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Synthesis, biological evaluation and SAR study of novel pyrazole analogues as inhibitors of Mycobacterium tuberculosis. [electronic resource] by
- Castagnolo, Daniele
- De Logu, Alessandro
- Radi, Marco
- Bechi, Beatrice
- Manetti, Fabrizio
- Magnani, Matteo
- Supino, Sibilla
- Meleddu, Rita
- Chisu, Lorenza
- Botta, Maurizio
Producer: 20081205
In:
Bioorganic & medicinal chemistry vol. 16
Availability: No items available.
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Exploring the thiazole scaffold for the identification of new agents for the treatment of fluconazole resistant Candida. [electronic resource] by
- Meleddu, Rita
- Distinto, Simona
- Corona, Angela
- Maccioni, Elias
- Arridu, Antonella
- Melis, Claudia
- Bianco, Giulia
- Matyus, Peter
- Cottiglia, Filippo
- Sanna, Adriana
- De Logu, Alessandro
Producer: 20170306
In:
Journal of enzyme inhibition and medicinal chemistry vol. 31
Availability: No items available.
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28.
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In vivo potent BM635 analogue with improved drug-like properties. [electronic resource] by
- Poce, Giovanna
- Cocozza, Martina
- Alfonso, Salvatore
- Consalvi, Sara
- Venditti, Giulia
- Fernandez-Menendez, Raquel
- Bates, Robert H
- Barros Aguirre, David
- Ballell, Lluis
- De Logu, Alessandro
- Vistoli, Giulio
- Biava, Mariangela
Producer: 20180302
In:
European journal of medicinal chemistry vol. 145
Availability: No items available.
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29.
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Discovery of in vitro antitubercular agents through in silico ligand-based approaches. [electronic resource] by
- De Vita, Daniela
- Pandolfi, Fabiana
- Cirilli, Roberto
- Scipione, Luigi
- Di Santo, Roberto
- Friggeri, Laura
- Mori, Mattia
- Fiorucci, Diego
- Maccari, Giorgio
- Arul Christopher, Robert Selwyne
- Zamperini, Claudio
- Pau, Valentina
- De Logu, Alessandro
- Tortorella, Silvano
- Botta, Maurizio
Producer: 20170214
In:
European journal of medicinal chemistry vol. 121
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30.
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Naturally occurring Diels-Alder-type adducts from Morus nigra as potent inhibitors of Mycobacterium tuberculosis protein tyrosine phosphatase B. [electronic resource] by
- Mascarello, Alessandra
- Orbem Menegatti, Angela Camila
- Calcaterra, Andrea
- Martins, Priscila Graziela Alves
- Chiaradia-Delatorre, Louise Domeneghini
- D'Acquarica, Ilaria
- Ferrari, Franco
- Pau, Valentina
- Sanna, Adriana
- De Logu, Alessandro
- Botta, Maurizio
- Botta, Bruno
- Terenzi, Hernán
- Mori, Mattia
Producer: 20180223
In:
European journal of medicinal chemistry vol. 144
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31.
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Novel Pyrazole-Containing Compounds Active against [electronic resource] by
- Poce, Giovanna
- Consalvi, Sara
- Venditti, Giulia
- Alfonso, Salvatore
- Desideri, Nicoletta
- Fernandez-Menendez, Raquel
- Bates, Robert H
- Ballell, Lluis
- Barros Aguirre, David
- Rullas, Joaquin
- De Logu, Alessandro
- Gardner, Michelle
- Ioerger, Thomas R
- Rubin, Eric J
- Biava, Mariangela
Publication details: ACS medicinal chemistry letters Oct 2019
In:
ACS medicinal chemistry letters vol. 10
Availability: No items available.
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32.
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Improved BM212 MmpL3 inhibitor analogue shows efficacy in acute murine model of tuberculosis infection. [electronic resource] by
- Poce, Giovanna
- Bates, Robert H
- Alfonso, Salvatore
- Cocozza, Martina
- Porretta, Giulio Cesare
- Ballell, Lluís
- Rullas, Joaquin
- Ortega, Fátima
- De Logu, Alessandro
- Agus, Emanuela
- La Rosa, Valentina
- Pasca, Maria Rosalia
- De Rossi, Edda
- Wae, Baojie
- Franzblau, Scott G
- Manetti, Fabrizio
- Botta, Maurizio
- Biava, Mariangela
Producer: 20130823
In:
PloS one vol. 8
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MmpL3 is the cellular target of the antitubercular pyrrole derivative BM212. [electronic resource] by
- La Rosa, Valentina
- Poce, Giovanna
- Canseco, Julio Ortiz
- Buroni, Silvia
- Pasca, Maria Rosalia
- Biava, Mariangela
- Raju, Ravikiran M
- Porretta, Giulio Cesare
- Alfonso, Salvatore
- Battilocchio, Claudio
- Javid, Babak
- Sorrentino, Flavia
- Ioerger, Thomas R
- Sacchettini, James C
- Manetti, Fabrizio
- Botta, Maurizio
- De Logu, Alessandro
- Rubin, Eric J
- De Rossi, Edda
Producer: 20120802
In:
Antimicrobial agents and chemotherapy vol. 56
Availability: No items available.
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