Results
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21.
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Synthesis, modelling, and antimitotic properties of tricyclic systems characterised by a 2-(5-Phenyl-1H-pyrrol-3-yl)-1,3,4-oxadiazole moiety. [electronic resource] by
- Pinna, Gérard A
- Murineddu, Gabriele
- Murruzzu, Caterina
- Zuco, Valentina
- Zunino, Franco
- Cappelletti, Graziella
- Artali, Roberto
- Cignarella, Giorgio
- Solano, Lucrezia
- Villa, Stefania
Producer: 20090806
In:
ChemMedChem vol. 4
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22.
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23.
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Tricyclic pyrazoles. Part 6. Benzofuro[3,2-c]pyrazole: a versatile architecture for CB2 selective ligands. [electronic resource] by
- Pinna, Giovanni
- Loriga, Giovanni
- Lazzari, Paolo
- Ruiu, Stefania
- Falzoi, Matteo
- Frau, Simona
- Pau, Amedeo
- Murineddu, Gabriele
- Asproni, Battistina
- Pinna, Gerard A
Producer: 20150330
In:
European journal of medicinal chemistry vol. 82
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24.
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Design of novel 3,6-diazabicyclo[3.1.1]heptane derivatives with potent and selective affinities for α4β2 neuronal nicotinic acetylcholine receptors. [electronic resource] by
- Deligia, Francesco
- Deiana, Valeria
- Gotti, Cecilia
- Lazzari, Paolo
- Bottazzi, Mirko E H
- Pucci, Luca
- Fasoli, Francesca
- Ragusa, Giulio
- Pinna, Gerard A
- Murineddu, Gabriele
Producer: 20160503
In:
European journal of medicinal chemistry vol. 103
Availability: No items available.
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25.
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Pyridinyl- and pyridazinyl-3,6-diazabicyclo[3.1.1]heptane-anilines: Novel selective ligands with subnanomolar affinity for α [electronic resource] by
- Deligia, Francesco
- Murineddu, Gabriele
- Gotti, Cecilia
- Ragusa, Giulio
- Fasoli, Francesca
- Sciaccaluga, Miriam
- Plutino, Simona
- Fucile, Sergio
- Loriga, Giovanni
- Asproni, Battistina
- Pinna, Gerard A
Producer: 20180619
In:
European journal of medicinal chemistry vol. 152
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26.
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27.
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Tricyclic Pyrazoles. Part 5. Novel 1,4-Dihydroindeno[1,2-c]pyrazole CB2 Ligands Using Molecular Hybridization Based on Scaffold Hopping. [electronic resource] by
- Murineddu, Gabriele
- Asproni, Battistina
- Ruiu, Stefania
- Deligia, Francesco
- Falzoi, Matteo
- Pau, Amedeo
- Thomas, Brian F
- Zhang, Yanan
- Pinna, Gérard A
- Pani, Luca
- Lazzari, Paolo
Producer: 20120823
In:
The open medicinal chemistry journal vol. 6
Availability: No items available.
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28.
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Tricyclic pyrazoles. 4. Synthesis and biological evaluation of analogues of the robust and selective CB2 cannabinoid ligand 1-(2',4'-dichlorophenyl)-6-methyl-N-piperidin-1-yl-1,4-dihydroindeno[1,2-c]pyrazole-3-carboxamide. [electronic resource] by
- Murineddu, Gabriele
- Lazzari, Paolo
- Ruiu, Stefania
- Sanna, Angela
- Loriga, Giovanni
- Manca, Ilaria
- Falzoi, Matteo
- Dessì, Christian
- Curzu, Maria M
- Chelucci, Giorgio
- Pani, Luca
- Pinna, Gérard A
Producer: 20070223
In:
Journal of medicinal chemistry vol. 49
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29.
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Synthesis, Pharmacological Evaluation, and Docking Studies of Novel Pyridazinone-Based Cannabinoid Receptor Type 2 Ligands. [electronic resource] by
- Ragusa, Giulio
- Bencivenni, Serena
- Morales, Paula
- Callaway, Tyra
- Hurst, Dow P
- Asproni, Battistina
- Merighi, Stefania
- Loriga, Giovanni
- Pinna, Gerard A
- Reggio, Patricia H
- Gessi, Stefania
- Murineddu, Gabriele
Producer: 20190624
In:
ChemMedChem vol. 13
Availability: No items available.
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30.
