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Evaluation of various static in vitro-in vivo extrapolation models for risk assessment of the CYP3A inhibition potential of an investigational drug. [electronic resource] by
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- Kirby, B
- Ragueneau-Majlessi, I
- Galetin, A
- Chien, J Y L
- Einolf, H J
- Fahmi, O A
- Fischer, V
- Fretland, A
- Grime, K
- Hall, S D
- Higgs, R
- Plowchalk, D
- Riley, R
- Seibert, E
- Skordos, K
- Snoeys, J
- Venkatakrishnan, K
- Waterhouse, T
- Obach, R S
- Berglund, E G
- Zhang, L
- Zhao, P
- Reynolds, K S
- Huang, S-M
Producer: 20140403
In:
Clinical pharmacology and therapeutics vol. 95
Availability: No items available.
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Overcoming Time-Dependent Inhibition (TDI) of Cytochrome P450 3A4 (CYP3A4) Resulting from Bioactivation of a Fluoropyrimidine Moiety. [electronic resource] by
- Mandal, Mihirbaran
- Mitra, Kaushik
- Grotz, Diane
- Lin, Xinjie
- Palamanda, Jairam
- Kumari, Pramila
- Buevich, Alexei
- Caldwell, John P
- Chen, Xia
- Cox, Kathleen
- Favreau, Leonard
- Hyde, Lynn
- Kennedy, Matthew E
- Kuvelkar, Reshma
- Liu, Xiaoxiang
- Mazzola, Robert D
- Parker, Eric
- Rindgen, Diane
- Sherer, Edward
- Wang, Hongwu
- Zhu, Zhaoning
- Stamford, Andrew W
- Cumming, Jared N
Producer: 20190930
In:
Journal of medicinal chemistry vol. 61
Availability: No items available.
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