Results
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2181.
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RNA-dependent chromatin targeting of TET2 for endogenous retrovirus control in pluripotent stem cells. [electronic resource] by
- Guallar, Diana
- Bi, Xianju
- Pardavila, Jose Angel
- Huang, Xin
- Saenz, Carmen
- Shi, Xianle
- Zhou, Hongwei
- Faiola, Francesco
- Ding, Junjun
- Haruehanroengra, Phensinee
- Yang, Fan
- Li, Dan
- Sanchez-Priego, Carlos
- Saunders, Arven
- Pan, Feng
- Valdes, Victor Julian
- Kelley, Kevin
- Blanco, Miguel G
- Chen, Lingyi
- Wang, Huayan
- Sheng, Jia
- Xu, Mingjiang
- Fidalgo, Miguel
- Shen, Xiaohua
- Wang, Jianlong
Producer: 20190510
In:
Nature genetics vol. 50
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2182.
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Azole-based inhibitors of AKT/PKB for the treatment of cancer. [electronic resource] by
- Zeng, Qingping
- Allen, John G
- Bourbeau, Matthew P
- Wang, Xianghong
- Yao, Guomin
- Tadesse, Seifu
- Rider, James T
- Yuan, Chester C
- Hong, Fang-Tsao
- Lee, Matthew R
- Zhang, Shiwen
- Lofgren, Julie A
- Freeman, Daniel J
- Yang, Suijin
- Li, Chun
- Tominey, Elizabeth
- Huang, Xin
- Hoffman, Douglas
- Yamane, Harvey K
- Fotsch, Christopher
- Dominguez, Celia
- Hungate, Randall
- Zhang, Xiaoling
Producer: 20100527
In:
Bioorganic & medicinal chemistry letters vol. 20
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2183.
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Discovery of imidazopyridazines as potent Pim-1/2 kinase inhibitors. [electronic resource] by
- Wurz, Ryan P
- Sastri, Christine
- D'Amico, Derin C
- Herberich, Brad
- Jackson, Claire L M
- Pettus, Liping H
- Tasker, Andrew S
- Wu, Bin
- Guerrero, Nadia
- Lipford, J Russell
- Winston, Jeffrey T
- Yang, Yajing
- Wang, Paul
- Nguyen, Yen
- Andrews, Kristin L
- Huang, Xin
- Lee, Matthew R
- Mohr, Christopher
- Zhang, J D
- Reid, Darren L
- Xu, Yang
- Zhou, Yihong
- Wang, Hui-Ling
Producer: 20170626
In:
Bioorganic & medicinal chemistry letters vol. 26
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2184.
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Concurrent Chemoradiotherapy versus Intensity-modulated Radiotherapy Alone for Elderly Nasopharyngeal Carcinoma Patients with Pre-treatment Epstein-Barr Virus DNA: A Cohort Study in an Endemic Area with Long-term Follow-up. [electronic resource] by
- Yang, Qin
- Zhao, Ting-Ting
- Qiang, Meng-Yun
- Hu, Liang
- Lv, Xing
- Ye, Yan-Fang
- Ke, Liang-Ru
- Yu, Ya-Hui
- Qiu, Wen-Ze
- Liu, Guo-Ying
- Huang, Xin-Jun
- Li, Wang-Zhong
- Lv, Shu-Hui
- Sun, Yao
- Zhang, Lu-Yao
- Pei, Fei
- Guo, Xiang
- Xiang, Yan-Qun
- Qian, Chao-Nan
- Huang, Bi-Jun
- Xia, Wei-Xiong
Publication details: Journal of Cancer 2018
In:
Journal of Cancer vol. 9
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2185.
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Pyridyl-pyrimidine benzimidazole derivatives as potent, selective, and orally bioavailable inhibitors of Tie-2 kinase. [electronic resource] by
- Cee, Victor J
- Cheng, Alan C
- Romero, Karina
- Bellon, Steve
- Mohr, Christopher
- Whittington, Douglas A
- Bak, Annette
- Bready, James
- Caenepeel, Sean
- Coxon, Angela
- Deak, Holly L
- Fretland, Jenne
- Gu, Yan
- Hodous, Brian L
- Huang, Xin
- Kim, Joseph L
- Lin, Jasmine
- Long, Alexander M
- Nguyen, Hanh
- Olivieri, Philip R
- Patel, Vinod F
- Wang, Ling
- Zhou, Yihong
- Hughes, Paul
- Geuns-Meyer, Stephanie
Producer: 20090302
In:
Bioorganic & medicinal chemistry letters vol. 19
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2186.
