Results
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21.
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Optimization of 1H-tetrazole-1-alkanenitriles as potent orally bioavailable growth hormone secretagogues. [electronic resource] by
- Hernández, Andrés S
- Swartz, Stephen G
- Slusarchyk, Dorothy
- Yan, Mujing
- Seethala, R Krishna
- Sleph, Paul
- Grover, Gary
- Dickinson, Kenneth
- Giupponi, Leah
- Harper, Timothy W
- Humphreys, W Griffith
- Longhi, Daniel A
- Flynn, Neil
- Murphy, Brian J
- Gordon, David A
- Biller, Scott A
- Robl, Jeffrey A
- Tino, Joseph A
Producer: 20080609
In:
Bioorganic & medicinal chemistry letters vol. 18
Availability: No items available.
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22.
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Potent and selective biphenyl azole inhibitors of adipocyte fatty acid binding protein (aFABP). [electronic resource] by
- Sulsky, Richard
- Magnin, David R
- Huang, Yanting
- Simpkins, Ligaya
- Taunk, Prakash
- Patel, Manorama
- Zhu, Yeheng
- Stouch, Terry R
- Bassolino-Klimas, Donna
- Parker, Rex
- Harrity, Thomas
- Stoffel, Robert
- Taylor, David S
- Lavoie, Thomas B
- Kish, Kevin
- Jacobson, Bruce L
- Sheriff, Steven
- Adam, Leonard P
- Ewing, William R
- Robl, Jeffrey A
Producer: 20070830
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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23.
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Discovery, synthesis, and structure-activity studies of tetrazole based growth hormone secretagogues. [electronic resource] by
- Hernández, Andrés S
- Cheng, Peter T W
- Musial, Christa M
- Swartz, Stephen G
- George, Rocco J
- Grover, Gary
- Slusarchyk, Dorothy
- Seethala, R Krishna
- Smith, Mark
- Dickinson, Kenneth
- Giupponi, Leah
- Longhi, Daniel A
- Flynn, Neil
- Murphy, Brian J
- Gordon, David A
- Biller, Scott A
- Robl, Jeffrey A
- Tino, Joseph A
Producer: 20080205
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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24.
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2-hydroxy-N-arylbenzenesulfonamides as ATP-citrate lyase inhibitors. [electronic resource] by
- Li, James J
- Wang, Haixia
- Tino, Joseph A
- Robl, Jeffrey A
- Herpin, Timothy F
- Lawrence, R Michael
- Biller, Scott
- Jamil, Haris
- Ponticiello, Randy
- Chen, Luping
- Chu, Ching-hsuen
- Flynn, Neil
- Cheng, Dong
- Zhao, Rulin
- Chen, Bangchi
- Schnur, Dora
- Obermeier, Mary T
- Sasseville, Vito
- Padmanabha, Ramesh
- Pike, Kristen
- Harrity, Thomas
Producer: 20070807
In:
Bioorganic & medicinal chemistry letters vol. 17
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25.
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Discovery of potent, orally-active, and muscle-selective androgen receptor modulators based on an N-aryl-hydroxybicyclohydantoin scaffold. [electronic resource] by
- Sun, Chongqing
- Robl, Jeffrey A
- Wang, Tammy C
- Huang, Yanting
- Kuhns, Joyce E
- Lupisella, John A
- Beehler, Blake C
- Golla, Rajasree
- Sleph, Paul G
- Seethala, Ramakrishna
- Fura, Aberra
- Krystek, Stanley R
- An, Yongmi
- Malley, Mary F
- Sack, John S
- Salvati, Mark E
- Grover, Gary J
- Ostrowski, Jacek
- Hamann, Lawrence G
Producer: 20070202
In:
Journal of medicinal chemistry vol. 49
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26.
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Synthesis and SAR of potent and selective tetrahydropyrazinoisoquinolinone 5-HT(2C) receptor agonists. [electronic resource] by
- Zhao, Guohua
- Kwon, Chet
- Bisaha, Sharon N
- Stein, Philip D
- Rossi, Karen A
- Cao, Xueying
- Ung, Thao
- Wu, Ginger
- Hung, Chen-Pin
- Malmstrom, Sarah E
- Zhang, Ge
- Qu, Qinling
- Gan, Jinping
- Keim, William J
- Cullen, Mary Jane
- Rohrbach, Kenneth W
- Devenny, James
- Pelleymounter, Mary Ann
- Miller, Keith J
- Robl, Jeffrey A
Producer: 20140113
In:
Bioorganic & medicinal chemistry letters vol. 23
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27.
