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61.
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Neratinib protects pancreatic beta cells in diabetes. [electronic resource] by
- Ardestani, Amin
- Li, Sijia
- Annamalai, Karthika
- Lupse, Blaz
- Geravandi, Shirin
- Dobrowolski, Aleksandra
- Yu, Shan
- Zhu, Siying
- Baguley, Tyler D
- Surakattula, Murali
- Oetjen, Janina
- Hauberg-Lotte, Lena
- Herranz, Raquel
- Awal, Sushil
- Altenhofen, Delsi
- Nguyen-Tran, Van
- Joseph, Sean
- Schultz, Peter G
- Chatterjee, Arnab K
- Rogers, Nikki
- Tremblay, Matthew S
- Shen, Weijun
- Maedler, Kathrin
Producer: 20200316
In:
Nature communications vol. 10
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62.
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Determinants of the Inhibition of DprE1 and CYP2C9 by Antitubercular Thiophenes. [electronic resource] by
- Liu, Renhe
- Lyu, Xiaoxuan
- Batt, Sarah M
- Hsu, Mei-Hui
- Harbut, Michael B
- Vilchèze, Catherine
- Cheng, Bo
- Ajayi, Kehinde
- Yang, Baiyuan
- Yang, Yun
- Guo, Hui
- Lin, Changyou
- Gan, Fei
- Wang, Chen
- Franzblau, Scott G
- Jacobs, William R
- Besra, Gurdyal S
- Johnson, Eric F
- Petrassi, Mike
- Chatterjee, Arnab K
- Fütterer, Klaus
- Wang, Feng
Producer: 20190318
In:
Angewandte Chemie (International ed. in English) vol. 56
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63.
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Repurposing isoxazoline veterinary drugs for control of vector-borne human diseases. [electronic resource] by
- Miglianico, Marie
- Eldering, Maarten
- Slater, Hannah
- Ferguson, Neil
- Ambrose, Pauline
- Lees, Rosemary S
- Koolen, Karin M J
- Pruzinova, Katerina
- Jancarova, Magdalena
- Volf, Petr
- Koenraadt, Constantianus J M
- Duerr, Hans-Peter
- Trevitt, Graham
- Yang, Baiyuan
- Chatterjee, Arnab K
- Wisler, John
- Sturm, Angelika
- Bousema, Teun
- Sauerwein, Robert W
- Schultz, Peter G
- Tremblay, Matthew S
- Dechering, Koen J
Producer: 20180918
In:
Proceedings of the National Academy of Sciences of the United States of America vol. 115
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64.
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Gene expression signatures and small-molecule compounds link a protein kinase to Plasmodium falciparum motility. [electronic resource] by
- Kato, Nobutaka
- Sakata, Tomoyo
- Breton, Ghislain
- Le Roch, Karine G
- Nagle, Advait
- Andersen, Carsten
- Bursulaya, Badry
- Henson, Kerstin
- Johnson, Jeffrey
- Kumar, Kota Arun
- Marr, Felix
- Mason, Daniel
- McNamara, Case
- Plouffe, David
- Ramachandran, Vandana
- Spooner, Muriel
- Tuntland, Tove
- Zhou, Yingyao
- Peters, Eric C
- Chatterjee, Arnab
- Schultz, Peter G
- Ward, Gary E
- Gray, Nathanael
- Harper, Jeffrey
- Winzeler, Elizabeth A
Producer: 20080910
In:
Nature chemical biology vol. 4
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65.
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Identification of inhibitors for putative malaria drug targets among novel antimalarial compounds. [electronic resource] by
- Crowther, Gregory J
- Napuli, Alberto J
- Gilligan, James H
- Gagaring, Kerstin
- Borboa, Rachel
- Francek, Carolyn
- Chen, Zhong
- Dagostino, Eleanor F
- Stockmyer, Justin B
- Wang, Yu
- Rodenbough, Philip P
- Castaneda, Lisa J
- Leibly, David J
- Bhandari, Janhavi
- Gelb, Michael H
- Brinker, Achim
- Engels, Ingo H
- Taylor, Jennifer
- Chatterjee, Arnab K
- Fantauzzi, Pascal
- Glynne, Richard J
- Van Voorhis, Wesley C
- Kuhen, Kelli L
Producer: 20110209
In:
Molecular and biochemical parasitology vol. 175
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66.
