Results
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2201.
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Discovery of AM-7209, a potent and selective 4-amidobenzoic acid inhibitor of the MDM2-p53 interaction. [electronic resource] by
- Rew, Yosup
- Sun, Daqing
- Yan, Xuelei
- Beck, Hilary P
- Canon, Jude
- Chen, Ada
- Duquette, Jason
- Eksterowicz, John
- Fox, Brian M
- Fu, Jiasheng
- Gonzalez, Ana Z
- Houze, Jonathan
- Huang, Xin
- Jiang, Min
- Jin, Lixia
- Li, Yihong
- Li, Zhihong
- Ling, Yun
- Lo, Mei-Chu
- Long, Alexander M
- McGee, Lawrence R
- McIntosh, Joel
- Oliner, Jonathan D
- Osgood, Tao
- Saiki, Anne Y
- Shaffer, Paul
- Wang, Yu Chung
- Wortman, Sarah
- Yakowec, Peter
- Ye, Qiuping
- Yu, Dongyin
- Zhao, Xiaoning
- Zhou, Jing
- Medina, Julio C
- Olson, Steven H
Producer: 20150310
In:
Journal of medicinal chemistry vol. 57
Availability: No items available.
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2202.
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Discovery of a potent, selective, and orally bioavailable pyridinyl-pyrimidine phthalazine aurora kinase inhibitor. [electronic resource] by
- Cee, Victor J
- Schenkel, Laurie B
- Hodous, Brian L
- Deak, Holly L
- Nguyen, Hanh N
- Olivieri, Philip R
- Romero, Karina
- Bak, Annette
- Be, Xuhai
- Bellon, Steve
- Bush, Tammy L
- Cheng, Alan C
- Chung, Grace
- Coats, Steve
- Eden, Patrick M
- Hanestad, Kelly
- Gallant, Paul L
- Gu, Yan
- Huang, Xin
- Kendall, Richard L
- Lin, Min-Hwa Jasmine
- Morrison, Michael J
- Patel, Vinod F
- Radinsky, Robert
- Rose, Paul E
- Ross, Sandra
- Sun, Ji-Rong
- Tang, Jin
- Zhao, Huilin
- Payton, Marc
- Geuns-Meyer, Stephanie D
Producer: 20100930
In:
Journal of medicinal chemistry vol. 53
Availability: No items available.
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2203.
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Discovery of 2,4-bis-arylamino-1,3-pyrimidines as insulin-like growth factor-1 receptor (IGF-1R) inhibitors. [electronic resource] by
- Buchanan, John L
- Newcomb, John R
- Carney, David P
- Chaffee, Stuart C
- Chai, Lilly
- Cupples, Rod
- Epstein, Linda F
- Gallant, Paul
- Gu, Yan
- Harmange, Jean-Christophe
- Hodge, Kathy
- Houk, Brett E
- Huang, Xin
- Jona, Janan
- Joseph, Smriti
- Jun, H Toni
- Kumar, Rakesh
- Li, Chun
- Lu, John
- Menges, Tom
- Morrison, Michael J
- Novak, Perry M
- van der Plas, Simon
- Radinsky, Robert
- Rose, Paul E
- Sawant, Satin
- Sun, Ji-Rong
- Surapaneni, Sekhar
- Turci, Susan M
- Xu, Keyang
- Yanez, Evelyn
- Zhao, Huilin
- Zhu, Xiaotian
Producer: 20110719
In:
Bioorganic & medicinal chemistry letters vol. 21
Availability: No items available.
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2204.
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Structure-based design of novel inhibitors of the MDM2-p53 interaction. [electronic resource] by
- Rew, Yosup
- Sun, Daqing
- Gonzalez-Lopez De Turiso, Felix
- Bartberger, Michael D
- Beck, Hilary P
- Canon, Jude
- Chen, Ada
- Chow, David
- Deignan, Jeffrey
- Fox, Brian M
- Gustin, Darin
- Huang, Xin
- Jiang, Min
- Jiao, Xianyun
- Jin, Lixia
- Kayser, Frank
- Kopecky, David J
- Li, Yihong
- Lo, Mei-Chu
- Long, Alexander M
- Michelsen, Klaus
- Oliner, Jonathan D
- Osgood, Tao
- Ragains, Mark
- Saiki, Anne Y
- Schneider, Steve
- Toteva, Maria
- Yakowec, Peter
- Yan, Xuelei
- Ye, Qiuping
- Yu, Dongyin
- Zhao, Xiaoning
- Zhou, Jing
- Medina, Julio C
- Olson, Steven H
Producer: 20121001
In:
Journal of medicinal chemistry vol. 55
Availability: No items available.
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2205.
