, Sumit
- Lane, Darius J R
- Fordham, Ashleigh M
- Pantarat, Namfon
- Hibbs, David E
- Richardson, Vera
- Doddareddy, Munikumar R
- Ong, Jennifer A
- Huang, Michael L H
- Richardson, Des R
- Kalinowski, Danuta S
Producer: 20160315
In:
Oncotarget vol. 6
Availability: No items available.
|
|
95.
|
The molecular effect of metastasis suppressors on Src signaling and tumorigenesis: new therapeutic targets. [electronic resource] by
- Liu, Wensheng
- Kovacevic, Zaklina
- Peng, Zhihai
- Jin, Runsen
- Wang, Puxiongzhi
- Yue, Fei
- Zheng, Minhua
- Huang, Michael L-H
- Jansson, Patric J
- Richardson, Vera
- Kalinowski, Danuta S
- Lane, Darius J R
- Merlot, Angelica M
- Sahni, Sumit
- Richardson, Des R
Producer: 20161020
In:
Oncotarget vol. 6
Availability: No items available.
|
|
96.
|
Novel Mechanism of Cytotoxicity for the Selective Selenosemicarbazone, 2-Acetylpyridine 4,4-Dimethyl-3-selenosemicarbazone (Ap44mSe): Lysosomal Membrane Permeabilization. [electronic resource] by
- Al-Eisawi, Zaynab
- Stefani, Christian
- Jansson, Patric J
- Arvind, Akanksha
- Sharpe, Philip C
- Basha, Maram T
- Iskander, George M
- Kumar, Naresh
- Kovacevic, Zaklina
- Lane, Darius J R
- Sahni, Sumit
- Bernhardt, Paul V
- Richardson, Des R
- Kalinowski, Danuta S
Producer: 20160518
In:
Journal of medicinal chemistry vol. 59
Availability: No items available.
|
|
97.
|
Structure-activity relationships of novel salicylaldehyde isonicotinoyl hydrazone (SIH) analogs: iron chelation, anti-oxidant and cytotoxic properties. [electronic resource] by
- Potůčková, Eliška
- Hrušková, Kateřina
- Bureš, Jan
- Kovaříková, Petra
- Špirková, Iva A
- Pravdíková, Kateřina
- Kolbabová, Lucie
- Hergeselová, Tereza
- Hašková, Pavlína
- Jansová, Hana
- Macháček, Miloslav
- Jirkovská, Anna
- Richardson, Vera
- Lane, Darius J R
- Kalinowski, Danuta S
- Richardson, Des R
- Vávrová, Kateřina
- Šimůnek, Tomáš
Producer: 20160115
In:
PloS one vol. 9
Availability: No items available.
|
|
98.
|
Redox cycling metals: Pedaling their roles in metabolism and their use in the development of novel therapeutics. [electronic resource] by
- Kalinowski, Danuta S
- Stefani, Christian
- Toyokuni, Shinya
- Ganz, Tomas
- Anderson, Gregory J
- Subramaniam, Nathan V
- Trinder, Debbie
- Olynyk, John K
- Chua, Anita
- Jansson, Patric J
- Sahni, Sumit
- Lane, Darius J R
- Merlot, Angelica M
- Kovacevic, Zaklina
- Huang, Michael L H
- Lee, C Soon
- Richardson, Des R
Producer: 20160606
In:
Biochimica et biophysica acta vol. 1863
Availability: No items available.
|