Results
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221.
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Discovery of (2S)-N-[(1R)-2-[4-cyclohexyl-4-[[(1,1-dimethylethyl)amino]carbonyl]-1-piperidinyl]-1-[(4-fluorophenyl)methyl]-2-oxoethyl]-4-methyl-2-piperazinecarboxamide (MB243), a potent and selective melanocortin subtype-4 receptor agonist. [electronic resource] by
- Palucki, Brenda L
- Park, Min K
- Nargund, Ravi P
- Ye, Zhixiong
- Sebhat, Iyassu K
- Pollard, Patrick G
- Kalyani, Rubana N
- Tang, Rui
- Macneil, Tanya
- Weinberg, David H
- Vongs, Aurawan
- Rosenblum, Charles I
- Doss, George A
- Miller, Randall R
- Stearns, Ralph A
- Peng, Qianping
- Tamvakopoulos, Constantin
- McGowan, Erin
- Martin, William J
- Metzger, Joseph M
- Shepherd, Cherrie A
- Strack, Alison M
- Macintyre, D Euan
- Van der Ploeg, Lex H T
- Patchett, Arthur A
Producer: 20050502
In:
Bioorganic & medicinal chemistry letters vol. 15
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222.
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A selective human beta3 adrenergic receptor agonist increases metabolic rate in rhesus monkeys. [electronic resource] by
- Fisher, M H
- Amend, A M
- Bach, T J
- Barker, J M
- Brady, E J
- Candelore, M R
- Carroll, D
- Cascieri, M A
- Chiu, S H
- Deng, L
- Forrest, M J
- Hegarty-Friscino, B
- Guan, X M
- Hom, G J
- Hutchins, J E
- Kelly, L J
- Mathvink, R J
- Metzger, J M
- Miller, R R
- Ok, H O
- Parmee, E R
- Saperstein, R
- Strader, C D
- Stearns, R A
- MacIntyre, D E
Producer: 19980626
In:
The Journal of clinical investigation vol. 101
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223.
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A potent, nonpeptidyl 1H-quinolone antagonist for the gonadotropin-releasing hormone receptor. [electronic resource] by
- DeVita, R J
- Walsh, T F
- Young, J R
- Jiang, J
- Ujjainwalla, F
- Toupence, R B
- Parikh, M
- Huang, S X
- Fair, J A
- Goulet, M T
- Wyvratt, M J
- Lo, J L
- Ren, N
- Yudkovitz, J B
- Yang, Y T
- Cheng, K
- Cui, J
- Mount, G
- Rohrer, S P
- Schaeffer, J M
- Rhodes, L
- Drisko, J E
- McGowan, E
- MacIntyre, D E
- Vincent, S
- Carlin, J R
- Cameron, J
- Smith, R G
Producer: 20010503
In:
Journal of medicinal chemistry vol. 44
Availability: No items available.
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224.
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Analgesic effects of a substituted N-triazole oxindole (TROX-1), a state-dependent, voltage-gated calcium channel 2 blocker. [electronic resource] by
- Abbadie, Catherine
- McManus, Owen B
- Sun, Shu-Yu
- Bugianesi, Randal M
- Dai, Ge
- Haedo, Rodolfo J
- Herrington, James B
- Kaczorowski, Gregory J
- Smith, McHardy M
- Swensen, Andrew M
- Warren, Vivien A
- Williams, Brande
- Arneric, Stephen P
- Eduljee, Cyrus
- Snutch, Terrance P
- Tringham, Elizabeth W
- Jochnowitz, Nina
- Liang, Annie
- Euan MacIntyre, D
- McGowan, Erin
- Mistry, Shruti
- White, Valerie V
- Hoyt, Scott B
- London, Clare
- Lyons, Kathryn A
- Bunting, Patricia B
- Volksdorf, Sylvia
- Duffy, Joseph L
Producer: 20100817
In:
The Journal of pharmacology and experimental therapeutics vol. 334
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225.
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Antiobesity efficacy of a novel cannabinoid-1 receptor inverse agonist, N-[(1S,2S)-3-(4-chlorophenyl)-2-(3-cyanophenyl)-1-methylpropyl]-2-methyl-2-[[5-(trifluoromethyl)pyridin-2-yl]oxy]propanamide (MK-0364), in rodents. [electronic resource] by
- Fong, Tung M
- Guan, Xiao-Ming
- Marsh, Donald J
- Shen, Chun-Pyn
- Stribling, D Sloan
- Rosko, Kim M
- Lao, Julie
- Yu, Hong
- Feng, Yue
- Xiao, Jing C
- Van der Ploeg, Lex H T
- Goulet, Mark T
- Hagmann, Williams K
- Lin, Linus S
- Lanza, Thomas J
- Jewell, James P
- Liu, Ping
- Shah, Shrenik K
- Qi, Hongbo
- Tong, Xinchun
- Wang, Junying
- Xu, Suoyu S
- Francis, Barbara
- Strack, Alison M
- MacIntyre, D Euan
- Shearman, Lauren P
Producer: 20070730
In:
The Journal of pharmacology and experimental therapeutics vol. 321
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226.
