Results
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61.
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Identification and structure-activity relationship of phenolic acyl hydrazones as selective agonists for the estrogen-related orphan nuclear receptors ERRbeta and ERRgamma. [electronic resource] by
- Zuercher, William J
- Gaillard, Stéphanie
- Orband-Miller, Lisa A
- Chao, Esther Y H
- Shearer, Barry G
- Jones, David G
- Miller, Aaron B
- Collins, Jon L
- McDonnell, Donald P
- Willson, Timothy M
Producer: 20050603
In:
Journal of medicinal chemistry vol. 48
Availability: No items available.
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62.
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Discovery of a novel class of PPARdelta partial agonists. [electronic resource] by
- Shearer, Barry G
- Patel, Hari S
- Billin, Andrew N
- Way, James M
- Winegar, Deborah A
- Lambert, Millard H
- Xu, Robert X
- Leesnitzer, Lisa M
- Merrihew, Raymond V
- Huet, Stephane
- Willson, Timothy M
Producer: 20081014
In:
Bioorganic & medicinal chemistry letters vol. 18
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63.
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Identification of a novel human constitutive androstane receptor (CAR) agonist and its use in the identification of CAR target genes. [electronic resource] by
- Maglich, Jodi M
- Parks, Derek J
- Moore, Linda B
- Collins, Jon L
- Goodwin, Bryan
- Billin, Andrew N
- Stoltz, Catherine A
- Kliewer, Steven A
- Lambert, Millard H
- Willson, Timothy M
- Moore, John T
Producer: 20030630
In:
The Journal of biological chemistry vol. 278
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64.
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Hepatocyte nuclear factor 4 is a transcription factor that constitutively binds fatty acids. [electronic resource] by
- Wisely, G Bruce
- Miller, Ann B
- Davis, Roderick G
- Thornquest, Alan D
- Johnson, Robert
- Spitzer, Tim
- Sefler, Andrea
- Shearer, Barry
- Moore, John T
- Miller, Aaron B
- Willson, Timothy M
- Williams, Shawn P
Producer: 20030703
In:
Structure (London, England : 1993) vol. 10
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65.
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A ligand-mediated hydrogen bond network required for the activation of the mineralocorticoid receptor. [electronic resource] by
- Bledsoe, Randy K
- Madauss, Kevin P
- Holt, Jason A
- Apolito, Christopher J
- Lambert, Millard H
- Pearce, Kenneth H
- Stanley, Thomas B
- Stewart, Eugene L
- Trump, Ryan P
- Willson, Timothy M
- Williams, Shawn P
Producer: 20051025
In:
The Journal of biological chemistry vol. 280
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66.
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A structural basis for constitutive activity in the human CAR/RXRalpha heterodimer. [electronic resource] by
- Xu, Robert X
- Lambert, Millard H
- Wisely, Bruce B
- Warren, Erin N
- Weinert, Emily E
- Waitt, Gregory M
- Williams, Jon D
- Collins, Jon L
- Moore, Linda B
- Willson, Timothy M
- Moore, John T
Producer: 20050210
In:
Molecular cell vol. 16
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67.
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Small molecule agonists of the orphan nuclear receptors steroidogenic factor-1 (SF-1, NR5A1) and liver receptor homologue-1 (LRH-1, NR5A2). [electronic resource] by
- Whitby, Richard J
- Stec, Jozef
- Blind, Raymond D
- Dixon, Sally
- Leesnitzer, Lisa M
- Orband-Miller, Lisa A
- Williams, Shawn P
- Willson, Timothy M
- Xu, Robert
- Zuercher, William J
- Cai, Fang
- Ingraham, Holly A
Producer: 20110606
In:
Journal of medicinal chemistry vol. 54
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68.
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The Drosophila orphan nuclear receptor DHR38 mediates an atypical ecdysteroid signaling pathway. [electronic resource] by
- Baker, Keith D
- Shewchuk, Lisa M
- Kozlova, Tatiana
- Makishima, Makoto
- Hassell, Annie
- Wisely, Bruce
- Caravella, Justin A
- Lambert, Millard H
- Reinking, Jeffrey L
- Krause, Henry
- Thummel, Carl S
- Willson, Timothy M
- Mangelsdorf, David J
Producer: 20030723
In:
Cell vol. 113
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69.
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Differential inhibition of macrophage foam-cell formation and atherosclerosis in mice by PPARalpha, beta/delta, and gamma. [electronic resource] by
- Li, Andrew C
- Binder, Christoph J
- Gutierrez, Alejandra
- Brown, Kathleen K
- Plotkin, Christine R
- Pattison, Jennifer W
- Valledor, Annabel F
- Davis, Roger A
- Willson, Timothy M
- Witztum, Joseph L
- Palinski, Wulf
- Glass, Christopher K
Producer: 20050208
In:
The Journal of clinical investigation vol. 114
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70.
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X-ray crystal structure of the liver X receptor beta ligand binding domain: regulation by a histidine-tryptophan switch. [electronic resource] by
- Williams, Shawn
- Bledsoe, Randy K
- Collins, Jon L
- Boggs, Sharon
- Lambert, Millard H
- Miller, Ann B
- Moore, John
- McKee, David D
- Moore, Linda
- Nichols, Jason
- Parks, Derek
- Watson, Mike
- Wisely, Bruce
- Willson, Timothy M
Producer: 20030827
In:
The Journal of biological chemistry vol. 278
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71.
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Discovery of novel quinoline-based estrogen receptor ligands using peptide interaction profiling. [electronic resource] by
- Hoekstra, William J
- Patel, Hari S
- Liang, Xi
- Blanc, Jean-Baptiste E
- Heyer, Dennis O
- Willson, Timothy M
- Iannone, Marie A
- Kadwell, Sue H
- Miller, Lisa A
- Pearce, Kenneth H
- Simmons, Catherine A
- Shearin, Jean
Producer: 20050503
In:
Journal of medicinal chemistry vol. 48
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72.
