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21.
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Synthesis, cannabinoid receptor affinity, and molecular modeling studies of substituted 1-aryl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamides. [electronic resource] by
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- Cascio, Maria Grazia
- La Regina, Giuseppe
- Piscitelli, Francesco
- Lavecchia, Antonio
- Brizzi, Antonella
- Pasquini, Serena
- Botta, Maurizio
- Novellino, Ettore
- Di Marzo, Vincenzo
- Corelli, Federico
Producer: 20080611
In:
Journal of medicinal chemistry vol. 51
Availability: No items available.
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22.
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Indolylarylsulfones as HIV-1 non-nucleoside reverse transcriptase inhibitors: new cyclic substituents at indole-2-carboxamide. [electronic resource] by
- La Regina, Giuseppe
- Coluccia, Antonio
- Brancale, Andrea
- Piscitelli, Francesco
- Gatti, Valerio
- Maga, Giovanni
- Samuele, Alberta
- Pannecouque, Christophe
- Schols, Dominique
- Balzarini, Jan
- Novellino, Ettore
- Silvestri, Romano
Producer: 20110617
In:
Journal of medicinal chemistry vol. 54
Availability: No items available.
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23.
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Indolyl aryl sulfones as HIV-1 non-nucleoside reverse transcriptase inhibitors: role of two halogen atoms at the indole ring in developing new analogues with improved antiviral activity. [electronic resource] by
- Regina, Giuseppe La
- Coluccia, Antonio
- Piscitelli, Francesco
- Bergamini, Alberto
- Sinistro, Anna
- Cavazza, Antonella
- Maga, Giovanni
- Samuele, Alberta
- Zanoli, Samantha
- Novellino, Ettore
- Artico, Marino
- Silvestri, Romano
Producer: 20071121
In:
Journal of medicinal chemistry vol. 50
Availability: No items available.
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24.
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Discovery of brain-penetrant, orally bioavailable aminothienopyridazine inhibitors of tau aggregation. [electronic resource] by
- Ballatore, Carlo
- Brunden, Kurt R
- Piscitelli, Francesco
- James, Michael J
- Crowe, Alex
- Yao, Yuemang
- Hyde, Edward
- Trojanowski, John Q
- Lee, Virginia M-Y
- Smith, Amos B
Producer: 20100611
In:
Journal of medicinal chemistry vol. 53
Availability: No items available.
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25.
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Aminothienopyridazine inhibitors of tau aggregation: evaluation of structure-activity relationship leads to selection of candidates with desirable in vivo properties. [electronic resource] by
- Ballatore, Carlo
- Crowe, Alex
- Piscitelli, Francesco
- James, Michael
- Lou, Kevin
- Rossidivito, Gabrielle
- Yao, Yuemang
- Trojanowski, John Q
- Lee, Virginia M-Y
- Brunden, Kurt R
- Smith, Amos B
Producer: 20121102
In:
Bioorganic & medicinal chemistry vol. 20
Availability: No items available.
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26.
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Cyclopentane-1,3-dione: a novel isostere for the carboxylic acid functional group. Application to the design of potent thromboxane (A2) receptor antagonists. [electronic resource] by
- Ballatore, Carlo
- Soper, James H
- Piscitelli, Francesco
- James, Michael
- Huang, Longchuan
- Atasoylu, Onur
- Huryn, Donna M
- Trojanowski, John Q
- Lee, Virginia M-Y
- Brunden, Kurt R
- Smith, Amos B
Producer: 20111212
In:
Journal of medicinal chemistry vol. 54
Availability: No items available.
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27.
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New nitrogen containing substituents at the indole-2-carboxamide yield high potent and broad spectrum indolylarylsulfone HIV-1 non-nucleoside reverse transcriptase inhibitors. [electronic resource] by
- La Regina, Giuseppe
- Coluccia, Antonio
- Brancale, Andrea
- Piscitelli, Francesco
- Famiglini, Valeria
- Cosconati, Sandro
- Maga, Giovanni
- Samuele, Alberta
- Gonzalez, Emmanuel
- Clotet, Bonaventura
- Schols, Dominique
- Esté, José A
- Novellino, Ettore
- Silvestri, Romano
Producer: 20121009
In:
Journal of medicinal chemistry vol. 55
Availability: No items available.
