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Cell viability assessed in a reproducible model of human osteoblasts derived from human adipose-derived stem cells. [electronic resource] by
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- Deprá, Igor C
- Mathias, Lucas S
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- Rodrigues, Bruna M
- Tilli, Helena P
- Coscrato, Virgínia E
- Costa, Sarah M B
- Mazeto, Gláucia M F S
- Fernandes, Célio J C
- Zambuzzi, Willian F
- Saraiva, Patrícia P
- Maria, Durvanei A
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Producer: 20180725
In:
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From a novel HTS hit to potent, selective, and orally bioavailable KDM5 inhibitors. [electronic resource] by
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- Ortwine, Daniel F
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- Vinogradova, Maia
- Kiefer, James R
- Mauer, Till
- Gehling, Victor S
- Harmange, Jean-Christophe
- Cummings, Richard
- Lai, Tommy
- Liao, Jiangpeng
- Zheng, Xiaoping
- Liu, Yichin
- Gustafson, Amy
- Van der Porten, Erica
- Mao, Weifeng
- Liederer, Bianca M
- Deshmukh, Gauri
- An, Le
- Ran, Yingqing
- Classon, Marie
- Trojer, Patrick
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Producer: 20170818
In:
Bioorganic & medicinal chemistry letters vol. 27
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RIP1 inhibition blocks inflammatory diseases but not tumor growth or metastases. [electronic resource] by
- Patel, Snahel
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- Zhang, Juan
- Dugger, Debra L
- Wickliffe, Kate E
- Maltzman, Allie
- Sujatha-Bhaskar, Swathi
- Bir Kohli, Pawan
- Ramaswamy, Sreema
- Deshmukh, Gauri
- Liederer, Bianca M
- Fong, Rina
- Hamilton, Greg
- Lupardus, Patrick
- Caplazi, Patrick
- Lee, Wyne P
- van Lookeren Campagne, Menno
- Johnson, Adam
- McKenzie, Brent S
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- Newton, Kim
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Structure-based discovery of novel amide-containing nicotinamide phosphoribosyltransferase (nampt) inhibitors. [electronic resource] by
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- Caligiuri, Maureen
- Clodfelter, Karl H
- Han, Bingsong
- Ho, Yen-Ching
- Kley, Nikolai
- Lin, Jian
- Reynolds, Dominic J
- Sharma, Geeta
- Smith, Chase C
- Wang, Zhongguo
- Dragovich, Peter S
- Gunzner-Toste, Janet
- Liederer, Bianca M
- Ly, Justin
- O'Brien, Thomas
- Oh, Angela
- Wang, Leslie
- Wang, Weiru
- Xiao, Yang
- Zak, Mark
- Zhao, Guiling
- Yuen, Po-Wai
- Bair, Kenneth W
Producer: 20131029
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Frequency of the Types of Alopecia at Twenty-Two Specialist Hair Clinics: A Multicenter Study. [electronic resource] by
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- Gavazzoni Dias, Maria Fernanda Reis
- Grimalt, Ramon
- Guzmán-Sánchez, Daniela
- Harries, Matthew
- Ho, Anthony
- Holmes, Susan
- Larrondo, Jorge
- Mosam, Anisa
- Oliveira-Soares, Rui
- Pinto, Giselle M
- Piraccini, Bianca M
- Pirmez, Rodrigo
- De la Rosa Carrillo, Daniel
- Rudnicka, Lidia
- Shapiro, Jerry
- Sinclair, Rodney
- Tosti, Antonella
- Trüeb, Ralph M
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Publication details: Skin appendage disorders Aug 2019
In:
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526.