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Tyrosine agonists reverse the molecular defects associated with dominant-negative mutations in human peroxisome proliferator-activated receptor gamma. [electronic resource] by
- Agostini, Maura
- Gurnell, Mark
- Savage, David B
- Wood, Emily M
- Smith, Aaron G
- Rajanayagam, Odelia
- Garnes, Keith T
- Levinson, Sidney H
- Xu, H Eric
- Schwabe, John W R
- Willson, Timothy M
- O'Rahilly, Stephen
- Chatterjee, V Krishna
Producer: 20040416
In:
Endocrinology vol. 145
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73.
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1,2,6-Thiadiazinones as Novel Narrow Spectrum Calcium/Calmodulin-Dependent Protein Kinase Kinase 2 (CaMKK2) Inhibitors. [electronic resource] by
- Asquith, Christopher R M
- Godoi, Paulo H
- Couñago, Rafael M
- Laitinen, Tuomo
- Scott, John W
- Langendorf, Christopher G
- Oakhill, Jonathan S
- Drewry, David H
- Zuercher, William J
- Koutentis, Panayiotis A
- Willson, Timothy M
- Kalogirou, Andreas S
Producer: 20180927
In:
Molecules (Basel, Switzerland) vol. 23
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74.
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In Depth Analysis of Kinase Cross Screening Data to Identify CAMKK2 Inhibitory Scaffolds. [electronic resource] by
- O'Byrne, Sean N
- Scott, John W
- Pilotte, Joseph R
- Santiago, André da S
- Langendorf, Christopher G
- Oakhill, Jonathan S
- Eduful, Benjamin J
- Couñago, Rafael M
- Wells, Carrow I
- Zuercher, William J
- Willson, Timothy M
- Drewry, David H
Producer: 20201007
In:
Molecules (Basel, Switzerland) vol. 25
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75.
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Novel selective small molecule agonists for peroxisome proliferator-activated receptor delta (PPARdelta)--synthesis and biological activity. [electronic resource] by
- Sznaidman, Marcos L
- Haffner, Curt D
- Maloney, Patrick R
- Fivush, Adam
- Chao, Esther
- Goreham, Donna
- Sierra, Michael L
- LeGrumelec, Christelle
- Xu, H Eric
- Montana, Valerie G
- Lambert, Millard H
- Willson, Timothy M
- Oliver, William R
- Sternbach, Daniel D
Producer: 20040106
In:
Bioorganic & medicinal chemistry letters vol. 13
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76.
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Identification and Optimization of 4-Anilinoquinolines as Inhibitors of Cyclin G Associated Kinase. [electronic resource] by
- Asquith, Christopher R M
- Laitinen, Tuomo
- Bennett, James M
- Godoi, Paulo H
- East, Michael P
- Tizzard, Graham J
- Graves, Lee M
- Johnson, Gary L
- Dornsife, Ronna E
- Wells, Carrow I
- Elkins, Jonathan M
- Willson, Timothy M
- Zuercher, William J
Producer: 20181004
In:
ChemMedChem vol. 13
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77.
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Co-crystal structure guided array synthesis of PPARgamma inverse agonists. [electronic resource] by
- Trump, Ryan P
- Cobb, Jeffrey E
- Shearer, Barry G
- Lambert, Millard H
- Nolte, Robert T
- Willson, Timothy M
- Buckholz, Richard G
- Zhao, Sumin M
- Leesnitzer, Lisa M
- Iannone, Marie A
- Pearce, Kenneth H
- Billin, Andrew N
- Hoekstra, William J
Producer: 20070924
In:
Bioorganic & medicinal chemistry letters vol. 17
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78.
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A public-private partnership to unlock the untargeted kinome. [electronic resource] by
- Knapp, Stefan
- Arruda, Paulo
- Blagg, Julian
- Burley, Stephen
- Drewry, David H
- Edwards, Aled
- Fabbro, Doriano
- Gillespie, Paul
- Gray, Nathanael S
- Kuster, Bernhard
- Lackey, Karen E
- Mazzafera, Paulo
- Tomkinson, Nicholas C O
- Willson, Timothy M
- Workman, Paul
- Zuercher, William J
Producer: 20130204
In:
Nature chemical biology vol. 9
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79.
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Identification and characterization of 4-chloro-N-(2-{[5-trifluoromethyl)-2-pyridyl]sulfonyl}ethyl)benzamide (GSK3787), a selective and irreversible peroxisome proliferator-activated receptor delta (PPARdelta) antagonist. [electronic resource] by
- Shearer, Barry G
- Wiethe, Robert W
- Ashe, Adam
- Billin, Andrew N
- Way, James M
- Stanley, Thomas B
- Wagner, Craig D
- Xu, Robert X
- Leesnitzer, Lisa M
- Merrihew, Raymond V
- Shearer, Todd W
- Jeune, Michael R
- Ulrich, John C
- Willson, Timothy M
Producer: 20100323
In:
Journal of medicinal chemistry vol. 53
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80.
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Crystal structure of the glucocorticoid receptor ligand binding domain reveals a novel mode of receptor dimerization and coactivator recognition. [electronic resource] by
- Bledsoe, Randy K
- Montana, Valerie G
- Stanley, Thomas B
- Delves, Chris J
- Apolito, Christopher J
- McKee, David D
- Consler, Thomas G
- Parks, Derek J
- Stewart, Eugene L
- Willson, Timothy M
- Lambert, Millard H
- Moore, John T
- Pearce, Kenneth H
- Xu, H Eric
Producer: 20020829
In:
Cell vol. 110
Availability: No items available.
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