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Selective and potent morpholinone inhibitors of the MDM2-p53 protein-protein interaction. [electronic resource] by
- Gonzalez, Ana Z
- Eksterowicz, John
- Bartberger, Michael D
- Beck, Hilary P
- Canon, Jude
- Chen, Ada
- Chow, David
- Duquette, Jason
- Fox, Brian M
- Fu, Jiasheng
- Huang, Xin
- Houze, Jonathan B
- Jin, Lixia
- Li, Yihong
- Li, Zhihong
- Ling, Yun
- Lo, Mei-Chu
- Long, Alexander M
- McGee, Lawrence R
- McIntosh, Joel
- McMinn, Dustin L
- Oliner, Jonathan D
- Osgood, Tao
- Rew, Yosup
- Saiki, Anne Y
- Shaffer, Paul
- Wortman, Sarah
- Yakowec, Peter
- Yan, Xuelei
- Ye, Qiuping
- Yu, Dongyin
- Zhao, Xiaoning
- Zhou, Jing
- Olson, Steven H
- Medina, Julio C
- Sun, Daqing
Producer: 20140527
In:
Journal of medicinal chemistry vol. 57
Availability: No items available.
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2206.
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Structure-guided design of aminopyrimidine amides as potent, selective inhibitors of lymphocyte specific kinase: synthesis, structure-activity relationships, and inhibition of in vivo T cell activation. [electronic resource] by
- DiMauro, Erin F
- Newcomb, John
- Nunes, Joseph J
- Bemis, Jean E
- Boucher, Christina
- Chai, Lilly
- Chaffee, Stuart C
- Deak, Holly L
- Epstein, Linda F
- Faust, Ted
- Gallant, Paul
- Gore, Anu
- Gu, Yan
- Henkle, Brad
- Hsieh, Faye
- Huang, Xin
- Kim, Joseph L
- Lee, Josie H
- Martin, Matthew W
- McGowan, David C
- Metz, Daniela
- Mohn, Deanna
- Morgenstern, Kurt A
- Oliveira-dos-Santos, Antonio
- Patel, Vinod F
- Powers, David
- Rose, Paul E
- Schneider, Stephen
- Tomlinson, Susan A
- Tudor, Yan-Yan
- Turci, Susan M
- Welcher, Andrew A
- Zhao, Huilin
- Zhu, Li
- Zhu, Xiaotian
Producer: 20080611
In:
Journal of medicinal chemistry vol. 51
Availability: No items available.
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2207.
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AMG 176, a Selective MCL1 Inhibitor, Is Effective in Hematologic Cancer Models Alone and in Combination with Established Therapies. [electronic resource] by
- Caenepeel, Sean
- Brown, Sean P
- Belmontes, Brian
- Moody, Gordon
- Keegan, Kathleen S
- Chui, Danny
- Whittington, Douglas A
- Huang, Xin
- Poppe, Leszek
- Cheng, Alan C
- Cardozo, Mario
- Houze, Jonathan
- Li, Yunxiao
- Lucas, Brian
- Paras, Nick A
- Wang, Xianghong
- Taygerly, Joshua P
- Vimolratana, Marc
- Zancanella, Manuel
- Zhu, Liusheng
- Cajulis, Elaina
- Osgood, Tao
- Sun, Jan
- Damon, Leah
- Egan, Regina K
- Greninger, Patricia
- McClanaghan, Joseph D
- Gong, Jianan
- Moujalled, Donia
- Pomilio, Giovanna
- Beltran, Pedro
- Benes, Cyril H
- Roberts, Andrew W
- Huang, David C
- Wei, Andrew
- Canon, Jude
- Coxon, Angela
- Hughes, Paul E
Producer: 20191223
In:
Cancer discovery vol. 8
Availability: No items available.
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2208.
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Discovery of aminoquinazolines as potent, orally bioavailable inhibitors of Lck: synthesis, SAR, and in vivo anti-inflammatory activity. [electronic resource] by
- DiMauro, Erin F
- Newcomb, John
- Nunes, Joseph J
- Bemis, Jean E
- Boucher, Christina
- Buchanan, John L
- Buckner, William H
- Cee, Victor J
- Chai, Lilly
- Deak, Holly L
- Epstein, Linda F
- Faust, Ted
- Gallant, Paul
- Geuns-Meyer, Stephanie D
- Gore, Anu
- Gu, Yan
- Henkle, Brad
- Hodous, Brian L
- Hsieh, Faye
- Huang, Xin
- Kim, Joseph L
- Lee, Josie H
- Martin, Matthew W
- Masse, Craig E
- McGowan, David C
- Metz, Daniela
- Mohn, Deanna
- Morgenstern, Kurt A
- Oliveira-dos-Santos, Antonio
- Patel, Vinod F
- Powers, David
- Rose, Paul E
- Schneider, Stephen
- Tomlinson, Susan A
- Tudor, Yan-Yan
- Turci, Susan M
- Welcher, Andrew A
- White, Ryan D
- Zhao, Huilin
- Zhu, Li
- Zhu, Xiaotian
Producer: 20061024
In:
Journal of medicinal chemistry vol. 49
Availability: No items available.