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GluN2A NMDA Receptor Enhancement Improves Brain Oscillations, Synchrony, and Cognitive Functions in Dravet Syndrome and Alzheimer's Disease Models. [electronic resource] by
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- Ma, Keran
- Elstrott, Justin
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- Khan, Abdullah S
- Simms, Jeffrey
- Liu, Benjamin
- Kim, Thomas A
- Yu, Gui-Qiu
- Chen, Yelin
- Wang, Tzu-Ming
- Jiang, Zhiyu
- Liederer, Bianca M
- Deshmukh, Gauri
- Solanoy, Hilda
- Chan, Connie
- Sellers, Benjamin D
- Volgraf, Matthew
- Schwarz, Jacob B
- Hackos, David H
- Weimer, Robby M
- Sheng, Morgan
- Gill, T Michael
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Identification of nicotinamide phosphoribosyltransferase (NAMPT) inhibitors with no evidence of CYP3A4 time-dependent inhibition and improved aqueous solubility. [electronic resource] by
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- Yuen, Po-Wai
- Bair, Kenneth W
- Baumeister, Timm
- Buckmelter, Alexandre J
- Clodfelter, Karl H
- Cheng, Eric
- Crocker, Lisa
- Fu, Bang
- Han, Bingsong
- Li, Guangkun
- Ho, Yen-Ching
- Lin, Jian
- Liu, Xiongcai
- Ly, Justin
- O'Brien, Thomas
- Reynolds, Dominic J
- Skelton, Nicholas
- Smith, Chase C
- Tay, Suzanne
- Wang, Weiru
- Wang, Zhongguo
- Xiao, Yang
- Zhang, Lei
- Zhao, Guiling
- Zheng, Xiaozhang
- Dragovich, Peter S
Producer: 20150915
In:
Bioorganic & medicinal chemistry letters vol. 25
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528.
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Fragment-based identification of amides derived from trans-2-(pyridin-3-yl)cyclopropanecarboxylic acid as potent inhibitors of human nicotinamide phosphoribosyltransferase (NAMPT). [electronic resource] by
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- Zheng, Xiaozhang
- Skelton, Nicholas J
- Wang, Weiru
- Bravo, Brandon J
- Bair, Kenneth W
- Baumeister, Timm
- Cheng, Eric
- Crocker, Lisa
- Feng, Yezhen
- Gunzner-Toste, Janet
- Ho, Yen-Ching
- Hua, Rongbao
- Liederer, Bianca M
- Liu, Yongbo
- Ma, Xiaolei
- O'Brien, Thomas
- Oeh, Jason
- Sampath, Deepak
- Shen, Youming
- Wang, Chengcheng
- Wang, Leslie
- Wu, Hongxing
- Xiao, Yang
- Yuen, Po-wai
- Zak, Mark
- Zhao, Guiling
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Producer: 20140415
In:
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Discovery of potent and efficacious urea-containing nicotinamide phosphoribosyltransferase (NAMPT) inhibitors with reduced CYP2C9 inhibition properties. [electronic resource] by
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- Baumeister, Timm
- Buckmelter, Alexandre J
- Caligiuri, Maureen
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- Fu, Bang
- Han, Bingsong
- Ho, Yen-Ching
- Kley, Nikolai
- Liang, Xiaorong
- Liederer, Bianca M
- Lin, Jian
- Mukadam, Sophie
- O'Brien, Thomas
- Oh, Angela
- Reynolds, Dominic J
- Sharma, Geeta
- Skelton, Nicholas
- Smith, Chase C
- Sodhi, Jasleen
- Wang, Weiru
- Wang, Zhongguo
- Xiao, Yang
- Yuen, Po-wai
- Zak, Mark
- Zhang, Lei
- Zheng, Xiaozhang
- Bair, Kenneth W
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Producer: 20140424
In:
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Loss-of-function mutations in PTPN11 cause metachondromatosis, but not Ollier disease or Maffucci syndrome. [electronic resource] by
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- Campos-Xavier, Belinda
- Bonafé, Luisa
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- Cormier-Daire, Valerie
- Bovée, Judith V
- Pansuriya, Twinkal C
- de Sousa, Sérgio B
- Savarirayan, Ravi
- Andreucci, Elena
- Vikkula, Miikka
- Garavelli, Livia