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A high-throughput screen to identify inhibitors of ATP homeostasis in non-replicating Mycobacterium tuberculosis. [electronic resource] by
- Mak, Puiying A
- Rao, Srinivasa P S
- Ping Tan, Mai
- Lin, Xiuhua
- Chyba, Jason
- Tay, Joann
- Ng, Seow Hwee
- Tan, Bee Huat
- Cherian, Joseph
- Duraiswamy, Jeyaraj
- Bifani, Pablo
- Lim, Vivian
- Lee, Boon Heng
- Ling Ma, Ngai
- Beer, David
- Thayalan, Pamela
- Kuhen, Kelli
- Chatterjee, Arnab
- Supek, Frantisek
- Glynne, Richard
- Zheng, Jun
- Boshoff, Helena I
- Barry, Clifton E
- Dick, Thomas
- Pethe, Kevin
- Camacho, Luis R
Producer: 20130517
In:
ACS chemical biology vol. 7
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67.
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Identification of a small molecule with activity against drug-resistant and persistent tuberculosis. [electronic resource] by
- Wang, Feng
- Sambandan, Dhinakaran
- Halder, Rajkumar
- Wang, Jianing
- Batt, Sarah M
- Weinrick, Brian
- Ahmad, Insha
- Yang, Pengyu
- Zhang, Yong
- Kim, John
- Hassani, Morad
- Huszar, Stanislav
- Trefzer, Claudia
- Ma, Zhenkun
- Kaneko, Takushi
- Mdluli, Khisi E
- Franzblau, Scott
- Chatterjee, Arnab K
- Johnsson, Kai
- Johnson, Kai
- Mikusova, Katarina
- Besra, Gurdyal S
- Fütterer, Klaus
- Robbins, Scott H
- Barnes, S Whitney
- Walker, John R
- Jacobs, William R
- Schultz, Peter G
Producer: 20130926
In:
Proceedings of the National Academy of Sciences of the United States of America vol. 110
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68.
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Imidazolopiperazines: lead optimization of the second-generation antimalarial agents. [electronic resource] by
- Nagle, Advait
- Wu, Tao
- Kuhen, Kelli
- Gagaring, Kerstin
- Borboa, Rachel
- Francek, Caroline
- Chen, Zhong
- Plouffe, David
- Lin, Xuena
- Caldwell, Christopher
- Ek, Jared
- Skolnik, Suzanne
- Liu, Fenghua
- Wang, Jianling
- Chang, Jonathan
- Li, Chun
- Liu, Bo
- Hollenbeck, Thomas
- Tuntland, Tove
- Isbell, John
- Chuan, Tiffany
- Alper, Philip B
- Fischli, Christoph
- Brun, Reto
- Lakshminarayana, Suresh B
- Rottmann, Matthias
- Diagana, Thierry T
- Winzeler, Elizabeth A
- Glynne, Richard
- Tully, David C
- Chatterjee, Arnab K
Producer: 20120912
In:
Journal of medicinal chemistry vol. 55
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69.
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KAI407, a potent non-8-aminoquinoline compound that kills Plasmodium cynomolgi early dormant liver stage parasites in vitro. [electronic resource] by
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- van Amsterdam, Sandra M
- McNamara, Case W
- Voorberg-van der Wel, Annemarie
- Klooster, Els J
- van den Berg, Alexander
- Remarque, Edmond J
- Plouffe, David M
- van Gemert, Geert-Jan
- Luty, Adrian
- Sauerwein, Robert
- Gagaring, Kerstin
- Borboa, Rachel
- Chen, Zhong
- Kuhen, Kelli
- Glynne, Richard J
- Chatterjee, Arnab K
- Nagle, Advait
- Roland, Jason
- Winzeler, Elizabeth A
- Leroy, Didier
- Campo, Brice
- Diagana, Thierry T
- Yeung, Bryan K S
- Thomas, Alan W
- Kocken, Clemens H M
Producer: 20141028
In:
Antimicrobial agents and chemotherapy vol. 58
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70.