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Structure-Based Design of Potent and Selective CK1γ Inhibitors. [electronic resource] by
- Huang, Hongbing
- Acquaviva, Lisa
- Berry, Virginia
- Bregman, Howard
- Chakka, Nagasree
- O'Connor, Anne
- DiMauro, Erin F
- Dovey, Jennifer
- Epstein, Oleg
- Grubinska, Barbara
- Goldstein, Jon
- Gunaydin, Hakan
- Hua, Zihao
- Huang, Xin
- Huang, Liyue
- Human, Jason
- Long, Alex
- Newcomb, John
- Patel, Vinod F
- Saffran, Doug
- Serafino, Randy
- Schneider, Steve
- Strathdee, Craig
- Tang, Jin
- Turci, Susan
- White, Ryan
- Yu, Violeta
- Zhao, Huilin
- Wilson, Cindy
- Martin, Matthew W
Producer: 20140605
In:
ACS medicinal chemistry letters vol. 3
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2187.
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Acalabrutinib in relapsed or refractory mantle cell lymphoma (ACE-LY-004): a single-arm, multicentre, phase 2 trial. [electronic resource] by
- Wang, Michael
- Rule, Simon
- Zinzani, Pier Luigi
- Goy, Andre
- Casasnovas, Olivier
- Smith, Stephen D
- Damaj, Gandhi
- Doorduijn, Jeanette
- Lamy, Thierry
- Morschhauser, Franck
- Panizo, Carlos
- Shah, Bijal
- Davies, Andrew
- Eek, Richard
- Dupuis, Jehan
- Jacobsen, Eric
- Kater, Arnon P
- Le Gouill, Steven
- Oberic, Lucie
- Robak, Taduesz
- Covey, Todd
- Dua, Richa
- Hamdy, Ahmed
- Huang, Xin
- Izumi, Raquel
- Patel, Priti
- Rothbaum, Wayne
- Slatter, J Greg
- Jurczak, Wojciech
Producer: 20180924
In:
Lancet (London, England) vol. 391
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2188.
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Phase 1/2 study of cyclin-dependent kinase (CDK)4/6 inhibitor palbociclib (PD-0332991) with bortezomib and dexamethasone in relapsed/refractory multiple myeloma. [electronic resource] by
- Niesvizky, Ruben
- Badros, Ashraf Z
- Costa, Luciano J
- Ely, Scott A
- Singhal, Seema B
- Stadtmauer, Edward A
- Haideri, Nisreen A
- Yacoub, Abdulraheem
- Hess, Georg
- Lentzsch, Suzanne
- Spicka, Ivan
- Chanan-Khan, Asher A
- Raab, Marc S
- Tarantolo, Stefano
- Vij, Ravi
- Zonder, Jeffrey A
- Huang, Xiangao
- Jayabalan, David
- Di Liberto, Maurizio
- Huang, Xin
- Jiang, Yuqiu
- Kim, Sindy T
- Randolph, Sophia
- Chen-Kiang, Selina
Producer: 20160920
In:
Leukemia & lymphoma vol. 56
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2189.
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Development of novel dual binders as potent, selective, and orally bioavailable tankyrase inhibitors. [electronic resource] by
- Hua, Zihao
- Bregman, Howard
- Buchanan, John L
- Chakka, Nagasree
- Guzman-Perez, Angel
- Gunaydin, Hakan
- Huang, Xin
- Gu, Yan
- Berry, Virginia
- Liu, Jingzhou
- Teffera, Yohannes
- Huang, Liyue
- Egge, Bryan
- Emkey, Renee
- Mullady, Erin L
- Schneider, Steve
- Andrews, Paul S
- Acquaviva, Lisa
- Dovey, Jennifer
- Mishra, Ankita
- Newcomb, John
- Saffran, Douglas
- Serafino, Randy
- Strathdee, Craig A
- Turci, Susan M
- Stanton, Mary
- Wilson, Cindy
- Dimauro, Erin F
Producer: 20140304
In:
Journal of medicinal chemistry vol. 56
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2190.
