Results
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61.
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1,3,4-Trisubstituted pyrrolidine CCR5 receptor antagonists. Part 3: polar functionality and its effect on anti-HIV-1 activity. [electronic resource] by
- Hale, Jeffrey J
- Budhu, Richard J
- Mills, Sander G
- MacCoss, Malcolm
- Gould, Sandra L
- DeMartino, Julie A
- Springer, Martin S
- Siciliano, Salvatore J
- Malkowitz, Lorraine
- Schleif, William A
- Hazuda, Daria
- Miller, Michael
- Kessler, Joseph
- Danzeisen, Renee
- Holmes, Karen
- Lineberger, Janet
- Carella, Anthony
- Carver, Gwen
- Emini, Emilio A
Producer: 20030311
In:
Bioorganic & medicinal chemistry letters vol. 12
Availability: No items available.
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62.
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Synthesis and evaluation of CCR5 antagonists containing modified 4-piperidinyl-2-phenyl-1-(phenylsulfonylamino)-butane. [electronic resource] by
- Shah, Shrenik K
- Chen, Natalie
- Guthikonda, Ravindra N
- Mills, Sander G
- Malkowitz, Lorraine
- Springer, Martin S
- Gould, Sandra L
- Demartino, Julie A
- Carella, Anthony
- Carver, Gwen
- Holmes, Karen
- Schleif, William A
- Danzeisen, Renee
- Hazuda, Daria
- Kessler, Joseph
- Lineberger, Janet
- Miller, Michael
- Emini, Emilio A
- MacCoss, Malcolm
Producer: 20050615
In:
Bioorganic & medicinal chemistry letters vol. 15
Availability: No items available.
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63.
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Universal influenza B vaccine based on the maturational cleavage site of the hemagglutinin precursor. [electronic resource] by
- Bianchi, Elisabetta
- Liang, Xiaoping
- Ingallinella, Paolo
- Finotto, Marco
- Chastain, Michael A
- Fan, Jiang
- Fu, Tong-Ming
- Song, Hong Chang
- Horton, Melanie S
- Freed, Daniel C
- Manger, Walter
- Wen, Emily
- Shi, Li
- Ionescu, Roxana
- Price, Colleen
- Wenger, Marc
- Emini, Emilio A
- Cortese, Riccardo
- Ciliberto, Gennaro
- Shiver, John W
- Pessi, Antonello
Producer: 20050628
In:
Journal of virology vol. 79
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64.
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Vaccine-induced immune responses in rodents and nonhuman primates by use of a humanized human immunodeficiency virus type 1 pol gene. [electronic resource] by
- Casimiro, Danilo R
- Tang, Aimin
- Perry, Helen C
- Long, Romnie S
- Chen, Minchun
- Heidecker, Gwendolyn J
- Davies, Mary-Ellen
- Freed, Daniel C
- Persaud, Natasha V
- Dubey, Sheri
- Smith, Jeffrey G
- Havlir, Diane
- Richman, Douglas
- Chastain, Michael A
- Simon, Adam J
- Fu, Tong-Ming
- Emini, Emilio A
- Shiver, John W
Producer: 20020110
In:
Journal of virology vol. 76
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65.
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Syntheses and SAR studies of 4-(heteroarylpiperdin-1-yl-methyl)-pyrrolidin-1-yl-acetic acid antagonists of the human CCR5 chemokine receptor. [electronic resource] by
- Shankaran, K
- Donnelly, Karla L
- Shah, Shrenik K
- Guthikonda, Ravindra N
- MacCoss, Malcolm
- Mills, Sander G
- Gould, Sandra L
- Malkowitz, Lorraine
- Siciliano, Salvatore J
- Springer, Martin S
- Carella, Anthony
- Carver, Gwen
- Hazuda, Daria
- Holmes, Karen
- Kessler, Joseph
- Lineberger, Janet
- Miller, Michael D
- Emini, Emilio A
- Schleif, William A
Producer: 20050202
In:
Bioorganic & medicinal chemistry letters vol. 14
Availability: No items available.
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66.
