Results
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21.
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Phase I Population Pharmacokinetic Assessment of the Oral Bromodomain Inhibitor OTX015 in Patients with Haematologic Malignancies. [electronic resource] by
- Odore, Elodie
- Lokiec, François
- Cvitkovic, Esteban
- Bekradda, Mohamed
- Herait, Patrice
- Bourdel, Fabrice
- Kahatt, Carmen
- Raffoux, Emmanuel
- Stathis, Anastasios
- Thieblemont, Catherine
- Quesnel, Bruno
- Cunningham, David
- Riveiro, Maria E
- Rezaï, Keyvan
Producer: 20161114
In:
Clinical pharmacokinetics vol. 55
Availability: No items available.
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22.
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Safety, pharmacokinetics, and activity of EZN-2208, a novel conjugate of polyethylene glycol and SN38, in patients with advanced malignancies. [electronic resource] by
- Kurzrock, Razelle
- Goel, Sanjay
- Wheler, Jennifer
- Hong, David
- Fu, Siqing
- Rezai, Keyvan
- Morgan-Linnell, Sonia K
- Urien, Saik
- Mani, Sridhar
- Chaudhary, Imran
- Ghalib, Mohammed H
- Buchbinder, Aby
- Lokiec, François
- Mulcahy, Mary
Producer: 20130205
In:
Cancer vol. 118
Availability: No items available.
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23.
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The bromodomain inhibitor OTX015 (MK-8628) exerts anti-tumor activity in triple-negative breast cancer models as single agent and in combination with everolimus. [electronic resource] by
- Vázquez, Ramiro
- Riveiro, María E
- Astorgues-Xerri, Lucile
- Odore, Elodie
- Rezai, Keyvan
- Erba, Eugenio
- Panini, Nicolò
- Rinaldi, Andrea
- Kwee, Ivo
- Beltrame, Luca
- Bekradda, Mohamed
- Cvitkovic, Esteban
- Bertoni, Francesco
- Frapolli, Roberta
- D'Incalci, Maurizio
Producer: 20180302
In:
Oncotarget vol. 8
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24.
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Phase Ib Trial With Birabresib, a Small-Molecule Inhibitor of Bromodomain and Extraterminal Proteins, in Patients With Selected Advanced Solid Tumors. [electronic resource] by
- Lewin, Jeremy
- Soria, Jean-Charles
- Stathis, Anastasios
- Delord, Jean-Pierre
- Peters, Solange
- Awada, Ahmad
- Aftimos, Philippe G
- Bekradda, Mohamed
- Rezai, Keyvan
- Zeng, Zhen
- Hussain, Azher
- Perez, Susan
- Siu, Lillian L
- Massard, Christophe
Producer: 20190913
In:
Journal of clinical oncology : official journal of the American Society of Clinical Oncology vol. 36
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25.
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OTX015 (MK-8628), a novel BET inhibitor, exhibits antitumor activity in non-small cell and small cell lung cancer models harboring different oncogenic mutations. [electronic resource] by
- Riveiro, Maria E
- Astorgues-Xerri, Lucile
- Vazquez, Ramiro
- Frapolli, Roberta
- Kwee, Ivo
- Rinaldi, Andrea
- Odore, Elodie
- Rezai, Keyvan
- Bekradda, Mohamed
- Inghirami, Giorgio
- D'Incalci, Maurizio
- Noel, Kay
- Cvitkovic, Esteban
- Raymond, Eric
- Bertoni, Francesco
Producer: 20180223
In:
Oncotarget vol. 7
Availability: No items available.
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26.
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Bromodomain inhibitor OTX015 in patients with acute leukaemia: a dose-escalation, phase 1 study. [electronic resource] by
- Berthon, Céline
- Raffoux, Emmanuel
- Thomas, Xavier
- Vey, Norbert
- Gomez-Roca, Carlos
- Yee, Karen
- Taussig, David Christopher
- Rezai, Keyvan
- Roumier, Christophe
- Herait, Patrice
- Kahatt, Carmen
- Quesnel, Bruno
- Michallet, Mauricette
- Recher, Christian
- Lokiec, François
- Preudhomme, Claude
- Dombret, Hervé
Producer: 20171018
In:
The Lancet. Haematology vol. 3
Availability: No items available.
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27.
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Insights into the cellular pharmacological properties of the BET-inhibitor OTX015/MK-8628 (birabresib), alone and in combination, in leukemia models. [electronic resource] by
- Astorgues-Xerri, Lucile
- Vázquez, Ramiro
- Odore, Elodie
- Rezai, Keyvan
- Kahatt, Carmen
- Mackenzie, Sarah
- Bekradda, Mohamed
- Coudé, Marie-Magdelaine
- Dombret, Herve
- Gardin, Claude
- Lokiec, Francois
- Raymond, Eric
- Noel, Kay
- Cvitkovic, Esteban
- Herait, Patrice
- Bertoni, Francesco
- Riveiro, María E
Producer: 20200910
In:
Leukemia & lymphoma vol. 60
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28.