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Non-lab and semi-lab algorithms for screening undiagnosed diabetes: A cross-sectional study. [electronic resource] by
- Li, Wei
- Xie, Bo
- Qiu, Shanhu
- Huang, Xin
- Chen, Juan
- Wang, Xinling
- Li, Hong
- Chen, Qingyun
- Wang, Qing
- Tu, Ping
- Zhang, Lihui
- Yan, Sunjie
- Li, Kaili
- Maimaitiming, Jimilanmu
- Nian, Xin
- Liang, Min
- Wen, Yan
- Liu, Jiang
- Wang, Mian
- Zhang, Yongze
- Ma, Li
- Wu, Hang
- Wang, Xuyi
- Wang, Xiaohang
- Liu, Jingbao
- Cai, Min
- Wang, Zhiyao
- Guo, Lin
- Chen, Fangqun
- Wang, Bei
- Monica, Sandberg
- Carlsson, Per-Ola
- Sun, Zilin
Producer: 20190122
In:
EBioMedicine vol. 35
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2191.
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Discovery of Potent and Simplified Piperidinone-Based Inhibitors of the MDM2-p53 Interaction. [electronic resource] by
- Yu, Ming
- Wang, Yingcai
- Zhu, Jiang
- Bartberger, Michael D
- Canon, Jude
- Chen, Ada
- Chow, David
- Eksterowicz, John
- Fox, Brian
- Fu, Jiasheng
- Gribble, Michael
- Huang, Xin
- Li, Zhihong
- Liu, Jiwen Jim
- Lo, Mei-Chu
- McMinn, Dustin
- Oliner, Jonathan D
- Osgood, Tao
- Rew, Yosup
- Saiki, Anne Y
- Shaffer, Paul
- Yan, Xuelei
- Ye, Qiuping
- Yu, Dongyin
- Zhao, Xiaoning
- Zhou, Jing
- Olson, Steven H
- Medina, Julio C
- Sun, Daqing
Producer: 20140822
In:
ACS medicinal chemistry letters vol. 5
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2192.
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Genome sequence of the Asian Tiger mosquito, Aedes albopictus, reveals insights into its biology, genetics, and evolution. [electronic resource] by
- Chen, Xiao-Guang
- Jiang, Xuanting
- Gu, Jinbao
- Xu, Meng
- Wu, Yang
- Deng, Yuhua
- Zhang, Chi
- Bonizzoni, Mariangela
- Dermauw, Wannes
- Vontas, John
- Armbruster, Peter
- Huang, Xin
- Yang, Yulan
- Zhang, Hao
- He, Weiming
- Peng, Hongjuan
- Liu, Yongfeng
- Wu, Kun
- Chen, Jiahua
- Lirakis, Manolis
- Topalis, Pantelis
- Van Leeuwen, Thomas
- Hall, Andrew Brantley
- Jiang, Xiaofang
- Thorpe, Chevon
- Mueller, Rachel Lockridge
- Sun, Cheng
- Waterhouse, Robert Michael
- Yan, Guiyun
- Tu, Zhijian Jake
- Fang, Xiaodong
- James, Anthony A
Producer: 20160229
In:
Proceedings of the National Academy of Sciences of the United States of America vol. 112
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2193.
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Discovery and in Vivo Evaluation of Macrocyclic Mcl-1 Inhibitors Featuring an α-Hydroxy Phenylacetic Acid Pharmacophore or Bioisostere. [electronic resource] by
- Rescourio, Gwenaella
- Gonzalez, Ana Z
- Jabri, Salman
- Belmontes, Brian
- Moody, Gordon
- Whittington, Doug
- Huang, Xin
- Caenepeel, Sean
- Cardozo, Mario
- Cheng, Alan C
- Chow, David
- Dou, Hannah
- Jones, Adrie
- Kelly, Ron C
- Li, Yihong
- Lizarzaburu, Mike
- Lo, Mei-Chu
- Mallari, Rommel
- Meleza, Cesar
- Rew, Yosup
- Simonovich, Scott
- Sun, Daqing
- Turcotte, Simon
- Yan, Xuelei
- Wong, Simon G
- Yanez, Evelyn
- Zancanella, Manuel
- Houze, Jonathan
- Medina, Julio C
- Hughes, Paul E
- Brown, Sean P
Producer: 20200714
In:
Journal of medicinal chemistry vol. 62
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2194.
