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2181.
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Discovery, mechanism and metabolism studies of 2,3-difluorophenyl-linker-containing PARP1 inhibitors with enhanced in vivo efficacy for cancer therapy. [electronic resource] by
- Chen, Wenhua
- Guo, Ne
- Qi, Minghui
- Dai, Haiying
- Hong, Minghuang
- Guan, Longfei
- Huan, Xiajuan
- Song, Shanshan
- He, Jinxue
- Wang, Yingqing
- Xi, Yong
- Yang, Xinying
- Shen, Yanyan
- Su, Yi
- Sun, Yiming
- Gao, Yinglei
- Chen, Yi
- Ding, Jian
- Tang, Yun
- Ren, Guobin
- Miao, Zehong
- Li, Jian
Producer: 20171002
In:
European journal of medicinal chemistry vol. 138
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2185.
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2186.
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The CHK1 Inhibitor Prexasertib Exhibits Monotherapy Activity in High-Grade Serous Ovarian Cancer Models and Sensitizes to PARP Inhibition. [electronic resource] by
- Parmar, Kalindi
- Kochupurakkal, Bose S
- Lazaro, Jean-Bernard
- Wang, Zhigang C
- Palakurthi, Sangeetha
- Kirschmeier, Paul T
- Yang, Chunyu
- Sambel, Larissa A
- Färkkilä, Anniina
- Reznichenko, Elizaveta
- Reavis, Hunter D
- Dunn, Connor E
- Zou, Lee
- Do, Khanh T
- Konstantinopoulos, Panagiotis A
- Matulonis, Ursula A
- Liu, Joyce F
- D'Andrea, Alan D
- Shapiro, Geoffrey I
Producer: 20200921
In:
Clinical cancer research : an official journal of the American Association for Cancer Research vol. 25
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2187.
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Olaparib and temozolomide in desmoplastic small round cell tumors: a promising combination in vitro and in vivo. [electronic resource] by
- van Erp, Anke E M
- van Houdt, Laurens
- Hillebrandt-Roeffen, Melissa H S
- van Bree, Niek F H N
- Flucke, Uta E
- Mentzel, Thomas
- Shipley, Janet
- Desar, Ingrid M E
- Fleuren, Emmy D G
- Versleijen-Jonkers, Yvonne M H
- van der Graaf, Winette T A
Producer: 20200615
In:
Journal of cancer research and clinical oncology vol. 146
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2188.
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2189.
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2190.
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Tyrosine kinase inhibitor PTK/ZK enhances the antitumor effects of interferon-α/5-fluorouracil therapy for hepatocellular carcinoma cells. [electronic resource] by
- Murakami, Masahiro
- Kobayashi, Shogo
- Marubashi, Shigeru
- Tomimaru, Yoshito
- Noda, Takehiro
- Wada, Hiroshi
- Eguchi, Hidetoshi
- Takeda, Yutaka
- Tanemura, Masahiro
- Umeshita, Koji
- Doki, Yuichiro
- Mori, Masaki
- Nagano, Hiroaki
Producer: 20110609
In:
Annals of surgical oncology vol. 18
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2191.
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Poly(ADP)-ribose polymerase inhibition: frequent durable responses in BRCA carrier ovarian cancer correlating with platinum-free interval. [electronic resource] by
- Fong, Peter C
- Yap, Timothy A
- Boss, David S
- Carden, Craig P
- Mergui-Roelvink, Marja
- Gourley, Charlie
- De Greve, Jacques
- Lubinski, Jan
- Shanley, Susan
- Messiou, Christina
- A'Hern, Roger
- Tutt, Andrew
- Ashworth, Alan
- Stone, John
- Carmichael, James
- Schellens, Jan H M
- de Bono, Johann S
- Kaye, Stan B
Producer: 20100908
In:
Journal of clinical oncology : official journal of the American Society of Clinical Oncology vol. 28
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2192.
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2193.
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PDGFRA gene rearrangements are frequent genetic events in PDGFRA-amplified glioblastomas. [electronic resource] by
- Ozawa, Tatsuya
- Brennan, Cameron W
- Wang, Lu
- Squatrito, Massimo
- Sasayama, Takashi
- Nakada, Mitsutoshi
- Huse, Jason T
- Pedraza, Alicia
- Utsuki, Satoshi
- Yasui, Yoshie
- Tandon, Adesh
- Fomchenko, Elena I
- Oka, Hidehiro
- Levine, Ross L
- Fujii, Kiyotaka
- Ladanyi, Marc
- Holland, Eric C
Producer: 20101008
In:
Genes & development vol. 24
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2194.
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Combined inhibition of Wee1 and PARP1/2 for radiosensitization in pancreatic cancer. [electronic resource] by
- Karnak, David
- Engelke, Carl G
- Parsels, Leslie A
- Kausar, Tasneem
- Wei, Dongping
- Robertson, Jordan R
- Marsh, Katherine B
- Davis, Mary A
- Zhao, Lili
- Maybaum, Jonathan
- Lawrence, Theodore S
- Morgan, Meredith A
Producer: 20150625
In:
Clinical cancer research : an official journal of the American Association for Cancer Research vol. 20
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2195.
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2196.
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Improved Therapeutic Window in [electronic resource] by
- Zhong, Haihong
- Chen, Cui
- Tammali, Ravinder
- Breen, Shannon
- Zhang, Jing
- Fazenbaker, Christine
- Kennedy, Maureen
- Conway, James
- Higgs, Brandon W
- Holoweckyj, Nicholas
- Raja, Rajiv
- Harper, Jay
- Pierce, Andrew J
- Herbst, Ronald
- Tice, David A
Producer: 20191125
In:
Molecular cancer therapeutics vol. 18
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2197.
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2198.
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A Subset of Colorectal Cancers with Cross-Sensitivity to Olaparib and Oxaliplatin. [electronic resource] by
- Arena, Sabrina
- Corti, Giorgio
- Durinikova, Erika
- Montone, Monica
- Reilly, Nicole M
- Russo, Mariangela
- Lorenzato, Annalisa
- Arcella, Pamela
- Lazzari, Luca
- Rospo, Giuseppe
- Pagani, Massimiliano
- Cancelliere, Carlotta
- Negrino, Carola
- Isella, Claudio
- Bartolini, Alice
- Cassingena, Andrea
- Amatu, Alessio
- Mauri, Gianluca
- Sartore-Bianchi, Andrea
- Mittica, Gloria
- Medico, Enzo
- Marsoni, Silvia
- Linnebacher, Michael
- Abrignani, Sergio
- Siena, Salvatore
- Di Nicolantonio, Federica
- Bardelli, Alberto
Producer: 20210114
In:
Clinical cancer research : an official journal of the American Association for Cancer Research vol. 26
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2200.
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