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Synthesis and pharmacological evaluation of novel 4-alkyl-5-thien-2'-yl pyrazole carboxamides. [electronic resource] by
- Lazzari, Paolo
- Pau, Amedeo
- Tambaro, Simone
- Asproni, Battistina
- Ruiu, Stefania
- Pinna, Giansalvo
- Mastinu, Andrea
- Curzu, Maria M
- Reali, Roberta
- Bottazzi, Mirko Emilio Heiner
- Pinna, Gérard A
- Murineddu, Gabriele
Producer: 20130606
In:
Central nervous system agents in medicinal chemistry vol. 12
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31.
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Tricyclic pyrazoles. Part 8. Synthesis, biological evaluation and modelling of tricyclic pyrazole carboxamides as potential CB2 receptor ligands with antagonist/inverse agonist properties. [electronic resource] by
- Deiana, Valeria
- Gómez-Cañas, María
- Pazos, M Ruth
- Fernández-Ruiz, Javier
- Asproni, Battistina
- Cichero, Elena
- Fossa, Paola
- Muñoz, Eduardo
- Deligia, Francesco
- Murineddu, Gabriele
- García-Arencibia, Moisés
- Pinna, Gerard A
Producer: 20161107
In:
European journal of medicinal chemistry vol. 112
Availability: No items available.
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32.
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Novel N-aryl nicotinamide derivatives: Taking stock on 3,6-diazabicyclo[3.1.1]heptanes as ligands for neuronal acetylcholine receptors. [electronic resource] by
- Murineddu, Gabriele
- Gotti, Cecilia
- Asproni, Battistina
- Corona, Paola
- Martinello, Katiuscia
- Plutino, Simona
- Fucile, Sergio
- Temml, Veronika
- Moretti, Milena
- Viani, Paola
- Schuster, Daniela
- Piras, Sandra
- Deligia, Francesco
- Pinna, Gerard A
Producer: 20191104
In:
European journal of medicinal chemistry vol. 180
Availability: No items available.
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33.
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Multitarget-directed tricyclic pyridazinones as G protein-coupled receptor ligands and cholinesterase inhibitors. [electronic resource] by
- Pau, Amedeo
- Catto, Marco
- Pinna, Giovanni
- Frau, Simona
- Murineddu, Gabriele
- Asproni, Battistina
- Curzu, Maria M
- Pisani, Leonardo
- Leonetti, Francesco
- Loza, Maria Isabel
- Brea, José
- Pinna, Gérard A
- Carotti, Angelo
Producer: 20160226
In:
ChemMedChem vol. 10
Availability: No items available.
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34.
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New pyridazinone-4-carboxamides as new cannabinoid receptor type-2 inverse agonists: Synthesis, pharmacological data and molecular docking. [electronic resource] by
- Ragusa, Giulio
- Gómez-Cañas, María
- Morales, Paula
- Rodríguez-Cueto, Carmen
- Pazos, María R
- Asproni, Battistina
- Cichero, Elena
- Fossa, Paola
- Pinna, Gerard A
- Jagerovic, Nadine
- Fernández-Ruiz, Javier
- Murineddu, Gabriele
Producer: 20170228
In:
European journal of medicinal chemistry vol. 127
Availability: No items available.
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35.
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Novel sulfenamides and sulfonamides based on pyridazinone and pyridazine scaffolds as CB [electronic resource] by
- Murineddu, Gabriele
- Deligia, Francesco
- Ragusa, Giulio
- García-Toscano, Laura
- Gómez-Cañas, María
- Asproni, Battistina
- Satta, Valentina
- Cichero, Elena
- Pazos, Ruth
- Fossa, Paola
- Loriga, Giovanni
- Fernández-Ruiz, Javier
- Pinna, Gerard A
Producer: 20180105
In:
Bioorganic & medicinal chemistry vol. 26
Availability: No items available.
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36.
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Synthesis, pharmacological evaluation and docking studies of pyrrole structure-based CB2 receptor antagonists. [electronic resource] by
- Ragusa, Giulio
- Gómez-Cañas, María
- Morales, Paula
- Hurst, Dow P
- Deligia, Francesco
- Pazos, Ruth
- Pinna, Gerard A
- Fernández-Ruiz, Javier
- Goya, Pilar
- Reggio, Patricia H
- Jagerovic, Nadine
- García-Arencibia, Moisés
- Murineddu, Gabriele
Producer: 20160524
In:
European journal of medicinal chemistry vol. 101
Availability: No items available.
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