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Antagonists of human CCR5 receptor containing 4-(pyrazolyl)piperidine side chains. Part 1: Discovery and SAR study of 4-pyrazolylpiperidine side chains. [electronic resource] by
- Shen, Dong-Ming
- Shu, Min
- Mills, Sander G
- Chapman, Kevin T
- Malkowitz, Lorraine
- Springer, Martin S
- Gould, Sandra L
- DeMartino, Julie A
- Siciliano, Salvatore J
- Kwei, Gloria Y
- Carella, Anthony
- Carver, Gwen
- Holmes, Karen
- Schleif, William A
- Danzeisen, Renee
- Hazuda, Daria
- Kessler, Joseph
- Lineberger, Janet
- Miller, Michael D
- Emini, Emilio A
Producer: 20040928
In:
Bioorganic & medicinal chemistry letters vol. 14
Availability: No items available.
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67.
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13-valent pneumococcal conjugate vaccine (PCV13) is immunogenic and safe in children 6-17 years of age with sickle cell disease previously vaccinated with 23-valent pneumococcal polysaccharide vaccine (PPSV23): Results of a phase 3 study. [electronic resource] by
- De Montalembert, Mariane
- Abboud, Miguel R
- Fiquet, Anne
- Inati, Adlette
- Lebensburger, Jeffrey D
- Kaddah, Normeen
- Mokhtar, Galila
- Piga, Antonio
- Halasa, Natasha
- Inusa, Baba
- Rees, David C
- Heath, Paul T
- Telfer, Paul
- Driscoll, Catherine
- Al Hajjar, Sami
- Tozzi, Alberto
- Jiang, Qin
- Emini, Emilio A
- Gruber, William C
- Gurtman, Alejandra
- Scott, Daniel A
Producer: 20150911
In:
Pediatric blood & cancer vol. 62
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68.
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Immunogenicity and reactogenicity of a 13-valent-pneumococcal conjugate vaccine administered at 2, 4, and 12 months of age: a double-blind randomized active-controlled trial. [electronic resource] by
- Snape, Matthew D
- Klinger, Chaam L
- Daniels, Elvis D
- John, Tessa M
- Layton, Helen
- Rollinson, Llinos
- Pestridge, Sarah
- Dymond, Sandra
- Galiza, Eva
- Tansey, Susan
- Scott, Daniel A
- Baker, Sherryl A
- Jones, Thomas R
- Yu, Ly-Mee
- Gruber, William C
- Emini, Emilio A
- Faust, Saul N
- Finn, Adam
- Heath, Paul T
- Pollard, Andrew J
Producer: 20110302
In:
The Pediatric infectious disease journal vol. 29
Availability: No items available.
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69.
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Preclinical study of influenza virus A M2 peptide conjugate vaccines in mice, ferrets, and rhesus monkeys. [electronic resource] by
- Fan, Jiang
- Liang, Xiaoping
- Horton, Melanie S
- Perry, Helen C
- Citron, Michael P
- Heidecker, Gwen J
- Fu, Tong-Ming
- Joyce, Joseph
- Przysiecki, Craig T
- Keller, Paul M
- Garsky, Victor M
- Ionescu, Roxana
- Rippeon, Yvette
- Shi, Li
- Chastain, Michael A
- Condra, Jon H
- Davies, Mary-Ellen
- Liao, Jason
- Emini, Emilio A
- Shiver, John W
Producer: 20041110
In:
Vaccine vol. 22
Availability: No items available.
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70.
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Potent 1,3,4-trisubstituted pyrrolidine CCR5 receptor antagonists: effects of fused heterocycles on antiviral activity and pharmacokinetic properties. [electronic resource] by
- Kim, Dooseop
- Wang, Liping
- Hale, Jeffrey J
- Lynch, Christopher L
- Budhu, Richard J
- Maccoss, Malcolm
- Mills, Sander G
- Malkowitz, Lorraine
- Gould, Sandra L
- DeMartino, Julie A
- Springer, Martin S
- Hazuda, Daria
- Miller, Michael
- Kessler, Joseph
- Hrin, Renee C
- Carver, Gwen
- Carella, Anthony
- Henry, Karen
- Lineberger, Janet
- Schleif, William A
- Emini, Emilio A
Producer: 20050818
In:
Bioorganic & medicinal chemistry letters vol. 15
Availability: No items available.
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71.
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CCR5 antagonists: bicyclic isoxazolidines as conformationally constrained N-1-substituted pyrrolidines. [electronic resource] by
- Lynch, Christopher L
- Gentry, Amy L
- Hale, Jeffrey J
- Mills, Sander G
- MacCoss, Malcolm
- Malkowitz, Lorraine
- Springer, Martin S
- Gould, Sandra L
- DeMartino, Julie A
- Siciliano, Salvatore J
- Cascieri, Margaret A
- Doss, George
- Carella, Anthony
- Carver, Gwen
- Holmes, Karen
- Schleif, William A
- Danzeisen, Renee
- Hazuda, Daria
- Kessler, Joseph
- Lineberger, Janet
- Miller, Michael
- Emini, Emilio A
Producer: 20030731
In:
Bioorganic & medicinal chemistry letters vol. 12
Availability: No items available.
