Results
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41.
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The discovery and optimization of aminooxadiazoles as potent Pim kinase inhibitors. [electronic resource] by
- Wurz, Ryan P
- Pettus, Liping H
- Jackson, Claire
- Wu, Bin
- Wang, Hui-Ling
- Herberich, Brad
- Cee, Victor
- Lanman, Brian A
- Reed, Anthony B
- Chavez, Frank
- Nixey, Thomas
- Laszlo, Jimmy
- Wang, Paul
- Nguyen, Yen
- Sastri, Christine
- Guerrero, Nadia
- Winston, Jeff
- Lipford, J Russell
- Lee, Matthew R
- Andrews, Kristin L
- Mohr, Christopher
- Xu, Yang
- Zhou, Yihong
- Reid, Darren L
- Tasker, Andrew S
Producer: 20151015
In:
Bioorganic & medicinal chemistry letters vol. 25
Availability: No items available.
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42.
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Discovery and Optimization of Macrocyclic Quinoxaline-pyrrolo-dihydropiperidinones as Potent Pim-1/2 Kinase Inhibitors. [electronic resource] by
- Cee, Victor J
- Chavez, Frank
- Herberich, Bradley
- Lanman, Brian A
- Pettus, Liping H
- Reed, Anthony B
- Wu, Bin
- Wurz, Ryan P
- Andrews, Kristin L
- Chen, Jie
- Hickman, Dean
- Laszlo, Jimmy
- Lee, Matthew R
- Guerrero, Nadia
- Mattson, Bethany K
- Nguyen, Yen
- Mohr, Christopher
- Rex, Karen
- Sastri, Christine E
- Wang, Paul
- Wu, Qiong
- Wu, Tian
- Xu, Yang
- Zhou, Yihong
- Winston, Jeffrey T
- Lipford, J Russell
- Tasker, Andrew S
- Wang, Hui-Ling
Producer: 20160420
In:
ACS medicinal chemistry letters vol. 7
Availability: No items available.
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43.
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Evaluation of a series of naphthamides as potent, orally active vascular endothelial growth factor receptor-2 tyrosine kinase inhibitors. [electronic resource] by
- Weiss, Matthew M
- Harmange, Jean-Christophe
- Polverino, Anthony J
- Bauer, David
- Berry, Loren
- Berry, Virginia
- Borg, George
- Bready, James
- Chen, Danlin
- Choquette, Deborah
- Coxon, Angela
- DeMelfi, Tom
- Doerr, Nicholas
- Estrada, Juan
- Flynn, Julie
- Graceffa, Russell F
- Harriman, Shawn P
- Kaufman, Stephen
- La, Daniel S
- Long, Alexander
- Neervannan, Sesha
- Patel, Vinod F
- Potashman, Michele
- Regal, Kelly
- Roveto, Phillip M
- Schrag, Michael L
- Starnes, Charlie
- Tasker, Andrew
- Teffera, Yohannes
- Whittington, Douglas A
- Zanon, Roger
Producer: 20080611
In:
Journal of medicinal chemistry vol. 51
Availability: No items available.
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44.
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Naphthamides as novel and potent vascular endothelial growth factor receptor tyrosine kinase inhibitors: design, synthesis, and evaluation. [electronic resource] by
- Harmange, Jean-Christophe
- Weiss, Matthew M
- Germain, Julie
- Polverino, Anthony J
- Borg, George
- Bready, James
- Chen, Danlin
- Choquette, Deborah
- Coxon, Angela
- DeMelfi, Tom
- DiPietro, Lucian
- Doerr, Nicholas
- Estrada, Juan
- Flynn, Julie
- Graceffa, Russell F
- Harriman, Shawn P
- Kaufman, Stephen
- La, Daniel S
- Long, Alexander
- Martin, Matthew W
- Neervannan, Sesha
- Patel, Vinod F
- Potashman, Michele
- Regal, Kelly
- Roveto, Phillip M
- Schrag, Michael L
- Starnes, Charlie
- Tasker, Andrew
- Teffera, Yohannes
- Wang, Ling
- White, Ryan D
- Whittington, Douglas A
- Zanon, Roger
Producer: 20080611
In:
Journal of medicinal chemistry vol. 51
Availability: No items available.
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45.
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Discovery and Optimization of Quinazolinone-pyrrolopyrrolones as Potent and Orally Bioavailable Pan-Pim Kinase Inhibitors. [electronic resource] by
- Pettus, Liping H
- Andrews, Kristin L
- Booker, Shon K
- Chen, Jie
- Cee, Victor J
- Chavez, Frank
- Chen, Yuping
- Eastwood, Heather
- Guerrero, Nadia
- Herberich, Bradley
- Hickman, Dean
- Lanman, Brian A
- Laszlo, Jimmy
- Lee, Matthew R
- Lipford, J Russell
- Mattson, Bethany
- Mohr, Christopher
- Nguyen, Yen
- Norman, Mark H
- Powers, David
- Reed, Anthony B
- Rex, Karen
- Sastri, Christine
- Tamayo, Nuria
- Wang, Paul
- Winston, Jeffrey T
- Wu, Bin
- Wu, Tian
- Wurz, Ryan P
- Xu, Yang
- Zhou, Yihong
- Tasker, Andrew S
- Wang, Hui-Ling
Producer: 20170529
In:
Journal of medicinal chemistry vol. 59
Availability: No items available.
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46.
