Results
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61.
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Synthesis, cytotoxic activity, and mechanism of action of furo[2,3-c]acridin-6-one and benzo[b]furo[3,2-h]acridin-6-one analogues of psorospermin and acronycine. [electronic resource] by
- Boutefnouchet, Sabrina
- Gaboriaud-Kolar, Nicolas
- Nguyen, Tuan Minh
- Depauw, Sabine
- David-Cordonnier, Marie-Hélène
- Pfeiffer, Bruno
- Léonce, Stéphane
- Pierré, Alain
- Tillequin, François
- Lallemand, Marie-Christine
- Michel, Sylvie
Producer: 20090403
In:
Journal of medicinal chemistry vol. 51
Availability: No items available.
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62.
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Synthesis and biological study of a new series of 4'-demethylepipodophyllotoxin derivatives. [electronic resource] by
- Duca, Maria
- Guianvarc'h, Dominique
- Meresse, Philippe
- Bertounesque, Emmanuel
- Dauzonne, Daniel
- Kraus-Berthier, Laurence
- Thirot, Sylvie
- Léonce, Stéphane
- Pierré, Alain
- Pfeiffer, Bruno
- Renard, Pierre
- Arimondo, Paola B
- Monneret, Claude
Producer: 20050304
In:
Journal of medicinal chemistry vol. 48
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63.
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Synthesis of mono- and bisdihydrodipyridopyrazines and assessment of their DNA binding and cytotoxic properties. [electronic resource] by
- Blanchard, Stéphanie
- Rodriguez, Ivan
- Tardy, Christelle
- Baldeyrou, Brigitte
- Bailly, Christian
- Colson, Pierre
- Houssier, Claude
- Léonce, Stéphane
- Kraus-Berthier, Laurence
- Pfeiffer, Bruno
- Renard, Pierre
- Pierré, Alain
- Caubère, Paul
- Guillaumet, Gérald
Producer: 20040405
In:
Journal of medicinal chemistry vol. 47
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64.
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Novel stable camptothecin derivatives replacing the E-ring lactone by a ketone function are potent inhibitors of topoisomerase I and promising antitumor drugs. [electronic resource] by
- Lansiaux, Amélie
- Léonce, Stéphane
- Kraus-Berthier, Laurence
- Bal-Mahieu, Christine
- Mazinghien, Romain
- Didier, Sébastien
- David-Cordonnier, Marie-Hélène
- Hautefaye, Patrick
- Lavielle, Gilbert
- Bailly, Christian
- Hickman, John A
- Pierré, Alain
Producer: 20070905
In:
Molecular pharmacology vol. 72
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65.
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Influence of the stereoisomeric position of the reactive acetate groups of the benzo[b]acronycine derivative S23906-1 on its DNA alkylation, helix-opening, cytotoxic, and antitumor activities. [electronic resource] by
- Depauw, Sabine
- Gaslonde, Thomas
- Léonce, Stéphane
- Kraus-Berthier, Laurence
- Laine, William
- Lenglet, Gaëlle
- Chiaroni, Angèle
- Pfeiffer, Bruno
- Bailly, Christian
- Michel, Sylvie
- Tillequin, François
- Pierré, Alain
- David-Cordonnier, Marie-Hélène
Producer: 20091217
In:
Molecular pharmacology vol. 76
Availability: No items available.
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66.
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A transesterification reaction is implicated in the covalent binding of benzo[b]acronycine anticancer agents with DNA and glutathion. [electronic resource] by
- David-Cordonnier, Marie Hélène
- Laine, William
- Kouach, Mostafa
- Briand, Gilbert
- Vezin, Hervé
- Gaslonde, Thomas
- Michel, Sylvie
- Doan Thi Mai, Huong
- Tillequin, Francois
- Koch, Michel
- Léonce, Stéphane
- Pierré, Alain
- Bailly, Christian
Producer: 20040916
In:
Bioorganic & medicinal chemistry vol. 12
Availability: No items available.
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67.
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Synthesis, antitumor activity, and mechanism of action of benzo[a]pyrano[3,2-h]acridin-7-one analogues of acronycine. [electronic resource] by
- Nguyen, Tuan Minh
- Sittisombut, Chavalit
- Boutefnouchet, Sabrina
- Lallemand, Marie-Christine
- Michel, Sylvie
- Koch, Michel
- Tillequin, François
- Mazinghien, Romain
- Lansiaux, Amélie
- David-Cordonnier, Marie-Hélène
- Pfeiffer, Bruno
- Kraus-Berthier, Laurence
- Léonce, Stéphane
- Pierré, Alain
Producer: 20060712
In:
Journal of medicinal chemistry vol. 49
Availability: No items available.