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PIKHER2: A phase IB study evaluating buparlisib in combination with lapatinib in trastuzumab-resistant HER2-positive advanced breast cancer. [electronic resource] by
- Guerin, Mathilde
- Rezai, Keyvan
- Isambert, Nicolas
- Campone, Mario
- Autret, Aurélie
- Pakradouni, Jihane
- Provansal, Magali
- Camerlo, Jacques
- Sabatier, Renaud
- Bertucci, François
- Charafe-Jauffret, Emmanuelle
- Hervieu, Alice
- Extra, Jean-Marc
- Viens, Patrice
- Lokiec, François
- Boher, Jean-Marie
- Gonçalves, Anthony
Producer: 20171121
In:
European journal of cancer (Oxford, England : 1990) vol. 86
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29.
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Bromodomain inhibitor OTX015 in patients with lymphoma or multiple myeloma: a dose-escalation, open-label, pharmacokinetic, phase 1 study. [electronic resource] by
- Amorim, Sandy
- Stathis, Anastasios
- Gleeson, Mary
- Iyengar, Sunil
- Magarotto, Valeria
- Leleu, Xavier
- Morschhauser, Franck
- Karlin, Lionel
- Broussais, Florence
- Rezai, Keyvan
- Herait, Patrice
- Kahatt, Carmen
- Lokiec, François
- Salles, Gilles
- Facon, Thierry
- Palumbo, Antonio
- Cunningham, David
- Zucca, Emanuele
- Thieblemont, Catherine
Producer: 20171018
In:
The Lancet. Haematology vol. 3
Availability: No items available.
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30.
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BET bromodomain inhibitor birabresib in mantle cell lymphoma: in vivo activity and identification of novel combinations to overcome adaptive resistance. [electronic resource] by
- Tarantelli, Chiara
- Bernasconi, Elena
- Gaudio, Eugenio
- Cascione, Luciano
- Restelli, Valentina
- Arribas, Alberto Jesus
- Spriano, Filippo
- Rinaldi, Andrea
- Mensah, Afua Adjeiwaa
- Kwee, Ivo
- Ponzoni, Maurilio
- Zucca, Emanuele
- Carrassa, Laura
- Riveiro, Maria E
- Rezai, Keyvan
- Stathis, Anastasios
- Cvitkovic, Esteban
- Bertoni, Francesco
Publication details: ESMO open 2018
In:
ESMO open vol. 3
Availability: No items available.
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31.
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Phase I study of onapristone, a type I antiprogestin, in female patients with previously treated recurrent or metastatic progesterone receptor-expressing cancers. [electronic resource] by
- Cottu, Paul H
- Bonneterre, Jacques
- Varga, Andrea
- Campone, Mario
- Leary, Alexandra
- Floquet, Anne
- Berton-Rigaud, Dominique
- Sablin, Marie-Paule
- Lesoin, Anne
- Rezai, Keyvan
- Lokiec, François M
- Lhomme, Catherine
- Bosq, Jacques
- Bexon, Alice S
- Gilles, Erard M
- Proniuk, Stefan
- Dieras, Veronique
- Jackson, David M
- Zukiwski, Alexander
- Italiano, Antoine
Producer: 20190319
In:
PloS one vol. 13
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32.
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Epigenetic Control of Mitochondrial Fission Enables Self-Renewal of Stem-like Tumor Cells in Human Prostate Cancer. [electronic resource] by
- Civenni, Gianluca
- Bosotti, Roberto
- Timpanaro, Andrea
- Vàzquez, Ramiro
- Merulla, Jessica
- Pandit, Shusil
- Rossi, Simona
- Albino, Domenico
- Allegrini, Sara
- Mitra, Abhishek
- Mapelli, Sarah N
- Vierling, Luca
- Giurdanella, Martina
- Marchetti, Martina
- Paganoni, Alyssa
- Rinaldi, Andrea
- Losa, Marco
- Mira-Catò, Enrica
- D'Antuono, Rocco
- Morone, Diego
- Rezai, Keyvan
- D'Ambrosio, Gioacchino
- Ouafik, L'Houcine
- Mackenzie, Sarah
- Riveiro, Maria E
- Cvitkovic, Esteban
- Carbone, Giuseppina M
- Catapano, Carlo V
Producer: 20201001
In:
Cell metabolism vol. 30
Availability: No items available.
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