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Discovery of N-[(1S,2S)-3-(4-Chlorophenyl)-2- (3-cyanophenyl)-1-methylpropyl]-2-methyl-2- {[5-(trifluoromethyl)pyridin-2-yl]oxy}propanamide (MK-0364), a novel, acyclic cannabinoid-1 receptor inverse agonist for the treatment of obesity. [electronic resource] by
- Lin, Linus S
- Lanza, Thomas J
- Jewell, James P
- Liu, Ping
- Shah, Shrenik K
- Qi, Hongbo
- Tong, Xinchun
- Wang, Junying
- Xu, Suoyu S
- Fong, Tung M
- Shen, Chun-Pyn
- Lao, Julie
- Xiao, Jing Chen
- Shearman, Lauren P
- Stribling, D Sloan
- Rosko, Kimberly
- Strack, Alison
- Marsh, Donald J
- Feng, Yue
- Kumar, Sanjeev
- Samuel, Koppara
- Yin, Wenji
- Van der Ploeg, Lex H T
- Goulet, Mark T
- Hagmann, William K
Producer: 20070202
In:
Journal of medicinal chemistry vol. 49
Availability: No items available.
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