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72.
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1,3,4-Trisubstituted pyrrolidine CCR5 receptor antagonists. Part 4: synthesis of N-1 acidic functionality affording analogues with enhanced antiviral activity against HIV. [electronic resource] by
- Lynch, Christopher L
- Hale, Jeffrey J
- Budhu, Richard J
- Gentry, Amy L
- Mills, Sander G
- Chapman, Kevin T
- MacCoss, Malcolm
- Malkowitz, Lorraine
- Springer, Martin S
- Gould, Sandra L
- DeMartino, Julie A
- Siciliano, Salvatore J
- Cascieri, Margaret A
- Carella, Anthony
- Carver, Gwen
- Holmes, Karen
- Schleif, William A
- Danzeisen, Renee
- Hazuda, Daria
- Kessler, Joseph
- Lineberger, Janet
- Miller, Michael
- Emini, Emilio A
Producer: 20030311
In:
Bioorganic & medicinal chemistry letters vol. 12
Availability: No items available.
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73.
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1,3,4 Trisubstituted pyrrolidine CCR5 receptor antagonists bearing 4-aminoheterocycle substituted piperidine side chains. [electronic resource] by
- Willoughby, Christopher A
- Rosauer, Keith G
- Hale, Jeffery J
- Budhu, Richard J
- Mills, Sander G
- Chapman, Kevin T
- MacCoss, Malcolm
- Malkowitz, Lorraine
- Springer, Martin S
- Gould, Sandra L
- DeMartino, Julie A
- Siciliano, Salvatore J
- Cascieri, Margaret A
- Carella, Anthony
- Carver, Gwen
- Holmes, Karen
- Schleif, William A
- Danzeisen, Renee
- Hazuda, Daria
- Kessler, Joseph
- Lineberger, Janet
- Miller, Michael
- Emini, Emilio A
Producer: 20030815
In:
Bioorganic & medicinal chemistry letters vol. 13
Availability: No items available.
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74.
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Vectored Gag and Env but not Tat show efficacy against simian-human immunodeficiency virus 89.6P challenge in Mamu-A*01-negative rhesus monkeys. [electronic resource] by
- Liang, Xiaoping
- Casimiro, Danilo R
- Schleif, William A
- Wang, Fubao
- Davies, Mary-Ellen
- Zhang, Zhi-Qiang
- Fu, Tong-Ming
- Finnefrock, Adam C
- Handt, Larry
- Citron, Michael P
- Heidecker, Gwendolyn
- Tang, Aimin
- Chen, Minchun
- Wilson, Keith A
- Gabryelski, Lori
- McElhaugh, Michael
- Carella, Anthony
- Moyer, Cheryl
- Huang, Lingyi
- Vitelli, Salvatore
- Patel, Deepa
- Lin, Jing
- Emini, Emilio A
- Shiver, John W
Producer: 20051021
In:
Journal of virology vol. 79
Availability: No items available.
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75.
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Syntheses and biological evaluation of 5-(piperidin-1-yl)-3-phenyl-pentylsulfones as CCR5 antagonists. [electronic resource] by
- Shankaran, K
- Donnelly, Karla L
- Shah, Shrenik K
- Caldwell, Charles G
- Chen, Ping
- Finke, Paul E
- Oates, Bryan
- MacCoss, Malcolm
- Mills, Sander G
- DeMartino, Julie A
- Gould, Sandra L
- Malkowitz, Lorraine
- Siciliano, Salvatore J
- Springer, Martin S
- Kwei, Gloria
- Carella, Anthony
- Carver, Gwen
- Danzeisen, Renee
- Hazuda, Daria
- Holmes, Karen
- Kessler, Joseph
- Lineberger, Janet
- Miller, Michael D
- Emini, Emilio A
- Schleif, William A
Producer: 20050202
In:
Bioorganic & medicinal chemistry letters vol. 14
Availability: No items available.
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76.
