Results
|
41.
|
Design and synthesis of benzofuranic derivatives as new ligands at the melatonin-binding site MT3. [electronic resource] by
- Ettaoussi, Mohamed
- Péres, Basile
- Klupsch, Fréderique
- Delagrange, Philippe
- Boutin, Jean-A
- Renard, Pierre
- Caignard, Daniel-H
- Chavatte, Philippe
- Berthelot, Pascal
- Lesieur, Daniel
- Yous, Saïd
Producer: 20080826
In:
Bioorganic & medicinal chemistry vol. 16
Availability: No items available.
|
|
42.
|
Novel 4-oxo-1,4-dihydroquinoline-3-carboxamide derivatives as new CB2 cannabinoid receptors agonists: synthesis, pharmacological properties and molecular modeling. [electronic resource] by
- Stern, Eric
- Muccioli, Giulio G
- Millet, Régis
- Goossens, Jean-François
- Farce, Amaury
- Chavatte, Philippe
- Poupaert, Jacques H
- Lambert, Didier M
- Depreux, Patrick
- Hénichart, Jean-Pierre
Producer: 20060216
In:
Journal of medicinal chemistry vol. 49
Availability: No items available.
|
|
43.
|
Potent farnesyltransferase inhibitors with 1,4-diazepane scaffolds as novel destabilizing microtubule agents in hormone-resistant prostate cancer. [electronic resource] by
- Wlodarczyk, Nicolas
- Le Broc-Ryckewaert, Delphine
- Gilleron, Pauline
- Lemoine, Amélie
- Farce, Amaury
- Chavatte, Philippe
- Dubois, Joëlle
- Pommery, Nicole
- Hénichart, Jean-Pierre
- Furman, Christophe
- Millet, Régis
Producer: 20110606
In:
Journal of medicinal chemistry vol. 54
Availability: No items available.
|
|
44.
|
Enantioseparation of pyroglutamide derivatives on polysaccharide based chiral stationary phases by high-performance liquid chromatography and supercritical fluid chromatography: a comparative study. [electronic resource] by
- Baudelet, Davy
- Schifano-Faux, Nadège
- Ghinet, Alina
- Dezitter, Xavier
- Barbotin, Florent
- Gautret, Philippe
- Rigo, Benoit
- Chavatte, Philippe
- Millet, Régis
- Furman, Christophe
- Vaccher, Claude
- Lipka, Emmanuelle
Producer: 20141201
In:
Journal of chromatography. A vol. 1363
Availability: No items available.
|
|
45.
|
Importance of the second extracellular loop for melatonin MT [electronic resource] by
- Clement, Nathalie
- Renault, Nicolas
- Guillaume, Jean-Luc
- Cecon, Erika
- Journé, Anne-Sophie
- Laurent, Xavier
- Tadagaki, Kenjiro
- Cogé, Francis
- Gohier, Arnaud
- Delagrange, Philippe
- Chavatte, Philippe
- Jockers, Ralf
Producer: 20191002
In:
British journal of pharmacology vol. 175
Availability: No items available.
|
|
46.
|
Design and synthesis of fused tetrahydroisoquinoline-iminoimidazolines. [electronic resource] by
- Moas-Héloire, Valeria
- Renault, Nicolas
- Batalha, Vania
- Arias, Angela Rincon
- Marchivie, Mathieu
- Yous, Said
- Deguine, Noémie
- Buée, Luc
- Chavatte, Philippe
- Blum, David
- Lopes, Luisa
- Melnyk, Patricia
- Agouridas, Laurence
Producer: 20160920
In:
European journal of medicinal chemistry vol. 106
Availability: No items available.
|
|
47.
|
Conformational Restriction Leading to a Selective CB2 Cannabinoid Receptor Agonist Orally Active Against Colitis. [electronic resource] by
- El Bakali, Jamal
- Muccioli, Giulio G
- Body-Malapel, Mathilde
- Djouina, Madjid
- Klupsch, Frédérique
- Ghinet, Alina
- Barczyk, Amélie
- Renault, Nicolas
- Chavatte, Philippe
- Desreumaux, Pierre
- Lambert, Didier M
- Millet, Régis
Producer: 20150220
In:
ACS medicinal chemistry letters vol. 6
Availability: No items available.
|
|
48.
|
4-Oxo-1,4-dihydropyridines as selective CB2 cannabinoid receptor ligands: structural insights into the design of a novel inverse agonist series. [electronic resource] by
- El Bakali, Jamal
- Muccioli, Giulio G
- Renault, Nicolas
- Pradal, Delphine
- Body-Malapel, Mathilde
- Djouina, Madjid
- Hamtiaux, Laurie
- Andrzejak, Virginie
- Desreumaux, Pierre
- Chavatte, Philippe
- Lambert, Didier M
- Millet, Régis
Producer: 20101230
In:
Journal of medicinal chemistry vol. 53
Availability: No items available.
|
|
49.
