Results
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41.
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N-Acyl-N'-arylpiperazines as negative allosteric modulators of mGlu1: identification of VU0469650, a potent and selective tool compound with CNS exposure in rats. [electronic resource] by
- Lovell, Kimberly M
- Felts, Andrew S
- Rodriguez, Alice L
- Venable, Daryl F
- Cho, Hyekyung P
- Morrison, Ryan D
- Byers, Frank W
- Daniels, J Scott
- Niswender, Colleen M
- Conn, P Jeffrey
- Lindsley, Craig W
- Emmitte, Kyle A
Producer: 20140113
In:
Bioorganic & medicinal chemistry letters vol. 23
Availability: No items available.
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42.
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Novel M [electronic resource] by
- Poslusney, Michael S
- Salovich, James M
- Wood, Michael R
- Melancon, Bruce J
- Bollinger, Katrina A
- Luscombe, Vincent B
- Rodriguez, Alice L
- Engers, Darren W
- Bridges, Thomas M
- Niswender, Colleen M
- Conn, P Jeffrey
- Lindsley, Craig W
Producer: 20191209
In:
Bioorganic & medicinal chemistry letters vol. 29
Availability: No items available.
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43.
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Discovery and characterization of a novel series of N-phenylsulfonyl-1H-pyrrole picolinamides as positive allosteric modulators of the metabotropic glutamate receptor 4 (mGlu4). [electronic resource] by
- Gogliotti, Rocco D
- Blobaum, Anna L
- Morrison, Ryan M
- Daniels, J Scott
- Salovich, James M
- Cheung, Yiu-Yin
- Rodriguez, Alice L
- Loch, Matthew T
- Conn, P Jeffrey
- Lindsley, Craig W
- Niswender, Colleen M
- Hopkins, Corey R
Producer: 20170710
In:
Bioorganic & medicinal chemistry letters vol. 26
Availability: No items available.
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44.
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N-Alkylpyrido[1',2':1,5]pyrazolo-[4,3-d]pyrimidin-4-amines: A new series of negative allosteric modulators of mGlu1/5 with CNS exposure in rodents. [electronic resource] by
- Felts, Andrew S
- Rodriguez, Alice L
- Morrison, Ryan D
- Venable, Daryl F
- Blobaum, Anna L
- Byers, Frank W
- Daniels, J Scott
- Niswender, Colleen M
- Jones, Carrie K
- Conn, P Jeffrey
- Lindsley, Craig W
- Emmitte, Kyle A
Producer: 20161213
In:
Bioorganic & medicinal chemistry letters vol. 26
Availability: No items available.
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45.
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Substituted 1-Phenyl-3-(pyridin-2-yl)urea negative allosteric modulators of mGlu5: discovery of a new tool compound VU0463841 with activity in rat models of cocaine addiction. [electronic resource] by
- Amato, Russell J
- Felts, Andrew S
- Rodriguez, Alice L
- Venable, Daryl F
- Morrison, Ryan D
- Byers, Frank W
- Daniels, J Scott
- Niswender, Colleen M
- Conn, P Jeffrey
- Lindsley, Craig W
- Jones, Carrie K
- Emmitte, Kyle A
Producer: 20140401
In:
ACS chemical neuroscience vol. 4
Availability: No items available.
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46.
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Discovery and optimization of 3-(4-aryl/heteroarylsulfonyl)piperazin-1-yl)-6-(piperidin-1-yl)pyridazines as novel, CNS penetrant pan-muscarinic antagonists. [electronic resource] by
- Bender, Aaron M
- Weiner, Rebecca L
- Luscombe, Vincent B
- Ajmera, Sonia
- Cho, Hyekyung P
- Chang, Sichen
- Zhan, Xiaoyan
- Rodriguez, Alice L
- Niswender, Colleen M
- Engers, Darren W
- Bridges, Thomas M
- Conn, P Jeffrey
- Lindsley, Craig W
Producer: 20170818
In:
Bioorganic & medicinal chemistry letters vol. 27
Availability: No items available.
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47.
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Discovery of a novel 2,4-dimethylquinoline-6-carboxamide M [electronic resource] by
- Long, Madeline F
- Engers, Julie L
- Chang, Sichen
- Zhan, Xiaoyan
- Weiner, Rebecca L
- Luscombe, Vincent B
- Rodriguez, Alice L
- Cho, Hyekyung P
- Niswender, Colleen M
- Bridges, Thomas M
- Conn, P Jeffrey
- Engers, Darren W
- Lindsley, Craig W
Producer: 20171121
In:
Bioorganic & medicinal chemistry letters vol. 27
Availability: No items available.
