Results
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541.
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542.
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543.
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544.
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545.
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546.
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547.
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548.
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549.
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550.
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Discovery of sodium R-(+)-4-{2-[5-(2-fluoro-3-methoxyphenyl)-3-(2-fluoro-6-[trifluoromethyl]benzyl)-4-methyl-2,6-dioxo-3,6-dihydro-2H-pyrimidin-1-yl]-1-phenylethylamino}butyrate (elagolix), a potent and orally available nonpeptide antagonist of the human gonadotropin-releasing hormone receptor. [electronic resource] by
- Chen, Chen
- Wu, Dongpei
- Guo, Zhiqiang
- Xie, Qiu
- Reinhart, Greg J
- Madan, Ajay
- Wen, Jenny
- Chen, Takung
- Huang, Charles Q
- Chen, Mi
- Chen, Yongsheng
- Tucci, Fabio C
- Rowbottom, Martin
- Pontillo, Joseph
- Zhu, Yun-Fei
- Wade, Warren
- Saunders, John
- Bozigian, Haig
- Struthers, R Scott
Producer: 20090403
In:
Journal of medicinal chemistry vol. 51
Availability: No items available.
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551.
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552.
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553.
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Discovery of 1-{4-[1-(2,6-difluorobenzyl)-5-[(dimethylamino)methyl]-3-(6-methoxypyridazin-3-yl)-2,4-dioxo-1,2,3,4-tetrahydrothieno[2,3-d]pyrimidin-6-yl]phenyl}-3-methoxyurea (TAK-385) as a potent, orally active, non-peptide antagonist of the human gonadotropin-releasing hormone receptor. [electronic resource] by
- Miwa, Kazuhiro
- Hitaka, Takenori
- Imada, Takashi
- Sasaki, Satoshi
- Yoshimatsu, Mie
- Kusaka, Masami
- Tanaka, Akira
- Nakata, Daisuke
- Furuya, Shuichi
- Endo, Satoshi
- Hamamura, Kazumasa
- Kitazaki, Tomoyuki
Producer: 20111010
In:
Journal of medicinal chemistry vol. 54
Availability: No items available.
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554.
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555.
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556.
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557.
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558.
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559.
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560.
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