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Rational design and binding mode duality of MDM2-p53 inhibitors. [electronic resource] by
- Gonzalez-Lopez de Turiso, Felix
- Sun, Daqing
- Rew, Yosup
- Bartberger, Michael D
- Beck, Hilary P
- Canon, Jude
- Chen, Ada
- Chow, David
- Correll, Tiffany L
- Huang, Xin
- Julian, Lisa D
- Kayser, Frank
- Lo, Mei-Chu
- Long, Alexander M
- McMinn, Dustin
- Oliner, Jonathan D
- Osgood, Tao
- Powers, Jay P
- Saiki, Anne Y
- Schneider, Steve
- Shaffer, Paul
- Xiao, Shou-Hua
- Yakowec, Peter
- Yan, Xuelei
- Ye, Qiuping
- Yu, Dongyin
- Zhao, Xiaoning
- Zhou, Jing
- Medina, Julio C
- Olson, Steven H
Producer: 20130723
In:
Journal of medicinal chemistry vol. 56
Availability: No items available.
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2195.
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Structure-based design of novel 2-amino-6-phenyl-pyrimido[5',4':5,6]pyrimido[1,2-a]benzimidazol-5(6H)-ones as potent and orally active inhibitors of lymphocyte specific kinase (Lck): synthesis, SAR, and in vivo anti-inflammatory activity. [electronic resource] by
- Martin, Matthew W
- Newcomb, John
- Nunes, Joseph J
- Boucher, Christina
- Chai, Lilly
- Epstein, Linda F
- Faust, Theodore
- Flores, Sylvia
- Gallant, Paul
- Gore, Anu
- Gu, Yan
- Hsieh, Faye
- Huang, Xin
- Kim, Joseph L
- Middleton, Scot
- Morgenstern, Kurt
- Oliveira-dos-Santos, Antonio
- Patel, Vinod F
- Powers, David
- Rose, Paul
- Tudor, Yanyan
- Turci, Susan M
- Welcher, Andrew A
- Zack, Debra
- Zhao, Huilin
- Zhu, Li
- Zhu, Xiaotian
- Ghiron, Chiara
- Ermann, Monika
- Johnston, David
- Saluste, Carl-Gustaf Pierre
Producer: 20080611
In:
Journal of medicinal chemistry vol. 51
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2196.
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A dominant autoinflammatory disease caused by non-cleavable variants of RIPK1. [electronic resource] by
- Tao, Panfeng
- Sun, Jinqiao
- Wu, Zheming
- Wang, Shihao
- Wang, Jun
- Li, Wanjin
- Pan, Heling
- Bai, Renkui
- Zhang, Jiahui
- Wang, Ying
- Lee, Pui Y
- Ying, Wenjing
- Zhou, Qinhua
- Hou, Jia
- Wang, Wenjie
- Sun, Bijun
- Yang, Mi
- Liu, Danru
- Fang, Ran
- Han, Huan
- Yang, Zhaohui
- Huang, Xin
- Li, Haibo
- Deuitch, Natalie
- Zhang, Yuan
- Dissanayake, Dilan
- Haude, Katrina
- McWalter, Kirsty
- Roadhouse, Chelsea
- MacKenzie, Jennifer J
- Laxer, Ronald M
- Aksentijevich, Ivona
- Yu, Xiaomin
- Wang, Xiaochuan
- Yuan, Junying
- Zhou, Qing
Producer: 20200408
In:
Nature vol. 577
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2197.
