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	61.	Structure-activity relationships of quinoxaline-based 5-HT3A and 5-HT3AB receptor-selective ligands. [electronic resource] by Thompson, Andrew J Verheij, Mark H P van Muijlwijk-Koezen, Jacqueline E Lummis, Sarah C R Leurs, Rob de Esch, Iwan J P Producer: 20140123 In: ChemMedChem vol. 8 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	62.	Synthesis and structure-activity relationships of 3H-quinazolin-4-ones and 3H-pyrido[2,3-d]pyrimidin-4-ones as CXCR3 receptor antagonists. [electronic resource] by Storelli, Stefania Verzijl, Dennis Al-Badie, Jawad Elders, Niels Bosch, Leontien Timmerman, Henk Smit, Martine J De Esch, Iwan J P Leurs, Rob Producer: 20070912 In: Archiv der Pharmazie vol. 340 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	63.	Chemical insights in the concept of hybrid drugs: the antitumor effect of nitric oxide-donating aspirin involves a quinone methide but not nitric oxide nor aspirin. [electronic resource] by Hulsman, Niels Medema, Jan Paul Bos, Carina Jongejan, Aldo Leurs, Rob Smit, Martine J de Esch, Iwan J P Richel, Dick Wijtmans, Maikel Producer: 20070706 In: Journal of medicinal chemistry vol. 50 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	64.	Design, synthesis, and structure-activity relationships of highly potent 5-HT₃ receptor ligands. [electronic resource] by Verheij, Mark H P Thompson, Andrew J van Muijlwijk-Koezen, Jacqueline E Lummis, Sarah C R Leurs, Rob de Esch, Iwan J P Producer: 20130205 In: Journal of medicinal chemistry vol. 55 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	65.	Combining quantum mechanical ligand conformation analysis and protein modeling to elucidate GPCR-ligand binding modes. [electronic resource] by Schultes, Sabine Engelhardt, Harald Roumen, Luc Zuiderveld, Obbe P Haaksma, Eric E J de Esch, Iwan J P Leurs, Rob de Graaf, Chris Producer: 20130528 In: ChemMedChem vol. 8 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	66.	Surface plasmon resonance biosensor assay for the analysis of small-molecule inhibitor binding to human and parasitic phosphodiesterases. [electronic resource] by Siderius, Marco Shanmugham, Anitha England, Paul van der Meer, Tiffany Bebelman, Jan Paul Blaazer, Antoni R de Esch, Iwan J P Leurs, Rob Producer: 20170504 In: Analytical biochemistry vol. 503 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	67.	Pharmacological characterization of [3H]VUF11211, a novel radiolabeled small-molecule inverse agonist for the chemokine receptor CXCR3. [electronic resource] by Scholten, Danny J Wijtmans, Maikel van Senten, Jeffrey R Custers, Hans Stunnenberg, Ailas de Esch, Iwan J P Smit, Martine J Leurs, Rob Producer: 20150526 In: Molecular pharmacology vol. 87 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	68.	Fragment based design of new H4 receptor-ligands with anti-inflammatory properties in vivo. [electronic resource] by Smits, Rogier A Lim, Herman D Hanzer, Agnes Zuiderveld, Obbe P Guaita, Elena Adami, Maristella Coruzzi, Gabriella Leurs, Rob de Esch, Iwan J P Producer: 20080602 In: Journal of medicinal chemistry vol. 51 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	69.	Combinatorial Consensus Scoring for Ligand-Based Virtual Fragment Screening: A Comparative Case Study for Serotonin 5-HT(3)A, Histamine H(1), and Histamine H(4) Receptors. [electronic resource] by Schultes, Sabine Kooistra, Albert J Vischer, Henry F Nijmeijer, Saskia Haaksma, Eric E J Leurs, Rob de Esch, Iwan J P de Graaf, Chris Producer: 20160218 In: Journal of chemical information and modeling vol. 55 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	70.	A chemical switch for the modulation of the functional activity of higher homologues of histamine on the human histamine H3 receptor: effect of various substitutions at the primary amino function. [electronic resource] by Govoni, Marinella Lim, Herman D El-Atmioui, Dris Menge, Wiro M P B Timmerman, Henk Bakker, Remko A Leurs, Rob De Esch, Iwan J P Producer: 20060522 In: Journal of medicinal chemistry vol. 49 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	71.	