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Discovery of ( R)-8-(6-Methyl-4-oxo-1,4,5,6-tetrahydropyrrolo[3,4- b]pyrrol-2-yl)-3-(1-methylcyclopropyl)-2-((1-methylcyclopropyl)amino)quinazolin-4(3 H)-one, a Potent and Selective Pim-1/2 Kinase Inhibitor for Hematological Malignancies. [electronic resource] by
- Wang, Hui-Ling
- Andrews, Kristin L
- Booker, Shon K
- Canon, Jude
- Cee, Victor J
- Chavez, Frank
- Chen, Yuping
- Eastwood, Heather
- Guerrero, Nadia
- Herberich, Brad
- Hickman, Dean
- Lanman, Brian A
- Laszlo, Jimmy
- Lee, Matthew R
- Lipford, J Russell
- Mattson, Bethany
- Mohr, Christopher
- Nguyen, Yen
- Norman, Mark H
- Pettus, Liping H
- Powers, David
- Reed, Anthony B
- Rex, Karen
- Sastri, Christine
- Tamayo, Nuria
- Wang, Paul
- Winston, Jeffrey T
- Wu, Bin
- Wu, Qiong
- Wu, Tian
- Wurz, Ryan P
- Xu, Yang
- Zhou, Yihong
- Tasker, Andrew S
Producer: 20200303
In:
Journal of medicinal chemistry vol. 62
Availability: No items available.
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47.
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Oxopyrido[2,3-d]pyrimidines as Covalent L858R/T790M Mutant Selective Epidermal Growth Factor Receptor (EGFR) Inhibitors. [electronic resource] by
- Wurz, Ryan P
- Pettus, Liping H
- Ashton, Kate
- Brown, James
- Chen, Jian Jeffrey
- Herberich, Brad
- Hong, Fang-Tsao
- Hu-Harrington, Essa
- Nguyen, Tom
- St Jean, David J
- Tadesse, Seifu
- Bauer, David
- Kubryk, Michele
- Zhan, Jinghui
- Cooke, Keegan
- Mitchell, Petia
- Andrews, Kristin L
- Hsieh, Faye
- Hickman, Dean
- Kalyanaraman, Nataraj
- Wu, Tian
- Reid, Darren L
- Lobenhofer, Edward K
- Andrews, Dina A
- Everds, Nancy
- Guzman, Roberto
- Parsons, Andrew T
- Hedley, Simon J
- Tedrow, Jason
- Thiel, Oliver R
- Potter, Matthew
- Radinsky, Robert
- Beltran, Pedro J
- Tasker, Andrew S
Producer: 20150923
In:
ACS medicinal chemistry letters vol. 6
Availability: No items available.
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48.
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Discovery and in vivo evaluation of (S)-N-(1-(7-fluoro-2-(pyridin-2-yl)quinolin-3-yl)ethyl)-9H-purin-6-amine (AMG319) and related PI3Kδ inhibitors for inflammation and autoimmune disease. [electronic resource] by
- Cushing, Timothy D
- Hao, Xiaolin
- Shin, Youngsook
- Andrews, Kristin
- Brown, Matthew
- Cardozo, Mario
- Chen, Yi
- Duquette, Jason
- Fisher, Ben
- Gonzalez-Lopez de Turiso, Felix
- He, Xiao
- Henne, Kirk R
- Hu, Yi-Ling
- Hungate, Randall
- Johnson, Michael G
- Kelly, Ron C
- Lucas, Brian
- McCarter, John D
- McGee, Lawrence R
- Medina, Julio C
- San Miguel, Tisha
- Mohn, Deanna
- Pattaropong, Vatee
- Pettus, Liping H
- Reichelt, Andreas
- Rzasa, Robert M
- Seganish, Jennifer
- Tasker, Andrew S
- Wahl, Robert C
- Wannberg, Sharon
- Whittington, Douglas A
- Whoriskey, John
- Yu, Gang
- Zalameda, Leeanne
- Zhang, Dawei
- Metz, Daniela P
Producer: 20150427
In:
Journal of medicinal chemistry vol. 58
Availability: No items available.
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49.
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Selective class I phosphoinositide 3-kinase inhibitors: optimization of a series of pyridyltriazines leading to the identification of a clinical candidate, AMG 511. [electronic resource] by
- Norman, Mark H
- Andrews, Kristin L
- Bo, Yunxin Y
- Booker, Shon K
- Caenepeel, Sean
- Cee, Victor J
- D'Angelo, Noel D
- Freeman, Daniel J
- Herberich, Bradley J
- Hong, Fang-Tsao
- Jackson, Claire L M
- Jiang, Jian
- Lanman, Brian A
- Liu, Longbin
- McCarter, John D
- Mullady, Erin L
- Nishimura, Nobuko
- Pettus, Liping H
- Reed, Anthony B
- Miguel, Tisha San
- Smith, Adrian L
- Stec, Markian M
- Tadesse, Seifu
- Tasker, Andrew
- Aidasani, Divesh
- Zhu, Xiaochun
- Subramanian, Raju
- Tamayo, Nuria A
- Wang, Ling
- Whittington, Douglas A
- Wu, Bin
- Wu, Tian
- Wurz, Ryan P
- Yang, Kevin
- Zalameda, Leeanne
- Zhang, Nancy
- Hughes, Paul E
Producer: 20121231
In:
Journal of medicinal chemistry vol. 55
Availability: No items available.
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