- Pottinger, Caroline
- Ogino, Toshihiko
- Sakai, Akinori
- Regazzoni, Bianca M
- Wuyts, Wim
- Sangiorgi, Luca
- Pedrini, Elena
- Zhu, Mei
- Kozakewich, Harry P
- Kasser, James R
- Seidman, Jon G
- Kurek, Kyle C
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Producer: 20110812
In:
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Pragmatic trial of a multidisciplinary lung cancer care model in a community healthcare setting: study design, implementation evaluation, and baseline clinical results. [electronic resource] by
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- Jackson, Bianca M
- Berryman, Courtney L
- Faris, Nicholas R
- Ray, Meredith A
- Meadows, Meghan
- Patel, Anita A
- Roark, Kristina S
- Kedia, Satish K
- DeBon, Margaret M
- Crossley, Fayre J
- Oliver, Georgia
- McHugh, Laura M
- Hastings, Willeen
- Osborne, Orion
- Osborne, Jackie
- Ill, Toni
- Ill, Mark
- Jones, Wynett
- Lee, Hyo K
- Signore, Raymond S
- Fox, Roy C
- Li, Jingshan
- Robbins, Edward T
- Ward, Kenneth D
- Klesges, Lisa M
- Osarogiagbon, Raymond U
Publication details: Translational lung cancer research Feb 2018
In:
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Discovery and preclinical pharmacology of a selective ATP-competitive Akt inhibitor (GDC-0068) for the treatment of human tumors. [electronic resource] by
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- Xiao, Dengming
- Kallan, Nicholas C
- Schlachter, Stephen
- Mitchell, Ian S
- Spencer, Keith L
- Banka, Anna L
- Wallace, Eli M
- Gloor, Susan L
- Martinson, Matthew
- Woessner, Richard D
- Vigers, Guy P A
- Brandhuber, Barbara J
- Liang, Jun
- Safina, Brian S
- Li, Jun
- Zhang, Birong
- Chabot, Christine
- Do, Steven
- Lee, Leslie
- Oeh, Jason
- Sampath, Deepak
- Lee, Brian B
- Lin, Kui
- Liederer, Bianca M
- Skelton, Nicholas J
Producer: 20121204
In:
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533.
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Discovery of GluN2A-Selective NMDA Receptor Positive Allosteric Modulators (PAMs): Tuning Deactivation Kinetics via Structure-Based Design. [electronic resource] by
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- Sellers, Benjamin D
- Jiang, Yu
- Wu, Guosheng
- Ly, Cuong Q
- Villemure, Elisia
- Pastor, Richard M
- Yuen, Po-wai
- Lu, Aijun
- Luo, Xifeng
- Liu, Mingcui
- Zhang, Shun
- Sun, Liang
- Fu, Yuhong
- Lupardus, Patrick J
- Wallweber, Heidi J A
- Liederer, Bianca M
- Deshmukh, Gauri
- Plise, Emile
- Tay, Suzanne
- Reynen, Paul
- Herrington, James
- Gustafson, Amy
- Liu, Yichin
- Dirksen, Akim
- Dietz, Matthias G A
- Liu, Yanzhou
- Wang, Tzu-Ming
- Hanson, Jesse E
- Hackos, David
- Scearce-Levie, Kimberly
- Schwarz, Jacob B
Producer: 20160823
In:
Journal of medicinal chemistry vol. 59
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534.
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Mutations in SMAD3 cause a syndromic form of aortic aneurysms and dissections with early-onset osteoarthritis. [electronic resource] by
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- Oldenburg, Rogier A
- Pals, Gerard
- Roos-Hesselink, Jolien W
- de Graaf, Bianca M
- Verhagen, Judith M A
- Hoedemaekers, Yvonne M
- Willemsen, Rob
- Severijnen, Lies-Anne
- Venselaar, Hanka
- Vriend, Gert
- Pattynama, Peter M
- Collée, Margriet
- Majoor-Krakauer, Danielle
- Poldermans, Don
- Frohn-Mulder, Ingrid M E
- Micha, Dimitra
- Timmermans, Janneke
- Hilhorst-Hofstee, Yvonne
- Bierma-Zeinstra, Sita M
- Willems, Patrick J
- Kros, Johan M
- Oei, Edwin H G
- Oostra, Ben A
- Wessels, Marja W
- Bertoli-Avella, Aida M
Producer: 20110331
In:
Nature genetics vol. 43
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535.