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68.
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Covalent binding to glutathione of the DNA-alkylating antitumor agent, S23906-1. [electronic resource] by
- David-Cordonnier, Marie-Hélène
- Laine, William
- Joubert, Alexandra
- Tardy, Christelle
- Goossens, Jean-François
- Kouach, Mostafa
- Briand, Gilbert
- Thi Mai, Huong Doan
- Michel, Sylvie
- Tillequin, Francois
- Koch, Michel
- Leonce, Stéphane
- Pierre, Alain
- Bailly, Christian
Producer: 20030829
In:
European journal of biochemistry vol. 270
Availability: No items available.
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69.
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Specific oncogenic activity of the Src-family tyrosine kinase c-Yes in colon carcinoma cells. [electronic resource] by
- Sancier, Florence
- Dumont, Aurélie
- Sirvent, Audrey
- Paquay de Plater, Ludmilla
- Edmonds, Thomas
- David, Géraldine
- Jan, Michel
- de Montrion, Catherine
- Cogé, Francis
- Léonce, Stéphane
- Burbridge, Michael
- Bruno, Alain
- Boutin, Jean A
- Lockhart, Brian
- Roche, Serge
- Cruzalegui, Francisco
Producer: 20110901
In:
PloS one vol. 6
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70.
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Characterization of novel checkpoint kinase 1 inhibitors by in vitro assays and in human cancer cells treated with topoisomerase inhibitors. [electronic resource] by
- Ferry, Gilles
- Studeny, Aurélie
- Bossard, Céline
- Kubara, Philip M
- Zeyer, Denis
- Renaud, Jean-Paul
- Casara, Patrick
- de Nanteuil, Guillaume
- Wierzbicki, Michel
- Pfeiffer, Bruno
- Prudhomme, Michelle
- Leonce, Stephane
- Pierré, Alain
- Boutin, Jean A
- Golsteyn, Roy M
Producer: 20110929
In:
Life sciences vol. 89
Availability: No items available.
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71.
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Synthesis, cytotoxic activity, and DNA binding properties of antitumor cis-1,2-dihydroxy-1,2-dihydrobenzo[b]acronycine cinnamoyl esters. [electronic resource] by
- Do, Quyên
- Tian, Wen
- Yougnia, Rodrigue
- Gaslonde, Thomas
- Pfeiffer, Bruno
- Pierré, Alain
- Léonce, Stéphane
- Kraus-Berthier, Laurence
- David-Cordonnier, Marie-Hélène
- Depauw, Sabine
- Lansiaux, Amélie
- Mazinghien, Romain
- Koch, Michel
- Tillequin, François
- Michel, Sylvie
- Dufat, Hanh
Producer: 20090529
In:
Bioorganic & medicinal chemistry vol. 17
Availability: No items available.
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72.
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Structure-activity relationships and mechanism of action of antitumor benzo[b]pyrano[3,2-h]acridin-7-one acronycine analogues. [electronic resource] by
- Thi Mai, Huong Doan
- Gaslonde, Thomas
- Michel, Sylvie
- Tillequin, François
- Koch, Michel
- Bongui, Jean-Bernard
- Elomri, Abdelhakim
- Seguin, Elisabeth
- Pfeiffer, Bruno
- Renard, Pierre
- David-Cordonnier, Marie-Hélène
- Laine, William
- Bailly, Christian
- Kraus-Berthier, Laurence
- Léonce, Stéphane
- Hickman, John A
- Pierré, Alain
Producer: 20030807
In:
Journal of medicinal chemistry vol. 46
Availability: No items available.
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73.
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S49076 is a novel kinase inhibitor of MET, AXL, and FGFR with strong preclinical activity alone and in association with bevacizumab. [electronic resource] by
- Burbridge, Mike F
- Bossard, Céline J
- Saunier, Carine
- Fejes, Imre
- Bruno, Alain
- Léonce, Stéphane
- Ferry, Gilles
- Da Violante, Georges
- Bouzom, François
- Cattan, Valérie
- Jacquet-Bescond, Anne
- Comoglio, Paolo M
- Lockhart, Brian P
- Boutin, Jean A
- Cordi, Alex
- Ortuno, Jean-Claude
- Pierré, Alain
- Hickman, John A
- Cruzalegui, Francisco H
- Depil, Stéphane
Producer: 20140401
In:
Molecular cancer therapeutics vol. 12
Availability: No items available.
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