|
Design, synthesis and pharmacological evaluation of novel naphthalenic derivatives as selective MT(1) melatoninergic ligands. [electronic resource] by
- Mésangeau, Christophe
- Pérès, Basile
- Descamps-François, Carole
- Chavatte, Philippe
- Audinot, Valérie
- Coumailleau, Sophie
- Boutin, Jean A
- Delagrange, Philippe
- Bennejean, Caroline
- Renard, Pierre
- Caignard, Daniel H
- Berthelot, Pascal
- Yous, Saïd
Producer: 20100827
In:
Bioorganic & medicinal chemistry vol. 18
Availability: No items available.
|
|
50.
|
2,6-Diphenylthiazolo[3,2-b][1,2,4]triazoles as telomeric G-quadruplex stabilizers. [electronic resource] by
- El Bakali, Jamal
- Klupsch, Frédérique
- Guédin, Aurore
- Brassart, Bertrand
- Fontaine, Gaëlle
- Farce, Amaury
- Roussel, Pascal
- Houssin, Raymond
- Bernier, Jean-Luc
- Chavatte, Philippe
- Mergny, Jean-Louis
- Riou, Jean-François
- Hénichart, Jean-Pierre
Producer: 20090901
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
|
|
51.
|
Intestinal antiinflammatory effect of 5-aminosalicylic acid is dependent on peroxisome proliferator-activated receptor-gamma. [electronic resource] by
- Rousseaux, Christel
- Lefebvre, Bruno
- Dubuquoy, Laurent
- Lefebvre, Philippe
- Romano, Olivier
- Auwerx, Johan
- Metzger, Daniel
- Wahli, Walter
- Desvergne, Béatrice
- Naccari, Gian Carlo
- Chavatte, Philippe
- Farce, Amaury
- Bulois, Philippe
- Cortot, Antoine
- Colombel, Jean Frédéric
- Desreumaux, Pierre
Producer: 20050617
In:
The Journal of experimental medicine vol. 201
Availability: No items available.
|
|
52.
|
4-Oxo-1,4-dihydropyridines as selective CB₂ cannabinoid receptor ligands. Part 2: discovery of new agonists endowed with protective effect against experimental colitis. [electronic resource] by
- El Bakali, Jamal
- Gilleron, Pauline
- Body-Malapel, Mathilde
- Mansouri, Roxane
- Muccioli, Giulio G
- Djouina, Madjid
- Barczyk, Amélie
- Klupsch, Frédérique
- Andrzejak, Virginie
- Lipka, Emmanuelle
- Furman, Christophe
- Lambert, Didier M
- Chavatte, Philippe
- Desreumaux, Pierre
- Millet, Régis
Producer: 20130205
In:
Journal of medicinal chemistry vol. 55
Availability: No items available.
|
|
53.
|
Toward the Discovery of a Novel Class of YAP⁻TEAD Interaction Inhibitors by Virtual Screening Approach Targeting YAP⁻TEAD Protein⁻Protein Interface. [electronic resource] by
- Gibault, Floriane
- Coevoet, Mathilde
- Sturbaut, Manon
- Farce, Amaury
- Renault, Nicolas
- Allemand, Frédéric
- Guichou, Jean-François
- Drucbert, Anne-Sophie
- Foulon, Catherine
- Magnez, Romain
- Thuru, Xavier
- Corvaisier, Matthieu
- Huet, Guillemette
- Chavatte, Philippe
- Melnyk, Patricia
- Bailly, Fabrice
- Cotelle, Philippe
Publication details: Cancers May 2018
In:
Cancers vol. 10
Availability: No items available.
|
|
54.
|
3-Carboxamido-5-aryl-isoxazoles as new CB2 agonists for the treatment of colitis. [electronic resource] by
- Tourteau, Aurélien
- Andrzejak, Virginie
- Body-Malapel, Mathilde
- Lemaire, Lucas
- Lemoine, Amélie
- Mansouri, Roxane
- Djouina, Madjid
- Renault, Nicolas
- El Bakali, Jamal
- Desreumaux, Pierre
- Muccioli, Giulio G
- Lambert, Didier M
- Chavatte, Philippe
- Rigo, Benoît
- Leleu-Chavain, Natascha
- Millet, Régis
Producer: 20140318
In:
Bioorganic & medicinal chemistry vol. 21
Availability: No items available.
|
|
55.
|
Novel 1,3-dicarbonyl compounds having 2(3H)-benzazolonic heterocycles as PPARgamma agonists. [electronic resource] by
- Blanc-Delmas, Elodie
- Lebegue, Nicolas
- Wallez, Valérie
- Leclerc, Véronique
- Yous, Saïd
- Carato, Pascal
- Farce, Amaury
- Bennejean, Caroline
- Renard, Pierre
- Caignard, Daniel-Henri
- Audinot-Bouchez, Valérie
- Chomarat, Pascale
- Boutin, Jean
- Hennuyer, Nathalie
- Louche, Katie
- Carmona, Maria Carmen
- Staels, Bart
- Pénicaud, Luc
- Casteilla, Louis
- Lonchampt, Michel
- Dacquet, Catherine
- Chavatte, Philippe
- Berthelot, Pascal
- Lesieur, Daniel
Producer: 20061222
In:
Bioorganic & medicinal chemistry vol. 14
Availability: No items available.
|