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Identification of amides derived from 1H-pyrazolo[3,4-b]pyridine-5-carboxylic acid as potent inhibitors of human nicotinamide phosphoribosyltransferase (NAMPT). [electronic resource] by
- Zheng, Xiaozhang
- Bair, Kenneth W
- Bauer, Paul
- Baumeister, Timm
- Bowman, Krista K
- Buckmelter, Alexandre J
- Caligiuri, Maureen
- Clodfelter, Karl H
- Feng, Yezhen
- Han, Bingsong
- Ho, Yen-Ching
- Kley, Nikolai
- Li, Hong
- Liang, Xiaorong
- Liederer, Bianca M
- Lin, Jian
- Ly, Justin
- O'Brien, Thomas
- Oeh, Jason
- Oh, Angela
- Reynolds, Dominic J
- Sampath, Deepak
- Sharma, Geeta
- Skelton, Nicholas
- Smith, Chase C
- Tremayne, Jarrod
- Wang, Leslie
- Wang, Weiru
- Wang, Zhongguo
- Wu, Hongxing
- Wu, Jiansheng
- Xiao, Yang
- Yang, Guangxing
- Yuen, Po-wai
- Zak, Mark
- Dragovich, Peter S
Producer: 20140505
In:
Bioorganic & medicinal chemistry letters vol. 23
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NPHP4 variants are associated with pleiotropic heart malformations. [electronic resource] by
- French, Vanessa M
- van de Laar, Ingrid M B H
- Wessels, Marja W
- Rohe, Christan
- Roos-Hesselink, Jolien W
- Wang, Guangliang
- Frohn-Mulder, Ingrid M E
- Severijnen, Lies-Anne
- de Graaf, Bianca M
- Schot, Rachel
- Breedveld, Guido
- Mientjes, Edwin
- van Tienhoven, Marianne
- Jadot, Elodie
- Jiang, Zhengxin
- Verkerk, Annemieke
- Swagemakers, Sigrid
- Venselaar, Hanka
- Rahimi, Zohreh
- Najmabadi, Hossein
- Meijers-Heijboer, Hanne
- de Graaff, Esther
- Helbing, Wim A
- Willemsen, Rob
- Devriendt, Koen
- Belmont, John W
- Oostra, Ben A
- Amack, Jeffrey D
- Bertoli-Avella, Aida M
Producer: 20120813
In:
Circulation research vol. 110
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Phenotypic spectrum of the SMAD3-related aneurysms-osteoarthritis syndrome. [electronic resource] by
- van de Laar, Ingrid M B H
- van der Linde, Denise
- Oei, Edwin H G
- Bos, Pieter K
- Bessems, Johannes H
- Bierma-Zeinstra, Sita M
- van Meer, Belle L
- Pals, Gerard
- Oldenburg, Rogier A
- Bekkers, Jos A
- Moelker, Adriaan
- de Graaf, Bianca M
- Matyas, Gabor
- Frohn-Mulder, Ingrid M E
- Timmermans, Janneke
- Hilhorst-Hofstee, Yvonne
- Cobben, Jan M
- Bruggenwirth, Hennie T
- van Laer, Lut
- Loeys, Bart
- De Backer, Julie
- Coucke, Paul J
- Dietz, Harry C
- Willems, Patrick J
- Oostra, Ben A
- De Paepe, Anne
- Roos-Hesselink, Jolien W
- Bertoli-Avella, Aida M
- Wessels, Marja W
Producer: 20120410
In:
Journal of medical genetics vol. 49
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Genomic and Phenotypic Characterization of a Broad Panel of Patient-Derived Xenografts Reflects the Diversity of Glioblastoma. [electronic resource] by
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- Remonde, Dioval
- Schroeder, Mark A
- Mladek, Ann C