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Integrase inhibitors and cellular immunity suppress retroviral replication in rhesus macaques. [electronic resource] by
- Hazuda, Daria J
- Young, Steven D
- Guare, James P
- Anthony, Neville J
- Gomez, Robert P
- Wai, John S
- Vacca, Joseph P
- Handt, Larry
- Motzel, Sherri L
- Klein, Hilton J
- Dornadula, Geethanjali
- Danovich, Robert M
- Witmer, Marc V
- Wilson, Keith A A
- Tussey, Lynda
- Schleif, William A
- Gabryelski, Lori S
- Jin, Lixia
- Miller, Michael D
- Casimiro, Danilo R
- Emini, Emilio A
- Shiver, John W
Producer: 20040809
In:
Science (New York, N.Y.) vol. 305
Availability: No items available.
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77.
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Vaccine-induced immunity in baboons by using DNA and replication-incompetent adenovirus type 5 vectors expressing a human immunodeficiency virus type 1 gag gene. [electronic resource] by
- Casimiro, Danilo R
- Tang, Aimin
- Chen, Ling
- Fu, Tong-Ming
- Evans, Robert K
- Davies, Mary-Ellen
- Freed, Daniel C
- Hurni, William
- Aste-Amezaga, Jose M
- Guan, Liming
- Long, Romnie
- Huang, Lingyi
- Harris, Virginia
- Nawrocki, Denise K
- Mach, Henryk
- Troutman, Robert D
- Isopi, Lynne A
- Murthy, Krishna K
- Rice, Karen
- Wilson, Keith A
- Volkin, David B
- Emini, Emilio A
- Shiver, John W
Producer: 20030801
In:
Journal of virology vol. 77
Availability: No items available.
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78.
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Antagonists of human CCR5 receptor containing 4-(pyrazolyl)piperidine side chains. Part 3: SAR studies on the benzylpyrazole segment. [electronic resource] by
- Shu, Min
- Loebach, Jennifer L
- Parker, Kerry A
- Mills, Sander G
- Chapman, Kevin T
- Shen, Dong-Ming
- Malkowitz, Lorraine
- Springer, Martin S
- Gould, Sandra L
- DeMartino, Julie A
- Siciliano, Salvatore J
- Salvo, Jerry Di
- Lyons, Kathy
- Pivnichny, James V
- Kwei, Gloria Y
- Carella, Anthony
- Carver, Gwen
- Holmes, Karen
- Schleif, William A
- Danzeisen, Renee
- Hazuda, Daria
- Kessler, Joseph
- Lineberger, Janet
- Miller, Michael D
- Emini, Emilio A
Producer: 20040928
In:
Bioorganic & medicinal chemistry letters vol. 14
Availability: No items available.
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79.
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CCR5 antagonists: 3-(pyrrolidin-1-yl)propionic acid analogues with potent anti-HIV activity. [electronic resource] by
- Lynch, Christopher L
- Hale, Jeffrey J
- Budhu, Richard J
- Gentry, Amy L
- Finke, Paul E
- Caldwell, Charles G
- Mills, Sander G
- MacCoss, Malcolm
- Shen, Dong-Ming
- Chapman, Kevin T
- Malkowitz, Lorraine
- Springer, Martin S
- Gould, Sandra L
- DeMartino, Julie A
- Siciliano, Salvatore J
- Cascieri, Margaret A
- Carella, Anthony
- Carver, Gwen
- Holmes, Karen
- Schleif, William A
- Danzeisen, Renee
- Hazuda, Daria
- Kessler, Joseph
- Lineberger, Janet
- Miller, Michael
- Emini, Emilio
Producer: 20031126
In:
Organic letters vol. 5
Availability: No items available.
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80.
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Antagonists of human CCR5 receptor containing 4-(pyrazolyl)piperidine side chains. Part 2: Discovery of potent, selective, and orally bioavailable compounds. [electronic resource] by
- Shen, Dong-Ming
- Shu, Min
- Willoughby, Christopher A
- Shah, Shrenik
- Lynch, Christopher L
- Hale, Jeffrey J
- Mills, Sander G
- Chapman, Kevin T
- Malkowitz, Lorraine
- Springer, Martin S
- Gould, Sandra L
- DeMartino, Julie A
- Siciliano, Salvatore J
- Lyons, Kathy
- Pivnichny, James V
- Kwei, Gloria Y
- Carella, Anthony
- Carver, Gwen
- Holmes, Karen
- Schleif, William A
- Danzeisen, Renee
- Hazuda, Daria
- Kessler, Joseph
- Lineberger, Janet
- Miller, Michael D
- Emini, Emilio A
Producer: 20040928
In:
Bioorganic & medicinal chemistry letters vol. 14
Availability: No items available.
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