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Optimization of 1,2,4-Triazolopyridines as Inhibitors of Human 11β-Hydroxysteroid Dehydrogenase Type 1 (11β-HSD-1). [electronic resource] by
- Li, Jun
- Kennedy, Lawrence J
- Wang, Haixia
- Li, James J
- Walker, Steven J
- Hong, Zhenqiu
- O'Connor, Stephen P
- Nayeem, Akbar
- Camac, Daniel M
- Morin, Paul E
- Sheriff, Steven
- Wang, Mengmeng
- Harper, Timothy
- Golla, Rajasree
- Seethala, Ramakrishna
- Harrity, Thomas
- Ponticiello, Randolph P
- Morgan, Nathan N
- Taylor, Joseph R
- Zebo, Rachel
- Gordon, David A
- Robl, Jeffrey A
Producer: 20140722
In:
ACS medicinal chemistry letters vol. 5
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28.
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Arylsulfonamidopiperidone derivatives as a novel class of factor Xa inhibitors. [electronic resource] by
- Shi, Yan
- O'Connor, Stephen P
- Sitkoff, Doree
- Zhang, Jing
- Shi, Mengxiao
- Bisaha, Sharon N
- Wang, Ying
- Li, Chi
- Ruan, Zheming
- Lawrence, R Michael
- Klei, Herbert E
- Kish, Kevin
- Liu, Eddie C-K
- Seiler, Steve M
- Schweizer, Liang
- Steinbacher, Thomas E
- Schumacher, William A
- Robl, Jeffrey A
- Macor, John E
- Atwal, Karnail S
- Stein, Philip D
Producer: 20120312
In:
Bioorganic & medicinal chemistry letters vol. 21
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29.
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Synthesis and Antiobesity Properties of 6-(4-Chlorophenyl)-3-(4-((3,3-difluoro-1-hydroxycyclobutyl)methoxy)-3-methoxyphenyl)thieno[3,2-d]pyrimidin-4(3H)-one (BMS-814580): A Highly Efficacious Melanin Concentrating Hormone Receptor 1 (MCHR1) Inhibitor. [electronic resource] by
- Ahmad, Saleem
- Washburn, William N
- Hernandez, Andres S
- Bisaha, Sharon
- Ngu, Khehyong
- Wang, Wei
- Pelleymounter, Mary Ann
- Longhi, Daniel
- Flynn, Neil
- Azzara, Anthony V
- Rohrbach, Kenneth
- Devenny, James
- Rooney, Suzanne
- Thomas, Michael
- Glick, Susan
- Godonis, Helen
- Harvey, Susan
- Zhang, Hongwei
- Gemzik, Brian
- Janovitz, Evan B
- Huang, Christine
- Zhang, Lisa
- Robl, Jeffrey A
- Murphy, Brian J
Producer: 20170619
In:
Journal of medicinal chemistry vol. 59
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30.
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Discovery of (R)-9-ethyl-1,3,4,10b-tetrahydro-7-trifluoromethylpyrazino[2,1-a]isoindol- 6(2H)-one, a selective, orally active agonist of the 5-HT(2C) receptor. [electronic resource] by
- Wacker, Dean A
- Varnes, Jeffrey G
- Malmstrom, Sarah E
- Cao, Xueying
- Hung, Chen-Pin
- Ung, Thao
- Wu, Ginger
- Zhang, Ge
- Zuvich, Eva
- Thomas, Michael A
- Keim, William J
- Cullen, Mary Jane
- Rohrbach, Kenneth W
- Qu, Qinling
- Narayanan, Rangaraj
- Rossi, Karen
- Janovitz, Evan
- Lehman-McKeeman, Lois
- Malley, Mary F
- Devenny, James
- Pelleymounter, Mary Ann
- Miller, Keith J
- Robl, Jeffrey A
Producer: 20070427
In:
Journal of medicinal chemistry vol. 50
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31.
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Discovery of brivanib alaninate ((S)-((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-methylpyrrolo[2,1-f][1,2,4]triazin-6-yloxy)propan-2-yl)2-aminopropanoate), a novel prodrug of dual vascular endothelial growth factor receptor-2 and fibroblast growth factor receptor-1 kinase inhibitor (BMS-540215). [electronic resource] by
- Cai, Zhen-wei
- Zhang, Yongzheng
- Borzilleri, Robert M
- Qian, Ligang
- Barbosa, Stephanie
- Wei, Donna
- Zheng, Xiaoping
- Wu, Lawrence
- Fan, Junying
- Shi, Zhongping
- Wautlet, Barri S
- Mortillo, Steve
- Jeyaseelan, Robert
- Kukral, Daniel W
- Kamath, Amrita
- Marathe, Punit
- D'Arienzo, Celia
- Derbin, George
- Barrish, Joel C
- Robl, Jeffrey A
- Hunt, John T
- Lombardo, Louis J
- Fargnoli, Joseph
- Bhide, Rajeev S
Producer: 20080611
In:
Journal of medicinal chemistry vol. 51
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32.