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Discovery of a spiroindane based compound as a potent, selective, orally bioavailable melanocortin subtype-4 receptor agonist. [electronic resource] by
- He, Shuwen
- Ye, Zhixiong
- Dobbelaar, Peter H
- Sebhat, Iyassu K
- Guo, Liangqin
- Liu, Jian
- Jian, Tianying
- Lai, Yingjie
- Franklin, Christopher L
- Bakshi, Raman K
- Dellureficio, James P
- Hong, Qingmei
- Tsou, Nancy N
- Ball, Richard G
- Cashen, Doreen E
- Martin, William J
- Weinberg, David H
- Macneil, Tanya
- Tang, Rui
- Tamvakopoulos, Constantin
- Peng, Qianping
- Miller, Randy R
- Stearns, Ralph A
- Chen, Howard Y
- Chen, Airu S
- Strack, Alison M
- Fong, Tung M
- Macintyre, D Euan
- Wyvratt, Matthew J
- Nargund, Ravi P
Producer: 20100705
In:
Bioorganic & medicinal chemistry letters vol. 20
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227.
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Discovery and activity of (1R,4S,6R)-N-[(1R)-2-[4-cyclohexyl-4-[[(1,1-dimethylethyl)amino]carbonyl]-1-piperidinyl]-1-[(4-fluorophenyl)methyl]-2-oxoethyl]-2-methyl-2-azabicyclo[2.2.2]octane-6-carboxamide (3, RY764), a potent and selective melanocortin subtype-4 receptor agonist. [electronic resource] by
- Ye, Zhixiong
- Guo, Liangqin
- Barakat, Khaled J
- Pollard, Patrick G
- Palucki, Brenda L
- Sebhat, Iyassu K
- Bakshi, Raman K
- Tang, Rui
- Kalyani, Rubana N
- Vongs, Aurawan
- Chen, Airu S
- Chen, Howard Y
- Rosenblum, Charles I
- MacNeil, Tanya
- Weinberg, David H
- Peng, Qianping
- Tamvakopoulos, Constantin
- Miller, Randy R
- Stearns, Ralph A
- Cashen, Doreen E
- Martin, William J
- Metzger, Joseph M
- Strack, Alison M
- MacIntyre, D Euan
- Van der Ploeg, Lex H T
- Patchett, Arthur A
- Wyvratt, Matthew J
- Nargund, Ravi P
Producer: 20051011
In:
Bioorganic & medicinal chemistry letters vol. 15
Availability: No items available.
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228.
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A role for the melanocortin 4 receptor in sexual function. [electronic resource] by
- Van der Ploeg, Lex H T
- Martin, William J
- Howard, Andrew D
- Nargund, Ravi P
- Austin, Christopher P
- Guan, Xiaoming
- Drisko, Jennifer
- Cashen, Doreen
- Sebhat, Iyassu
- Patchett, Arthur A
- Figueroa, David J
- DiLella, Anthony G
- Connolly, Brett M
- Weinberg, David H
- Tan, Carina P
- Palyha, Oksana C
- Pong, Sheng-Shung
- MacNeil, Tanya
- Rosenblum, Charles
- Vongs, Aurawan
- Tang, Rui
- Yu, Hong
- Sailer, Andreas W
- Fong, Tung Ming
- Huang, Cathy
- Tota, Michael R
- Chang, Ray S
- Stearns, Ralph
- Tamvakopoulos, Constantin
- Christ, George
- Drazen, Deborah L
- Spar, Brian D
- Nelson, Randy J
- MacIntyre, D Euan
Producer: 20020927
In:
Proceedings of the National Academy of Sciences of the United States of America vol. 99
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229.
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Whole-genome association study of bipolar disorder. [electronic resource] by
- Sklar, P
- Smoller, J W
- Fan, J
- Ferreira, M A R
- Perlis, R H
- Chambert, K
- Nimgaonkar, V L
- McQueen, M B
- Faraone, S V
- Kirby, A
- de Bakker, P I W
- Ogdie, M N
- Thase, M E
- Sachs, G S
- Todd-Brown, K
- Gabriel, S B
- Sougnez, C
- Gates, C
- Blumenstiel, B
- Defelice, M
- Ardlie, K G
- Franklin, J
- Muir, W J
- McGhee, K A
- MacIntyre, D J
- McLean, A
- VanBeck, M
- McQuillin, A
- Bass, N J
- Robinson, M
- Lawrence, J
- Anjorin, A
- Curtis, D
- Scolnick, E M
- Daly, M J
- Blackwood, D H
- Gurling, H M
- Purcell, S M
Producer: 20080806
In:
Molecular psychiatry vol. 13
Availability: No items available.