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28.
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Design, molecular modeling, synthesis, and anti-HIV-1 activity of new indolyl aryl sulfones. Novel derivatives of the indole-2-carboxamide. [electronic resource] by
- Ragno, Rino
- Coluccia, Antonio
- La Regina, Giuseppe
- De Martino, Gabriella
- Piscitelli, Francesco
- Lavecchia, Antonio
- Novellino, Ettore
- Bergamini, Alberto
- Ciaprini, Chiara
- Sinistro, Anna
- Maga, Giovanni
- Crespan, Emanuele
- Artico, Marino
- Silvestri, Romano
Producer: 20060712
In:
Journal of medicinal chemistry vol. 49
Availability: No items available.
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29.
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1-Aryl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide: an effective scaffold for the design of either CB1 or CB2 receptor ligands. [electronic resource] by
- Piscitelli, Francesco
- Ligresti, Alessia
- La Regina, Giuseppe
- Gatti, Valerio
- Brizzi, Antonella
- Pasquini, Serena
- Allarà, Marco
- Carai, Mauro Antonio Maria
- Novellino, Ettore
- Colombo, Giancarlo
- Di Marzo, Vincenzo
- Corelli, Federico
- Silvestri, Romano
Producer: 20120213
In:
European journal of medicinal chemistry vol. 46
Availability: No items available.
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30.
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Indolylarylsulfones bearing natural and unnatural amino acids. Discovery of potent inhibitors of HIV-1 non-nucleoside wild type and resistant mutant strains reverse transcriptase and coxsackie B4 virus. [electronic resource] by
- Piscitelli, Francesco
- Coluccia, Antonio
- Brancale, Andrea
- La Regina, Giuseppe
- Sansone, Anna
- Giordano, Cesare
- Balzarini, Jan
- Maga, Giovanni
- Zanoli, Samantha
- Samuele, Alberta
- Cirilli, Roberto
- La Torre, Francesco
- Lavecchia, Antonio
- Novellino, Ettore
- Silvestri, Romano
Producer: 20090428
In:
Journal of medicinal chemistry vol. 52
Availability: No items available.
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31.
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Synthesis, cannabinoid receptor affinity, molecular modeling studies and in vivo pharmacological evaluation of new substituted 1-aryl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamides. 2. Effect of the 3-carboxamide substituent on the affinity and selectivity profile. [electronic resource] by
- Silvestri, Romano
- Ligresti, Alessia
- La Regina, Giuseppe
- Piscitelli, Francesco
- Gatti, Valerio
- Brizzi, Antonella
- Pasquini, Serena
- Lavecchia, Antonio
- Allarà, Marco
- Fantini, Noemi
- Carai, Mauro Antonio Maria
- Novellino, Ettore
- Colombo, Giancarlo
- Di Marzo, Vincenzo
- Corelli, Federico
Producer: 20091013
In:
Bioorganic & medicinal chemistry vol. 17
Availability: No items available.
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32.
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Arylthioindole inhibitors of tubulin polymerization. 3. Biological evaluation, structure-activity relationships and molecular modeling studies. [electronic resource] by
- La Regina, Giuseppe
- Edler, Michael C
- Brancale, Andrea
- Kandil, Sahar
- Coluccia, Antonio
- Piscitelli, Francesco
- Hamel, Ernest
- De Martino, Gabriella
- Matesanz, Ruth
- Díaz, José Fernando
- Scovassi, Anna Ivana
- Prosperi, Ennio
- Lavecchia, Antonio
- Novellino, Ettore
- Artico, Marino
- Silvestri, Romano
Producer: 20070815
In:
Journal of medicinal chemistry vol. 50
Availability: No items available.
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33.
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1-[(3-Aryloxy-3-aryl)propyl]-1H-imidazoles, new imidazoles with potent activity against Candida albicans and dermatophytes. Synthesis, structure-activity relationship, and molecular modeling studies. [electronic resource] by
- La Regina, Giuseppe
- D'Auria, Felicia Diodata
- Tafi, Andrea
- Piscitelli, Francesco
- Olla, Stefania
- Caporuscio, Fabiana
- Nencioni, Lucia
- Cirilli, Roberto
- La Torre, Francesco
- De Melo, Nadja Rodrigues
- Kelly, Steven L
- Lamb, David C
- Artico, Marino
- Botta, Maurizio
- Palamara, Anna Teresa
- Silvestri, Romano
Producer: 20080812
In:
Journal of medicinal chemistry vol. 51
Availability: No items available.
