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Conformational mimetics of the α-methyl chalcone TUB091 binding tubulin: Design, synthesis and antiproliferative activity. [electronic resource] by
- Bueno, Oskía
- Tobajas, Gloria
- Quesada, Ernesto
- Estévez-Gallego, Juan
- Noppen, Sam
- Camarasa, María-José
- Díaz, José-Fernando
- Liekens, Sandra
- Priego, Eva-María
- Pérez-Pérez, María-Jesús
Producer: 20180323
In:
European journal of medicinal chemistry vol. 148
Availability: No items available.
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The crystal structure of the BAR domain from human Bin1/amphiphysin II and its implications for molecular recognition. [electronic resource] by
- Casal, Eva
- Federici, Luca
- Zhang, Wei
- Fernandez-Recio, Juan
- Priego, Eva-Maria
- Miguel, Ricardo Nuñez
- DuHadaway, James B
- Prendergast, George C
- Luisi, Ben F
- Laue, Ernest D
Producer: 20061219
In:
Biochemistry vol. 45
Availability: No items available.
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Identification of a novel 2-oxindole fluorinated derivative as in vivo antitumor agent for prostate cancer acting via AMPK activation. [electronic resource] by
- Bort, Alicia
- Quesada, Sergio
- Ramos-Torres, Ágata
- Gargantilla, Marta
- Priego, Eva María
- Raynal, Sophie
- Lepifre, Franck
- Gasalla, Jose M
- Rodriguez-Henche, Nieves
- Castro, Ana
- Díaz-Laviada, Inés
Producer: 20191021
In:
Scientific reports vol. 8
Availability: No items available.
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27.
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High-affinity ligands of the colchicine domain in tubulin based on a structure-guided design. [electronic resource] by
- Bueno, Oskía
- Estévez Gallego, Juan
- Martins, Solange
- Prota, Andrea E
- Gago, Federico
- Gómez-SanJuan, Asier
- Camarasa, María-José
- Barasoain, Isabel
- Steinmetz, Michel O
- Díaz, J Fernando
- Pérez-Pérez, María-Jesús
- Liekens, Sandra
- Priego, Eva-María
Producer: 20190918
In:
Scientific reports vol. 8
Availability: No items available.
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28.
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Antiviral activity of [1,2,3]triazolo[4,5-d]pyrimidin-7(6H)-ones against chikungunya virus targeting the viral capping nsP1. [electronic resource] by
- Gigante, Alba
- Gómez-SanJuan, Asier
- Delang, Leen
- Li, Changqing
- Bueno, Oskía
- Gamo, Ana-María
- Priego, Eva-María
- Camarasa, María-José
- Jochmans, Dirk
- Leyssen, Pieter
- Decroly, Etienne
- Coutard, Bruno
- Querat, Gilles
- Neyts, Johan
- Pérez-Pérez, María-Jesús
Producer: 20180329
In:
Antiviral research vol. 144
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Chalcones and Chalcone-mimetic Derivatives as Notch Inhibitors in a Model of T-cell Acute Lymphoblastic Leukemia. [electronic resource] by
- Quaglio, Deborah
- Zhdanovskaya, Nadezda
- Tobajas, Gloria
- Cuartas, Viviana
- Balducci, Silvia
- Christodoulou, Michael S
- Fabrizi, Giancarlo
- Gargantilla, Marta
- Priego, Eva-María
- Carmona Pestaña, Álvaro
- Passarella, Daniele
- Screpanti, Isabella
- Botta, Bruno
- Palermo, Rocco
- Mori, Mattia
- Ghirga, Francesca
- Pérez-Pérez, María-Jesús
Publication details: ACS medicinal chemistry letters Apr 2019
In:
ACS medicinal chemistry letters vol. 10
Availability: No items available.
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30.
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Inhibition of the Replication of Different Strains of Chikungunya Virus by 3-Aryl-[1,2,3]triazolo[4,5- d]pyrimidin-7(6 H)-ones. [electronic resource] by
- Gómez-SanJuan, Asier
- Gamo, Ana-María
- Delang, Leen
- Pérez-Sánchez, Alfonso
- Amrun, Siti Naqiah
- Abdelnabi, Rana
- Jacobs, Sofie
- Priego, Eva-María
- Camarasa, María-José
- Jochmans, Dirk
- Leyssen, Pieter
- Ng, Lisa F P
- Querat, Gilles
- Neyts, Johan
- Pérez-Pérez, María-Jesús
Producer: 20190618
In:
ACS infectious diseases vol. 4
Availability: No items available.
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31.
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Antivascular and antitumor properties of the tubulin-binding chalcone TUB091. [electronic resource] by
- Canela, María-Dolores
- Noppen, Sam
- Bueno, Oskía
- Prota, Andrea E
- Bargsten, Katja
- Sáez-Calvo, Gonzalo
- Jimeno, María-Luisa
- Benkheil, Mohammed
- Ribatti, Domenico
- Velázquez, Sonsoles
- Camarasa, María-José
- Díaz, J Fernando
- Steinmetz, Michel O
- Priego, Eva-María
- Pérez-Pérez, María-Jesús
- Liekens, Sandra
Producer: 20171009
In:
Oncotarget vol. 8
Availability: No items available.
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