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Discovery of tetrahydropyrazolopyrimidine carboxamide derivatives as potent and orally active antitubercular agents. [electronic resource] by
- Yokokawa, Fumiaki
- Wang, Gang
- Chan, Wai Ling
- Ang, Shi Hua
- Wong, Josephine
- Ma, Ida
- Rao, Srinivasa P S
- Manjunatha, Ujjini
- Lakshminarayana, Suresh B
- Herve, Maxime
- Kounde, Cyrille
- Tan, Bee Huat
- Thayalan, Pamela
- Ng, Seow Hwee
- Nanjundappa, Mahesh
- Ravindran, Sindhu
- Gee, Peck
- Tan, Maria
- Wei, Liu
- Goh, Anne
- Chen, Pei-Yu
- Lee, Kok Sin
- Zhong, Chen
- Wagner, Trixie
- Dix, Ina
- Chatterjee, Arnab K
- Pethe, Kevin
- Kuhen, Kelli
- Glynne, Richard
- Smith, Paul
- Bifani, Pablo
- Jiricek, Jan
Producer: 20140605
In:
ACS medicinal chemistry letters vol. 4
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71.
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Lead optimization of imidazopyrazines: a new class of antimalarial with activity on Plasmodium liver stages. [electronic resource] by
- Zou, Bin
- Nagle, Advait
- Chatterjee, Arnab K
- Leong, Seh Yong
- Tan, Liying Jocelyn
- Sim, Wei Lin Sandra
- Mishra, Pranab
- Guntapalli, Prasuna
- Tully, David C
- Lakshminarayana, Suresh B
- Lim, Chek Shik
- Tan, Yong Cheng
- Abas, Siti Nurdiana
- Bodenreider, Christophe
- Kuhen, Kelli L
- Gagaring, Kerstin
- Borboa, Rachel
- Chang, Jonathan
- Li, Chun
- Hollenbeck, Thomas
- Tuntland, Tove
- Zeeman, Anne-Marie
- Kocken, Clemens H M
- McNamara, Case
- Kato, Nobutaka
- Winzeler, Elizabeth A
- Yeung, Bryan K S
- Diagana, Thierry T
- Smith, Paul W
- Roland, Jason
Producer: 20140822
In:
ACS medicinal chemistry letters vol. 5
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72.
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Pyrazoleamide compounds are potent antimalarials that target Na+ homeostasis in intraerythrocytic Plasmodium falciparum. [electronic resource] by
- Vaidya, Akhil B
- Morrisey, Joanne M
- Zhang, Zhongsheng
- Das, Sudipta
- Daly, Thomas M
- Otto, Thomas D
- Spillman, Natalie J
- Wyvratt, Matthew
- Siegl, Peter
- Marfurt, Jutta
- Wirjanata, Grennady
- Sebayang, Boni F
- Price, Ric N
- Chatterjee, Arnab
- Nagle, Advait
- Stasiak, Marcin
- Charman, Susan A
- Angulo-Barturen, Iñigo
- Ferrer, Santiago
- Belén Jiménez-Díaz, María
- Martínez, María Santos
- Gamo, Francisco Javier
- Avery, Vicky M
- Ruecker, Andrea
- Delves, Michael
- Kirk, Kiaran
- Berriman, Matthew
- Kortagere, Sandhya
- Burrows, Jeremy
- Fan, Erkang
- Bergman, Lawrence W
Producer: 20151015
In:
Nature communications vol. 5
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73.
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Imidazolopiperazines: hit to lead optimization of new antimalarial agents. [electronic resource] by
- Wu, Tao
- Nagle, Advait
- Kuhen, Kelli
- Gagaring, Kerstin
- Borboa, Rachel
- Francek, Caroline
- Chen, Zhong
- Plouffe, David
- Goh, Anne
- Lakshminarayana, Suresh B
- Wu, Jeanette
- Ang, Hui Qing
- Zeng, Peiting
- Kang, Min Low
- Tan, William
- Tan, Maria
- Ye, Nicole
- Lin, Xuena
- Caldwell, Christopher
- Ek, Jared
- Skolnik, Suzanne
- Liu, Fenghua
- Wang, Jianling
- Chang, Jonathan
- Li, Chun
- Hollenbeck, Thomas
- Tuntland, Tove
- Isbell, John
- Fischli, Christoph
- Brun, Reto
- Rottmann, Matthias
- Dartois, Veronique
- Keller, Thomas
- Diagana, Thierry
- Winzeler, Elizabeth
- Glynne, Richard
- Tully, David C
- Chatterjee, Arnab K
Producer: 20111010
In:
Journal of medicinal chemistry vol. 54
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74.