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48.
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Discovery of a novel, CNS penetrant M [electronic resource] by
- Bewley, Blake R
- Spearing, Paul K
- Weiner, Rebecca L
- Luscombe, Vincent B
- Zhan, Xiaoyan
- Chang, Sichen
- Cho, Hyekyung P
- Rodriguez, Alice L
- Niswender, Colleen M
- Conn, P Jeffrey
- Bridges, Thomas M
- Engers, Darren W
- Lindsley, Craig W
Producer: 20170915
In:
Bioorganic & medicinal chemistry letters vol. 27
Availability: No items available.
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49.
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Discovery of a novel 2,3-dimethylimidazo[1,2-a]pyrazine-6-carboxamide M [electronic resource] by
- Temple, Kayla J
- Engers, Julie L
- Long, Madeline F
- Watson, Katherine J
- Chang, Sichen
- Luscombe, Vincent B
- Jenkins, Matthew T
- Rodriguez, Alice L
- Niswender, Colleen M
- Bridges, Thomas M
- Conn, P Jeffrey
- Engers, Darren W
- Lindsley, Craig W
Producer: 20210128
In:
Bioorganic & medicinal chemistry letters vol. 30
Availability: No items available.
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50.
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Chemical modulation of mutant mGlu1 receptors derived from deleterious GRM1 mutations found in schizophrenics. [electronic resource] by
- Cho, Hyekyung P
- Garcia-Barrantes, Pedro M
- Brogan, John T
- Hopkins, Corey R
- Niswender, Colleen M
- Rodriguez, Alice L
- Venable, Daryl F
- Morrison, Ryan D
- Bubser, Michael
- Daniels, J Scott
- Jones, Carrie K
- Conn, P Jeffrey
- Lindsley, Craig W
Producer: 20150714
In:
ACS chemical biology vol. 9
Availability: No items available.
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51.
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Discovery of an Orally Bioavailable and Central Nervous System (CNS) Penetrant mGlu [electronic resource] by
- Reed, Carson W
- Yohn, Samantha E
- Washecheck, Jordan P
- Roenfanz, Hanna F
- Quitalig, Marc C
- Luscombe, Vincent B
- Jenkins, Matthew T
- Rodriguez, Alice L
- Engers, Darren W
- Blobaum, Anna L
- Conn, P Jeffrey
- Niswender, Colleen M
- Lindsley, Craig W
Producer: 20200303
In:
Journal of medicinal chemistry vol. 62
Availability: No items available.
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52.
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Discovery of Novel Central Nervous System Penetrant Metabotropic Glutamate Receptor Subtype 2 (mGlu [electronic resource] by
- Childress, Elizabeth S
- Wieting, Joshua M
- Felts, Andrew S
- Breiner, Megan M
- Long, Madeline F
- Luscombe, Vincent B
- Rodriguez, Alice L
- Cho, Hyekyung P
- Blobaum, Anna L
- Niswender, Colleen M
- Emmitte, Kyle A
- Conn, P Jeffrey
- Lindsley, Craig W
Producer: 20191014
In:
Journal of medicinal chemistry vol. 62
Availability: No items available.
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53.
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Development and Antiparkinsonian Activity of VU0418506, a Selective Positive Allosteric Modulator of Metabotropic Glutamate Receptor 4 Homomers without Activity at mGlu2/4 Heteromers. [electronic resource] by
- Niswender, Colleen M
- Jones, Carrie K
- Lin, Xin
- Bubser, Michael
- Thompson Gray, Analisa
- Blobaum, Anna L
- Engers, Darren W
- Rodriguez, Alice L
- Loch, Matthew T
- Daniels, J Scott
- Lindsley, Craig W
- Hopkins, Corey R
- Javitch, Jonathan A
- Conn, P Jeffrey
Producer: 20171027
In:
ACS chemical neuroscience vol. 7
Availability: No items available.
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54.
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Investigating metabotropic glutamate receptor 5 allosteric modulator cooperativity, affinity, and agonism: enriching structure-function studies and structure-activity relationships. [electronic resource] by
- Gregory, Karen J
- Noetzel, Meredith J
- Rook, Jerri M
- Vinson, Paige N
- Stauffer, Shaun R
- Rodriguez, Alice L
- Emmitte, Kyle A
- Zhou, Ya
- Chun, Aspen C
- Felts, Andrew S
- Chauder, Brian A
- Lindsley, Craig W
- Niswender, Colleen M
- Conn, P Jeffrey
Producer: 20130212
In:
Molecular pharmacology vol. 82
Availability: No items available.