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34.
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Synthesis and biological evaluation of new N-alkyl 1-aryl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamides as cannabinoid receptor ligands. [electronic resource] by
- Silvestri, Romano
- Ligresti, Alessia
- La Regina, Giuseppe
- Piscitelli, Francesco
- Gatti, Valerio
- Lavecchia, Antonio
- Brizzi, Antonella
- Pasquini, Serena
- Allarà, Marco
- Fantini, Noemi
- Carai, Mauro Antonio Maria
- Bigogno, Chiara
- Rozio, Marco Giulio
- Sinisi, Roberta
- Novellino, Ettore
- Colombo, Giancarlo
- Di Marzo, Vincenzo
- Dondio, Giulio
- Corelli, Federico
Producer: 20110307
In:
European journal of medicinal chemistry vol. 45
Availability: No items available.
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35.
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New arylthioindoles and related bioisosteres at the sulfur bridging group. 4. Synthesis, tubulin polymerization, cell growth inhibition, and molecular modeling studies. [electronic resource] by
- La Regina, Giuseppe
- Sarkar, Taradas
- Bai, Ruoli
- Edler, Michael C
- Saletti, Roberto
- Coluccia, Antonio
- Piscitelli, Francesco
- Minelli, Lara
- Gatti, Valerio
- Mazzoccoli, Carmela
- Palermo, Vanessa
- Mazzoni, Cristina
- Falcone, Claudio
- Scovassi, Anna Ivana
- Giansanti, Vincenzo
- Campiglia, Pietro
- Porta, Amalia
- Maresca, Bruno
- Hamel, Ernest
- Brancale, Andrea
- Novellino, Ettore
- Silvestri, Romano
Producer: 20091231
In:
Journal of medicinal chemistry vol. 52
Availability: No items available.
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36.
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Design and synthesis of 2-heterocyclyl-3-arylthio-1H-indoles as potent tubulin polymerization and cell growth inhibitors with improved metabolic stability. [electronic resource] by
- La Regina, Giuseppe
- Bai, Ruoli
- Rensen, Willeke
- Coluccia, Antonio
- Piscitelli, Francesco
- Gatti, Valerio
- Bolognesi, Alessio
- Lavecchia, Antonio
- Granata, Ilaria
- Porta, Amalia
- Maresca, Bruno
- Soriani, Alessandra
- Iannitto, Maria Luisa
- Mariani, Marisa
- Santoni, Angela
- Brancale, Andrea
- Ferlini, Cristiano
- Dondio, Giulio
- Varasi, Mario
- Mercurio, Ciro
- Hamel, Ernest
- Lavia, Patrizia
- Novellino, Ettore
- Silvestri, Romano
Producer: 20120308
In:
Journal of medicinal chemistry vol. 54
Availability: No items available.
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37.
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Toward highly potent cancer agents by modulating the C-2 group of the arylthioindole class of tubulin polymerization inhibitors. [electronic resource] by
- La Regina, Giuseppe
- Bai, Ruoli
- Rensen, Whilelmina Maria
- Di Cesare, Erica
- Coluccia, Antonio
- Piscitelli, Francesco
- Famiglini, Valeria
- Reggio, Alessia
- Nalli, Marianna
- Pelliccia, Sveva
- Da Pozzo, Eleonora
- Costa, Barbara
- Granata, Ilaria
- Porta, Amalia
- Maresca, Bruno
- Soriani, Alessandra
- Iannitto, Maria Luisa
- Santoni, Angela
- Li, Junjie
- Miranda Cona, Marlein
- Chen, Feng
- Ni, Yicheng
- Brancale, Andrea
- Dondio, Giulio
- Vultaggio, Stefania
- Varasi, Mario
- Mercurio, Ciro
- Martini, Claudia
- Hamel, Ernest
- Lavia, Patrizia
- Novellino, Ettore
- Silvestri, Romano
Producer: 20130417
In:
Journal of medicinal chemistry vol. 56
Availability: No items available.
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