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- Kollmeyer, Thomas M
- Grove, Rebecca
- Peng, Sen
- Carlson, Brett L
- Ma, Daniel J
- Sarkar, Gobinda
- Evers, Lisa
- Decker, Paul A
- Yan, Huihuang
- Dhruv, Harshil D
- Berens, Michael E
- Wang, Qianghu
- Marin, Bianca M
- Klee, Eric W
- Califano, Andrea
- LaChance, Daniel H
- Eckel-Passow, Jeanette E
- Verhaak, Roel G
- Sulman, Erik P
- Burns, Terry C
- Meyer, Fredrick B
- O'Neill, Brian P
- Tran, Nhan L
- Giannini, Caterina
- Jenkins, Robert B
- Parney, Ian F
- Sarkaria, Jann N
Producer: 20210104
In:
Clinical cancer research : an official journal of the American Association for Cancer Research vol. 26
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Genome Sequence of Lactococcus lactis subsp. lactis NCDO 2118, a GABA-Producing Strain. [electronic resource] by
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- Ramos, Rommel T J
- Sá, Pablo H C G
- Carneiro, Adriana R
- Miranda, Fábio
- Freire, Matheus
- Renan, Wendel
- Júnior, Alberto F O
- Santos, Anderson R
- Pinto, Anne C
- Souza, Bianca M
- Castro, Camila P
- Diniz, Carlos A A
- Rocha, Clarissa S
- Mariano, Diego C B
- de Aguiar, Edgar L
- Folador, Edson L
- Barbosa, Eudes G V
- Aburjaile, Flavia F
- Gonçalves, Lucas A
- Guimarães, Luís C
- Azevedo, Marcela
- Agresti, Pamela C M
- Silva, Renata F
- Tiwari, Sandeep
- Almeida, Sintia S
- Hassan, Syed S
- Pereira, Vanessa B
- Abreu, Vinicius A C
- Pereira, Ulisses P
- Dorella, Fernanda A
- Carvalho, Alex F
- Pereira, Felipe L
- Leal, Carlos A G
- Figueiredo, Henrique C P
- Silva, Artur
- Miyoshi, Anderson
- Azevedo, Vasco
Producer: 20141003
In:
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Mutations in a TGF-β ligand, TGFB3, cause syndromic aortic aneurysms and dissections. [electronic resource] by
- Bertoli-Avella, Aida M
- Gillis, Elisabeth
- Morisaki, Hiroko
- Verhagen, Judith M A
- de Graaf, Bianca M
- van de Beek, Gerarda
- Gallo, Elena
- Kruithof, Boudewijn P T
- Venselaar, Hanka
- Myers, Loretha A
- Laga, Steven
- Doyle, Alexander J
- Oswald, Gretchen
- van Cappellen, Gert W A
- Yamanaka, Itaru
- van der Helm, Robert M
- Beverloo, Berna
- de Klein, Annelies
- Pardo, Luba
- Lammens, Martin
- Evers, Christina
- Devriendt, Koenraad
- Dumoulein, Michiel
- Timmermans, Janneke
- Bruggenwirth, Hennie T
- Verheijen, Frans
- Rodrigus, Inez
- Baynam, Gareth
- Kempers, Marlies
- Saenen, Johan
- Van Craenenbroeck, Emeline M
- Minatoya, Kenji
- Matsukawa, Ritsu
- Tsukube, Takuro
- Kubo, Noriaki
- Hofstra, Robert
- Goumans, Marie Jose
- Bekkers, Jos A
- Roos-Hesselink, Jolien W
- van de Laar, Ingrid M B H
- Dietz, Harry C
- Van Laer, Lut
- Morisaki, Takayuki
- Wessels, Marja W
- Loeys, Bart L
Producer: 20150604
In:
Journal of the American College of Cardiology vol. 65
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