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55.
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Discovery of a novel 3,4-dimethylcinnoline carboxamide M [electronic resource] by
- Temple, Kayla J
- Engers, Julie L
- Long, Madeline F
- Gregro, Alison R
- Watson, Katherine J
- Chang, Sichen
- Jenkins, Matthew T
- Luscombe, Vincent B
- Rodriguez, Alice L
- Niswender, Colleen M
- Bridges, Thomas M
- Conn, P Jeffrey
- Engers, Darren W
- Lindsley, Craig W
Producer: 20200914
In:
Bioorganic & medicinal chemistry letters vol. 29
Availability: No items available.
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56.
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Discovery, Structure-Activity Relationship, and Biological Characterization of a Novel Series of 6-((1 H-Pyrazolo[4,3- b]pyridin-3-yl)amino)-benzo[ d]isothiazole-3-carboxamides as Positive Allosteric Modulators of the Metabotropic Glutamate Receptor 4 (mGlu [electronic resource] by
- Bollinger, Sean R
- Engers, Darren W
- Panarese, Joseph D
- West, Mary
- Engers, Julie L
- Loch, Matthew T
- Rodriguez, Alice L
- Blobaum, Anna L
- Jones, Carrie K
- Thompson Gray, Analisa
- Conn, P Jeffrey
- Lindsley, Craig W
- Niswender, Colleen M
- Hopkins, Corey R
Producer: 20191014
In:
Journal of medicinal chemistry vol. 62
Availability: No items available.
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57.
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Design and Synthesis of mGlu [electronic resource] by
- Bollinger, Katrina A
- Felts, Andrew S
- Brassard, Christopher J
- Engers, Julie L
- Rodriguez, Alice L
- Weiner, Rebecca L
- Cho, Hyekyung P
- Chang, Sichen
- Bubser, Michael
- Jones, Carrie K
- Blobaum, Anna L
- Niswender, Colleen M
- Conn, P Jeffrey
- Emmitte, Kyle A
- Lindsley, Craig W
Publication details: ACS medicinal chemistry letters Sep 2017
In:
ACS medicinal chemistry letters vol. 8
Availability: No items available.
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58.
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Discovery of VU0431316: a negative allosteric modulator of mGlu5 with activity in a mouse model of anxiety. [electronic resource] by
- Bates, Brittney S
- Rodriguez, Alice L
- Felts, Andrew S
- Morrison, Ryan D
- Venable, Daryl F
- Blobaum, Anna L
- Byers, Frank W
- Lawson, Kera P
- Daniels, J Scott
- Niswender, Colleen M
- Jones, Carrie K
- Conn, P Jeffrey
- Lindsley, Craig W
- Emmitte, Kyle A
Producer: 20150305
In:
Bioorganic & medicinal chemistry letters vol. 24
Availability: No items available.
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59.
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Discovery of imidazo[1,2-a]-, [1,2,4]triazolo[4,3-a]-, and [1,2,4]triazolo[1,5-a]pyridine-8-carboxamide negative allosteric modulators of metabotropic glutamate receptor subtype 5. [electronic resource] by
- Felts, Andrew S
- Rodriguez, Alice L
- Morrison, Ryan D
- Bollinger, Katrina A
- Venable, Daryl F
- Blobaum, Anna L
- Byers, Frank W
- Thompson Gray, Analisa
- Daniels, J Scott
- Niswender, Colleen M
- Jones, Carrie K
- Conn, P Jeffrey
- Lindsley, Craig W
- Emmitte, Kyle A
Producer: 20171206
In:
Bioorganic & medicinal chemistry letters vol. 27
Availability: No items available.
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60.
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Discovery of VU0409106: A negative allosteric modulator of mGlu5 with activity in a mouse model of anxiety. [electronic resource] by
- Felts, Andrew S
- Rodriguez, Alice L
- Morrison, Ryan D
- Venable, Daryl F
- Manka, Jason T
- Bates, Brittney S
- Blobaum, Anna L
- Byers, Frank W
- Daniels, J Scott
- Niswender, Colleen M
- Jones, Carrie K
- Conn, P Jeffrey
- Lindsley, Craig W
- Emmitte, Kyle A
Producer: 20140430
In:
Bioorganic & medicinal chemistry letters vol. 23
Availability: No items available.
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