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Acridone-based inhibitors of inosine 5'-monophosphate dehydrogenase: discovery and SAR leading to the identification of N-(2-(6-(4-ethylpiperazin-1-yl)pyridin-3-yl)propan-2-yl)-2- fluoro-9-oxo-9,10-dihydroacridine-3-carboxamide (BMS-566419). [electronic resource] by
- Watterson, Scott H
- Chen, Ping
- Zhao, Yufen
- Gu, Henry H
- Dhar, T G Murali
- Xiao, Zili
- Ballentine, Shelley K
- Shen, Zhongqi
- Fleener, Catherine A
- Rouleau, Katherine A
- Obermeier, Mary
- Yang, Zheng
- McIntyre, Kim W
- Shuster, David J
- Witmer, Mark
- Dambach, Donna
- Chao, Sam
- Mathur, Arvind
- Chen, Bang-Chi
- Barrish, Joel C
- Robl, Jeffrey A
- Townsend, Robert
- Iwanowicz, Edwin J
Producer: 20071015
In:
Journal of medicinal chemistry vol. 50
Availability: No items available.
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33.
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Potent non-nitrile dipeptidic dipeptidyl peptidase IV inhibitors. [electronic resource] by
- Simpkins, Ligaya M
- Bolton, Scott
- Pi, Zulan
- Sutton, James C
- Kwon, Chet
- Zhao, Guohua
- Magnin, David R
- Augeri, David J
- Gungor, Timur
- Rotella, David P
- Sun, Zhong
- Liu, Yajun
- Slusarchyk, William S
- Marcinkeviciene, Jovita
- Robertson, James G
- Wang, Aiying
- Robl, Jeffrey A
- Atwal, Karnail S
- Zahler, Robert L
- Parker, Rex A
- Kirby, Mark S
- Hamann, Lawrence G
Producer: 20080303
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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34.
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The Guinea pig as a preclinical model for demonstrating the efficacy and safety of statins. [electronic resource] by
- Madsen, Cort S
- Janovitz, Evan
- Zhang, Rongan
- Nguyen-Tran, Van
- Ryan, Carol S
- Yin, Xiaohong
- Monshizadegan, Hossain
- Chang, Ming
- D'Arienzo, Celia
- Scheer, Susan
- Setters, Robert
- Search, Debra
- Chen, Xing
- Zhuang, Shaobin
- Kunselman, Lori
- Peters, Andrew
- Harrity, Thomas
- Apedo, Atsu
- Huang, Christine
- Cuff, Carolyn A
- Kowala, Mark C
- Blanar, Michael A
- Sun, Chong-Qing
- Robl, Jeffrey A
- Stein, Philip D
Producer: 20080219
In:
The Journal of pharmacology and experimental therapeutics vol. 324
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35.
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Design and synthesis of tetrazole-based growth hormone secretagogue: the SAR studies of the O-benzyl serine side chain. [electronic resource] by
- Li, Jun
- Chen, Stephanie Y
- Tao, Shiwei
- Wang, Haixia
- Li, James J
- Swartz, Steve
- Musial, Christa
- Hernandez, Andres A
- Flynn, Neil
- Murphy, Brian J
- Beehler, Blake
- Dickinson, Kenneth E
- Giupponi, Leah
- Grover, Gary
- Seethala, Ramakrishna
- Sleph, Paul
- Slusarchyk, Dorothy
- Yan, Mujing
- Humphreys, William G
- Zhang, Hongjian
- Ewing, William R
- Robl, Jeffrey A
- Gordon, David
- Tino, Joseph A
Producer: 20080609
In:
Bioorganic & medicinal chemistry letters vol. 18
Availability: No items available.
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36.