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Activation of the STAT3 signaling pathway is associated with poor survival in diffuse large B-cell lymphoma treated with R-CHOP. [electronic resource] by
- Huang, Xin
- Meng, Bin
- Iqbal, Javeed
- Ding, B Belinda
- Perry, Anamarija M
- Cao, Wenfeng
- Smith, Lynette M
- Bi, Chengfeng
- Jiang, Chunsun
- Greiner, Timothy C
- Weisenburger, Dennis D
- Rimsza, Lisa
- Rosenwald, Andreas
- Ott, German
- Delabie, Jan
- Campo, Elias
- Braziel, Rita M
- Gascoyne, Randy D
- Cook, James R
- Tubbs, Raymond R
- Jaffe, Elaine S
- Armitage, James O
- Vose, Julie M
- Staudt, Louis M
- McKeithan, Timothy W
- Chan, Wing C
- Ye, B Hilda
- Fu, Kai
Producer: 20140224
In:
Journal of clinical oncology : official journal of the American Society of Clinical Oncology vol. 31
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2198.
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Global microRNA expression profiling uncovers molecular markers for classification and prognosis in aggressive B-cell lymphoma. [electronic resource] by
- Iqbal, Javeed
- Shen, Yulei
- Huang, Xin
- Liu, Yanyan
- Wake, Laura
- Liu, Cuiling
- Deffenbacher, Karen
- Lachel, Cynthia M
- Wang, Chao
- Rohr, Joseph
- Guo, Shuangping
- Smith, Lynette M
- Wright, George
- Bhagavathi, Sharathkumar
- Dybkaer, Karen
- Fu, Kai
- Greiner, Timothy C
- Vose, Julie M
- Jaffe, Elaine
- Rimsza, Lisa
- Rosenwald, Andreas
- Ott, German
- Delabie, Jan
- Campo, Elias
- Braziel, Rita M
- Cook, James R
- Tubbs, Raymond R
- Armitage, James O
- Weisenburger, Dennis D
- Staudt, Louis M
- Gascoyne, Randy D
- McKeithan, Timothy W
- Chan, Wing C
Producer: 20150421
In:
Blood vol. 125
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2199.
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The discovery of benzoxazine sulfonamide inhibitors of Na [electronic resource] by
- La, Daniel S
- Peterson, Emily A
- Bode, Christiane
- Boezio, Alessandro A
- Bregman, Howard
- Chu-Moyer, Margaret Y
- Coats, James
- DiMauro, Erin F
- Dineen, Thomas A
- Du, Bingfan
- Gao, Hua
- Graceffa, Russell
- Gunaydin, Hakan
- Guzman-Perez, Angel
- Fremeau, Robert
- Huang, Xin
- Ilch, Christopher
- Kornecook, Thomas J
- Kreiman, Charles
- Ligutti, Joseph
- Jasmine Lin, Min-Hwa
- McDermott, Jeff S
- Marx, Isaac
- Matson, David J
- McDonough, Stefan I
- Moyer, Bryan D
- Nho Nguyen, Hanh
- Taborn, Kristin
- Yu, Violeta
- Weiss, Matthew M
Producer: 20170818
In:
Bioorganic & medicinal chemistry letters vol. 27
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2200.
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Novel inhibitors of the MDM2-p53 interaction featuring hydrogen bond acceptors as carboxylic acid isosteres. [electronic resource] by
- Gonzalez, Ana Z
- Li, Zhihong
- Beck, Hilary P
- Canon, Jude
- Chen, Ada
- Chow, David
- Duquette, Jason
- Eksterowicz, John
- Fox, Brian M
- Fu, Jiasheng
- Huang, Xin
- Houze, Jonathan
- Jin, Lixia
- Li, Yihong
- Ling, Yun
- Lo, Mei-Chu
- Long, Alexander M
- McGee, Lawrence R
- McIntosh, Joel
- Oliner, Jonathan D
- Osgood, Tao
- Rew, Yosup
- Saiki, Anne Y
- Shaffer, Paul
- Wortman, Sarah
- Yakowec, Peter
- Yan, Xuelei
- Ye, Qiuping
- Yu, Dongyin
- Zhao, Xiaoning
- Zhou, Jing
- Olson, Steven H
- Sun, Daqing
- Medina, Julio C
Producer: 20140708
In:
Journal of medicinal chemistry vol. 57
Availability: No items available.
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