Discovery of quinazolines as histamine H4 receptor inverse agonists using a scaffold hopping approach. [electronic resource] by Smits, Rogier A de Esch, Iwan J P Zuiderveld, Obbe P Broeker, Joachim Sansuk, Kamonchanok Guaita, Elena Coruzzi, Gabriella Adami, Maristella Haaksma, Eric Leurs, Rob Producer: 20090122 In: Journal of medicinal chemistry vol. 51 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	72.	When fragments link: a bibliometric perspective on the development of fragment-based drug discovery. [electronic resource] by Romasanta, Angelo K S van der Sijde, Peter Hellsten, Iina Hubbard, Roderick E Keseru, Gyorgy M van Muijlwijk-Koezen, Jacqueline de Esch, Iwan J P Producer: 20190114 In: Drug discovery today vol. 23 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	73.	A novel series of histamine H4 receptor antagonists based on the pyrido[3,2-d]pyrimidine scaffold: comparison of hERG binding and target residence time with PF-3893787. [electronic resource] by Andaloussi, Mounir Lim, Herman D van der Meer, Tiffany Sijm, Maarten Poulie, Chris B M de Esch, Iwan J P Leurs, Rob Smits, Rogier A Producer: 20131108 In: Bioorganic & medicinal chemistry letters vol. 23 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	74.	Synthesis and structure-activity relationship of 3-phenyl-3H-quinazolin-4-one derivatives as CXCR3 chemokine receptor antagonists. [electronic resource] by Storelli, Stefania Verdijk, Pauline Verzijl, Dennis Timmerman, Henk van de Stolpe, Andrea C Tensen, Cornelis P Smit, Martine J De Esch, Iwan J P Leurs, Rob Producer: 20051031 In: Bioorganic & medicinal chemistry letters vol. 15 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	75.	Antinociceptive activity of chemical congeners of improgan: optimization of side chain length leads to the discovery of a new, potent, non-opioid analgesic. [electronic resource] by Hough, Lindsay B de Esch, Iwan J P Janssen, Elwin Phillips, James Svokos, Konstantina Kern, Brian Trachler, Jennifer Abood, Mary E Leurs, Rob Nalwalk, Julia W Producer: 20061214 In: Neuropharmacology vol. 51 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	76.	Pharmacological characterization of the new histamine H4 receptor agonist VUF 8430. [electronic resource] by Lim, Herman D Adami, Maristella Guaita, Elena Werfel, Thomas Smits, Rogier A de Esch, Iwan J P Bakker, Remko A Gutzmer, Ralf Coruzzi, Gabriella Leurs, Rob Producer: 20090617 In: British journal of pharmacology vol. 157 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	77.	Ligand based design of novel histamine H₄ receptor antagonists; fragment optimization and analysis of binding kinetics. [electronic resource] by Smits, Rogier A Lim, Herman D van der Meer, Tiffany Kuhne, Sebastiaan Bessembinder, Karin Zuiderveld, Obbe P Wijtmans, Maikel de Esch, Iwan J P Leurs, Rob Producer: 20120803 In: Bioorganic & medicinal chemistry letters vol. 22 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	78.	Fragment based lead discovery of small molecule inhibitors for the EPHA4 receptor tyrosine kinase. [electronic resource] by van Linden, Oscar P J Farenc, Carine Zoutman, Willem H Hameetman, Liesbeth Wijtmans, Maikel Leurs, Rob Tensen, Cornelis P Siegal, Gregg de Esch, Iwan J P Producer: 20120529 In: European journal of medicinal chemistry vol. 47 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	79.	EPHA4 is overexpressed but not functionally active in Sézary syndrome. [electronic resource] by Hameetman, Liesbeth van der Fits, Leslie Zoutman, Willem H Out-Luiting, Jacoba J Siegal, Gregg de Esch, Iwan J P Vermeer, Maarten H Tensen, Cornelis P Producer: 20160818 In: Oncotarget vol. 6 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	80.	Identification of novel allosteric nonpeptidergic inhibitors of the human cytomegalovirus-encoded chemokine receptor US28. [electronic resource] by Vischer, Henry F Hulshof, Janneke W Hulscher, Saskia Fratantoni, Silvina A Verheij, Mark H P Victorina, Jane Smit, Martine J de Esch, Iwan J P Leurs, Rob Producer: 20100427 In: Bioorganic & medicinal chemistry vol. 18 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)

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Your search returned 132 results.