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230.
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Genome-wide association study of major depressive disorder: new results, meta-analysis, and lessons learned. [electronic resource] by
- Wray, N R
- Pergadia, M L
- Blackwood, D H R
- Penninx, B W J H
- Gordon, S D
- Nyholt, D R
- Ripke, S
- MacIntyre, D J
- McGhee, K A
- Maclean, A W
- Smit, J H
- Hottenga, J J
- Willemsen, G
- Middeldorp, C M
- de Geus, E J C
- Lewis, C M
- McGuffin, P
- Hickie, I B
- van den Oord, E J C G
- Liu, J Z
- Macgregor, S
- McEvoy, B P
- Byrne, E M
- Medland, S E
- Statham, D J
- Henders, A K
- Heath, A C
- Montgomery, G W
- Martin, N G
- Boomsma, D I
- Madden, P A F
- Sullivan, P F
Producer: 20120508
In:
Molecular psychiatry vol. 17
Availability: No items available.
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231.
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Genome-wide association for major depressive disorder: a possible role for the presynaptic protein piccolo. [electronic resource] by
- Sullivan, P F
- de Geus, E J C
- Willemsen, G
- James, M R
- Smit, J H
- Zandbelt, T
- Arolt, V
- Baune, B T
- Blackwood, D
- Cichon, S
- Coventry, W L
- Domschke, K
- Farmer, A
- Fava, M
- Gordon, S D
- He, Q
- Heath, A C
- Heutink, P
- Holsboer, F
- Hoogendijk, W J
- Hottenga, J J
- Hu, Y
- Kohli, M
- Lin, D
- Lucae, S
- Macintyre, D J
- Maier, W
- McGhee, K A
- McGuffin, P
- Montgomery, G W
- Muir, W J
- Nolen, W A
- Nöthen, M M
- Perlis, R H
- Pirlo, K
- Posthuma, D
- Rietschel, M
- Rizzu, P
- Schosser, A
- Smit, A B
- Smoller, J W
- Tzeng, J-Y
- van Dyck, R
- Verhage, M
- Zitman, F G
- Martin, N G
- Wray, N R
- Boomsma, D I
- Penninx, B W J H
Producer: 20090804
In:
Molecular psychiatry vol. 14
Availability: No items available.
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232.
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Genetic effects influencing risk for major depressive disorder in China and Europe. [electronic resource] by
- Bigdeli, T B
- Ripke, S
- Peterson, R E
- Trzaskowski, M
- Bacanu, S-A
- Abdellaoui, A
- Andlauer, T F M
- Beekman, A T F
- Berger, K
- Blackwood, D H R
- Boomsma, D I
- Breen, G
- Buttenschøn, H N
- Byrne, E M
- Cichon, S
- Clarke, T-K
- Couvy-Duchesne, B
- Craddock, N
- de Geus, E J C
- Degenhardt, F
- Dunn, E C
- Edwards, A C
- Fanous, A H
- Forstner, A J
- Frank, J
- Gill, M
- Gordon, S D
- Grabe, H J
- Hamilton, S P
- Hardiman, O
- Hayward, C
- Heath, A C
- Henders, A K
- Herms, S
- Hickie, I B
- Hoffmann, P
- Homuth, G
- Hottenga, J-J
- Ising, M
- Jansen, R
- Kloiber, S
- Knowles, J A
- Lang, M
- Li, Q S
- Lucae, S
- MacIntyre, D J
- Madden, P A F
- Martin, N G
- McGrath, P J
- McGuffin, P
- McIntosh, A M
- Medland, S E
- Mehta, D
- Middeldorp, C M
- Milaneschi, Y
- Montgomery, G W
- Mors, O
- Müller-Myhsok, B
- Nauck, M
- Nyholt, D R
- Nöthen, M M
- Owen, M J
- Penninx, B W J H
- Pergadia, M L
- Perlis, R H
- Peyrot, W J
- Porteous, D J
- Potash, J B
- Rice, J P
- Rietschel, M
- Riley, B P
- Rivera, M
- Schoevers, R
- Schulze, T G
- Shi, J
- Shyn, S I
- Smit, J H
- Smoller, J W
- Streit, F
- Strohmaier, J
- Teumer, A
- Treutlein, J
- Van der Auwera, S
- van Grootheest, G
- van Hemert, A M
- Völzke, H
- Webb, B T
- Weissman, M M
- Wellmann, J
- Willemsen, G
- Witt, S H
- Levinson, D F
- Lewis, C M
- Wray, N R
- Flint, J
- Sullivan, P F
- Kendler, K S
Producer: 20171116
In:
Translational psychiatry vol. 7
Availability: No items available.
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