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Imaging of Plasmodium liver stages to drive next-generation antimalarial drug discovery. [electronic resource] by
- Meister, Stephan
- Plouffe, David M
- Kuhen, Kelli L
- Bonamy, Ghislain M C
- Wu, Tao
- Barnes, S Whitney
- Bopp, Selina E
- Borboa, Rachel
- Bright, A Taylor
- Che, Jianwei
- Cohen, Steve
- Dharia, Neekesh V
- Gagaring, Kerstin
- Gettayacamin, Montip
- Gordon, Perry
- Groessl, Todd
- Kato, Nobutaka
- Lee, Marcus C S
- McNamara, Case W
- Fidock, David A
- Nagle, Advait
- Nam, Tae-gyu
- Richmond, Wendy
- Roland, Jason
- Rottmann, Matthias
- Zhou, Bin
- Froissard, Patrick
- Glynne, Richard J
- Mazier, Dominique
- Sattabongkot, Jetsumon
- Schultz, Peter G
- Tuntland, Tove
- Walker, John R
- Zhou, Yingyao
- Chatterjee, Arnab
- Diagana, Thierry T
- Winzeler, Elizabeth A
Producer: 20120125
In:
Science (New York, N.Y.) vol. 334
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75.
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Indolcarboxamide is a preclinical candidate for treating multidrug-resistant tuberculosis. [electronic resource] by
- Rao, Srinivasa P S
- Lakshminarayana, Suresh B
- Kondreddi, Ravinder R
- Herve, Maxime
- Camacho, Luis R
- Bifani, Pablo
- Kalapala, Sarath K
- Jiricek, Jan
- Ma, Ng L
- Tan, Bee H
- Ng, Seow H
- Nanjundappa, Mahesh
- Ravindran, Sindhu
- Seah, Peck G
- Thayalan, Pamela
- Lim, Siao H
- Lee, Boon H
- Goh, Anne
- Barnes, Whitney S
- Chen, Zhong
- Gagaring, Kerstin
- Chatterjee, Arnab K
- Pethe, Kevin
- Kuhen, Kelli
- Walker, John
- Feng, Gu
- Babu, Sreehari
- Zhang, Lijun
- Blasco, Francesca
- Beer, David
- Weaver, Margaret
- Dartois, Veronique
- Glynne, Richard
- Dick, Thomas
- Smith, Paul W
- Diagana, Thierry T
- Manjunatha, Ujjini H
Producer: 20140728
In:
Science translational medicine vol. 5
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76.
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A chemical genetic screen in Mycobacterium tuberculosis identifies carbon-source-dependent growth inhibitors devoid of in vivo efficacy. [electronic resource] by
- Pethe, Kevin
- Sequeira, Patricia C
- Agarwalla, Sanjay
- Rhee, Kyu
- Kuhen, Kelli
- Phong, Wai Yee
- Patel, Viral
- Beer, David
- Walker, John R
- Duraiswamy, Jeyaraj
- Jiricek, Jan
- Keller, Thomas H
- Chatterjee, Arnab
- Tan, Mai Ping
- Ujjini, Manjunatha
- Rao, Srinivasa P S
- Camacho, Luis
- Bifani, Pablo
- Mak, Puiying A
- Ma, Ida
- Barnes, S Whitney
- Chen, Zhong
- Plouffe, David
- Thayalan, Pamela
- Ng, Seow Hwee
- Au, Melvin
- Lee, Boon Heng
- Tan, Bee Huat
- Ravindran, Sindhu
- Nanjundappa, Mahesh
- Lin, Xiuhua
- Goh, Anne
- Lakshminarayana, Suresh B
- Shoen, Carolyn
- Cynamon, Michael
- Kreiswirth, Barry
- Dartois, Veronique
- Peters, Eric C
- Glynne, Richard
- Brenner, Sydney
- Dick, Thomas
Producer: 20110701
In:
Nature communications vol. 1
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77.
