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Identification of RC-33 as a potent and selective σ1 receptor agonist potentiating NGF-induced neurite outgrowth in PC12 cells. Part 2: g-scale synthesis, physicochemical characterization and in vitro metabolic stability. [electronic resource] by
- Rossi, Daniela
- Marra, Annamaria
- Picconi, Pietro
- Serra, Massimo
- Catenacci, Laura
- Sorrenti, Milena
- Laurini, Erik
- Fermeglia, Maurizio
- Pricl, Sabrina
- Brambilla, Stefania
- Almirante, Nicoletta
- Peviani, Marco
- Curti, Daniela
- Collina, Simona
Producer: 20131112
In:
Bioorganic & medicinal chemistry vol. 21
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Toward the identification of neuroprotective agents: g-scale synthesis, pharmacokinetic evaluation and CNS distribution of (R)-RC-33, a promising SIGMA1 receptor agonist. [electronic resource] by
- Marra, Annamaria
- Rossi, Daniela
- Pignataro, Luca
- Bigogno, Chiara
- Canta, Annalisa
- Oggioni, Norberto
- Malacrida, Alessio
- Corbo, Massimo
- Cavaletti, Guido
- Peviani, Marco
- Curti, Daniela
- Dondio, Giulio
- Collina, Simona
Producer: 20161031
In:
Future medicinal chemistry vol. 8
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312.
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Glutathione peroxidase-1 gene rescues cocaine-induced conditioned place preference in mice by inhibiting σ-1 receptor expression. [electronic resource] by
- Pham, Duc Toan
- Chung, Yoon Hee
- Mai, Huynh Nhu
- Sharma, Naveen
- Yun, Jaesuk
- Kim, Hee Jin
- Cheong, Jae Hoon
- Jeong, Ji Hoon
- Kim, Dae-Joong
- Shin, Eun-Joo
- Kim, Hyoung-Chun
Producer: 20200825
In:
Clinical and experimental pharmacology & physiology vol. 46
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Novel Potent N-Methyl-d-aspartate (NMDA) Receptor Antagonists or σ1 Receptor Ligands Based on Properly Substituted 1,4-Dioxane Ring. [electronic resource] by
- Bonifazi, Alessandro
- Del Bello, Fabio
- Mammoli, Valerio
- Piergentili, Alessandro
- Petrelli, Riccardo
- Cimarelli, Cristina
- Pellei, Maura
- Schepmann, Dirk
- Wünsch, Bernhard
- Barocelli, Elisabetta
- Bertoni, Simona
- Flammini, Lisa
- Amantini, Consuelo
- Nabissi, Massimo
- Santoni, Giorgio
- Vistoli, Giulio
- Quaglia, Wilma
Producer: 20160225
In:
Journal of medicinal chemistry vol. 58
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Pharmacological properties of S1RA, a new sigma-1 receptor antagonist that inhibits neuropathic pain and activity-induced spinal sensitization. [electronic resource] by
- Romero, L
- Zamanillo, D
- Nadal, X
- Sánchez-Arroyos, R
- Rivera-Arconada, I
- Dordal, A
- Montero, A
- Muro, A
- Bura, A
- Segalés, C
- Laloya, M
- Hernández, E
- Portillo-Salido, E
- Escriche, M
- Codony, X
- Encina, G
- Burgueño, J
- Merlos, M
- Baeyens, J M
- Giraldo, J
- López-García, J A
- Maldonado, R
- Plata-Salamán, C R
- Vela, J M
Producer: 20121210
In:
British journal of pharmacology vol. 166
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