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2209.
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Novel 2-aminopyrimidine carbamates as potent and orally active inhibitors of Lck: synthesis, SAR, and in vivo antiinflammatory activity. [electronic resource] by
- Martin, Matthew W
- Newcomb, John
- Nunes, Joseph J
- McGowan, David C
- Armistead, David M
- Boucher, Christina
- Buchanan, John L
- Buckner, William
- Chai, Lilly
- Elbaum, Daniel
- Epstein, Linda F
- Faust, Theodore
- Flynn, Shaun
- Gallant, Paul
- Gore, Anu
- Gu, Yan
- Hsieh, Faye
- Huang, Xin
- Lee, Josie H
- Metz, Daniela
- Middleton, Scot
- Mohn, Deanna
- Morgenstern, Kurt
- Morrison, Michael J
- Novak, Perry M
- Oliveira-dos-Santos, Antonio
- Powers, David
- Rose, Paul
- Schneider, Stephen
- Sell, Stephanie
- Tudor, Yanyan
- Turci, Susan M
- Welcher, Andrew A
- White, Ryan D
- Zack, Debra
- Zhao, Huilin
- Zhu, Li
- Zhu, Xiaotian
- Ghiron, Chiara
- Amouzegh, Patricia
- Ermann, Monika
- Jenkins, James
- Johnston, David
- Napier, Spencer
- Power, Eoin
Producer: 20060913
In:
Journal of medicinal chemistry vol. 49
Availability: No items available.
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2210.
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miRTarBase update 2018: a resource for experimentally validated microRNA-target interactions. [electronic resource] by
- Chou, Chih-Hung
- Shrestha, Sirjana
- Yang, Chi-Dung
- Chang, Nai-Wen
- Lin, Yu-Ling
- Liao, Kuang-Wen
- Huang, Wei-Chi
- Sun, Ting-Hsuan
- Tu, Siang-Jyun
- Lee, Wei-Hsiang
- Chiew, Men-Yee
- Tai, Chun-San
- Wei, Ting-Yen
- Tsai, Tzi-Ren
- Huang, Hsin-Tzu
- Wang, Chung-Yu
- Wu, Hsin-Yi
- Ho, Shu-Yi
- Chen, Pin-Rong
- Chuang, Cheng-Hsun
- Hsieh, Pei-Jung
- Wu, Yi-Shin
- Chen, Wen-Liang
- Li, Meng-Ju
- Wu, Yu-Chun
- Huang, Xin-Yi
- Ng, Fung Ling
- Buddhakosai, Waradee
- Huang, Pei-Chun
- Lan, Kuan-Chun
- Huang, Chia-Yen
- Weng, Shun-Long
- Cheng, Yeong-Nan
- Liang, Chao
- Hsu, Wen-Lian
- Huang, Hsien-Da
Producer: 20190801
In:
Nucleic acids research vol. 46
Availability: No items available.
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2211.
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Discovery of AMG 232, a potent, selective, and orally bioavailable MDM2-p53 inhibitor in clinical development. [electronic resource] by
- Sun, Daqing
- Li, Zhihong
- Rew, Yosup
- Gribble, Michael
- Bartberger, Michael D
- Beck, Hilary P
- Canon, Jude
- Chen, Ada
- Chen, Xiaoqi
- Chow, David
- Deignan, Jeffrey
- Duquette, Jason
- Eksterowicz, John
- Fisher, Benjamin
- Fox, Brian M
- Fu, Jiasheng
- Gonzalez, Ana Z
- Gonzalez-Lopez De Turiso, Felix
- Houze, Jonathan B
- Huang, Xin
- Jiang, Min
- Jin, Lixia
- Kayser, Frank
- Liu, Jiwen Jim
- Lo, Mei-Chu
- Long, Alexander M
- Lucas, Brian
- McGee, Lawrence R
- McIntosh, Joel
- Mihalic, Jeff
- Oliner, Jonathan D
- Osgood, Tao
- Peterson, Matthew L
- Roveto, Philip
- Saiki, Anne Y
- Shaffer, Paul
- Toteva, Maria
- Wang, Yingcai
- Wang, Yu Chung
- Wortman, Sarah
- Yakowec, Peter
- Yan, Xuelei
- Ye, Qiuping
- Yu, Dongyin
- Yu, Ming
- Zhao, Xiaoning
- Zhou, Jing
- Zhu, Jiang
- Olson, Steven H
- Medina, Julio C
Producer: 20140429
In:
Journal of medicinal chemistry vol. 57
Availability: No items available.
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