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KAF156 is an antimalarial clinical candidate with potential for use in prophylaxis, treatment, and prevention of disease transmission. [electronic resource] by
- Kuhen, Kelli L
- Chatterjee, Arnab K
- Rottmann, Matthias
- Gagaring, Kerstin
- Borboa, Rachel
- Buenviaje, Jennifer
- Chen, Zhong
- Francek, Carolyn
- Wu, Tao
- Nagle, Advait
- Barnes, S Whitney
- Plouffe, David
- Lee, Marcus C S
- Fidock, David A
- Graumans, Wouter
- van de Vegte-Bolmer, Marga
- van Gemert, Geert J
- Wirjanata, Grennady
- Sebayang, Boni
- Marfurt, Jutta
- Russell, Bruce
- Suwanarusk, Rossarin
- Price, Ric N
- Nosten, Francois
- Tungtaeng, Anchalee
- Gettayacamin, Montip
- Sattabongkot, Jetsumon
- Taylor, Jennifer
- Walker, John R
- Tully, David
- Patra, Kailash P
- Flannery, Erika L
- Vinetz, Joseph M
- Renia, Laurent
- Sauerwein, Robert W
- Winzeler, Elizabeth A
- Glynne, Richard J
- Diagana, Thierry T
Producer: 20150909
In:
Antimicrobial agents and chemotherapy vol. 58
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78.
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Targeting Plasmodium PI(4)K to eliminate malaria. [electronic resource] by
- McNamara, Case W
- Lee, Marcus Cs
- Lim, Chek Shik
- Lim, Siau Hoi
- Roland, Jason
- Simon, Oliver
- Yeung, Bryan Ks
- Chatterjee, Arnab K
- McCormack, Susan L
- Manary, Micah J
- Zeeman, Anne-Marie
- Dechering, Koen J
- Kumar, Tr Santha
- Henrich, Philipp P
- Gagaring, Kerstin
- Ibanez, Maureen
- Kato, Nobutaka
- Kuhen, Kelli L
- Fischli, Christoph
- Nagle, Advait
- Rottmann, Matthias
- Plouffe, David M
- Bursulaya, Badry
- Meister, Stephan
- Rameh, Lucia
- Trappe, Joerg
- Haasen, Dorothea
- Timmerman, Martijn
- Sauerwein, Robert W
- Suwanarusk, Rossarin
- Russell, Bruce
- Renia, Laurent
- Nosten, Francois
- Tully, David C
- Kocken, Clemens Hm
- Glynne, Richard J
- Bodenreider, Christophe
- Fidock, David A
- Diagana, Thierry T
- Winzeler, Elizabeth A
Producer: 20140107
In:
Nature vol. 504
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79.
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Discovery of short-course antiwolbachial quinazolines for elimination of filarial worm infections. [electronic resource] by
- Bakowski, Malina A
- Shiroodi, Roohollah Kazem
- Liu, Renhe
- Olejniczak, Jason
- Yang, Baiyuan
- Gagaring, Kerstin
- Guo, Hui
- White, Pamela M
- Chappell, Laura
- Debec, Alain
- Landmann, Frédéric
- Dubben, Bettina
- Lenz, Franziska
- Struever, Dominique
- Ehrens, Alexandra
- Frohberger, Stefan J
- Sjoberg, Hanna
- Pionnier, Nicolas
- Murphy, Emma
- Archer, John
- Steven, Andrew
- Chunda, Valerine C
- Fombad, Fanny F
- Chounna, Patrick W
- Njouendou, Abdel J
- Metuge, Haelly M
- Ndzeshang, Bertrand L
- Gandjui, Narcisse V
- Akumtoh, Desmond N
- Kwenti, Tayong D B
- Woods, Ashley K
- Joseph, Sean B
- Hull, Mitchell V
- Xiong, Wen
- Kuhen, Kelli L
- Taylor, Mark J
- Wanji, Samuel
- Turner, Joseph D
- Hübner, Marc P
- Hoerauf, Achim
- Chatterjee, Arnab K
- Roland, Jason
- Tremblay, Matt S
- Schultz, Peter G
- Sullivan, William
- Chu, Xin-Jie
- Petrassi, H Michael
- McNamara, Case W
Producer: 20200714
In:
Science translational medicine vol. 11
Availability: No items available.
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