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Synthesis of novel potent dipeptidyl peptidase IV inhibitors with enhanced chemical stability: interplay between the N-terminal amino acid alkyl side chain and the cyclopropyl group of alpha-aminoacyl-l-cis-4,5-methanoprolinenitrile-based inhibitors. [electronic resource] by
- Magnin, David R
- Robl, Jeffrey A
- Sulsky, Richard B
- Augeri, David J
- Huang, Yanting
- Simpkins, Ligaya M
- Taunk, Prakash C
- Betebenner, David A
- Robertson, James G
- Abboa-Offei, Benoni E
- Wang, Aiying
- Cap, Michael
- Xin, Li
- Tao, Li
- Sitkoff, Doree F
- Malley, Mary F
- Gougoutas, Jack Z
- Khanna, Ashish
- Huang, Qi
- Han, Song-Ping
- Parker, Rex A
- Hamann, Lawrence G
Producer: 20040616
In:
Journal of medicinal chemistry vol. 47
Availability: No items available.
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37.
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Discovery and preclinical profile of Saxagliptin (BMS-477118): a highly potent, long-acting, orally active dipeptidyl peptidase IV inhibitor for the treatment of type 2 diabetes. [electronic resource] by
- Augeri, David J
- Robl, Jeffrey A
- Betebenner, David A
- Magnin, David R
- Khanna, Ashish
- Robertson, James G
- Wang, Aiying
- Simpkins, Ligaya M
- Taunk, Prakash
- Huang, Qi
- Han, Song-Ping
- Abboa-Offei, Benoni
- Cap, Michael
- Xin, Li
- Tao, Li
- Tozzo, Effie
- Welzel, Gustav E
- Egan, Donald M
- Marcinkeviciene, Jovita
- Chang, Shu Y
- Biller, Scott A
- Kirby, Mark S
- Parker, Rex A
- Hamann, Lawrence G
Producer: 20050823
In:
Journal of medicinal chemistry vol. 48
Availability: No items available.
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38.
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Utilization of an Active Site Mutant Receptor for the Identification of Potent and Selective Atypical 5-HT [electronic resource] by
- Carpenter, Joseph
- Wang, Ying
- Wu, Gang
- Feng, Jianxin
- Ye, Xiang-Yang
- Morales, Christian L
- Broekema, Matthias
- Rossi, Karen A
- Miller, Keith J
- Murphy, Brian J
- Wu, Ginger
- Malmstrom, Sarah E
- Azzara, Anthony V
- Sher, Philip M
- Fevig, John M
- Alt, Andrew
- Bertekap, Robert L
- Cullen, Mary Jane
- Harper, Timothy M
- Foster, Kimberly
- Luk, Emily
- Xiang, Qian
- Grubb, Mary F
- Robl, Jeffrey A
- Wacker, Dean A
Producer: 20170905
In:
Journal of medicinal chemistry vol. 60
Availability: No items available.
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39.
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11β-hydroxysteroid dehydrogenase type 1 gene knockout attenuates atherosclerosis and in vivo foam cell formation in hyperlipidemic apoE⁻/⁻ mice. [electronic resource] by
- García, Ricardo A
- Search, Debra J
- Lupisella, John A
- Ostrowski, Jacek
- Guan, Bo
- Chen, Jian
- Yang, Wen-Pin
- Truong, Amy
- He, Aiqing
- Zhang, Rongan
- Yan, Mujing
- Hellings, Samuel E
- Gargalovic, Peter S
- Ryan, Carol S
- Watson, Linda M
- Langish, Robert A
- Shipkova, Petia A
- Carson, Nancy L
- Taylor, Joseph R
- Yang, Richard
- Psaltis, George C
- Harrity, Thomas W
- Robl, Jeffrey A
- Gordon, David A
Producer: 20130715
In:
PloS one vol. 8
Availability: No items available.
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40.
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Pyridine amides as potent and selective inhibitors of 11beta-hydroxysteroid dehydrogenase type 1. [electronic resource] by
- Wang, Haixia
- Ruan, Zheming
- Li, James J
- Simpkins, Ligaya M
- Smirk, Rebecca A
- Wu, Shung C
- Hutchins, Robert D
- Nirschl, David S
- Van Kirk, Katy
- Cooper, Christopher B
- Sutton, James C
- Ma, Zhengping
- Golla, Rajasree
- Seethala, Ramakrishna
- Salyan, Mary Ellen K
- Nayeem, Akbar
- Krystek, Stanley R
- Sheriff, Steven
- Camac, Daniel M
- Morin, Paul E
- Carpenter, Brian
- Robl, Jeffrey A
- Zahler, Robert
- Gordon, David A
- Hamann, Lawrence G
Producer: 20080709
In:
Bioorganic & medicinal chemistry letters vol. 18
Availability: No items available.
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