Results
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Evidence for C-Cl/C-Br...pi interactions as an important contribution to protein-ligand binding affinity. [electronic resource] by
- Matter, Hans
- Nazaré, Marc
- Güssregen, Stefan
- Will, David W
- Schreuder, Herman
- Bauer, Armin
- Urmann, Matthias
- Ritter, Kurt
- Wagner, Michael
- Wehner, Volkmar
Producer: 20090619
In:
Angewandte Chemie (International ed. in English) vol. 48
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23.
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Fragment deconstruction of small, potent factor Xa inhibitors: exploring the superadditivity energetics of fragment linking in protein-ligand complexes. [electronic resource] by
- Nazaré, Marc
- Matter, Hans
- Will, David W
- Wagner, Michael
- Urmann, Matthias
- Czech, Jörg
- Schreuder, Herman
- Bauer, Armin
- Ritter, Kurt
- Wehner, Volkmar
Producer: 20120507
In:
Angewandte Chemie (International ed. in English) vol. 51
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Discovery of N-[4-(1H-Pyrazolo[3,4-b]pyrazin-6-yl)-phenyl]-sulfonamides as Highly Active and Selective SGK1 Inhibitors. [electronic resource] by
- Halland, Nis
- Schmidt, Friedemann
- Weiss, Tilo
- Saas, Joachim
- Li, Ziyu
- Czech, Jörg
- Dreyer, Matthias
- Hofmeister, Armin
- Mertsch, Katharina
- Dietz, Uwe
- Strübing, Carsten
- Nazare, Marc
Producer: 20150115
In:
ACS medicinal chemistry letters vol. 6
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26.
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Identification of high-affinity P2Y₁₂ antagonists based on a phenylpyrazole glutamic acid piperazine backbone. [electronic resource] by
- Zech, Gernot
- Hessler, Gerhard
- Evers, Andreas
- Weiss, Tilo
- Florian, Peter
- Just, Melitta
- Czech, Jörg
- Czechtizky, Werngard
- Görlitzer, Jochen
- Ruf, Sven
- Kohlmann, Markus
- Nazaré, Marc
Producer: 20130205
In:
Journal of medicinal chemistry vol. 55
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27.
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DOTAM derivatives as active cartilage-targeting drug carriers for the treatment of osteoarthritis. [electronic resource] by
- Hu, Hai-Yu
- Lim, Ngee-Han
- Ding-Pfennigdorff, Danping
- Saas, Joachim
- Wendt, K Ulrich
- Ritzeler, Olaf
- Nagase, Hideaki
- Plettenburg, Oliver
- Schultz, Carsten
- Nazare, Marc
Producer: 20160122
In:
Bioconjugate chemistry vol. 26
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28.
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Novel factor Xa inhibitors based on a 2-carboxyindole scaffold: SAR of P4 substituents in combination with a neutral P1 ligand. [electronic resource] by
- Nazaré, Marc
- Essrich, Melanie
- Will, David W
- Matter, Hans
- Ritter, Kurt
- Urmann, Matthias
- Bauer, Armin
- Schreuder, Herman
- Czech, Jörg
- Lorenz, Martin
- Laux, Volker
- Wehner, Volkmar
Producer: 20050223
In:
Bioorganic & medicinal chemistry letters vol. 14
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29.
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Use of a sequential high throughput screening assay to identify novel inhibitors of the eukaryotic SRP-Sec61 targeting/translocation pathway. [electronic resource] by
- Klein, Wolfgang
- Rutz, Claudia
- Eckhard, Jamina
- Provinciael, Becky
- Specker, Edgar
- Neuenschwander, Martin
- Kleinau, Gunnar
- Scheerer, Patrick
- von Kries, Jens-Peter
- Nazaré, Marc
- Vermeire, Kurt
- Schülein, Ralf
Producer: 20190507
In:
PloS one vol. 13
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30.
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Probing the subpockets of factor Xa reveals two binding modes for inhibitors based on a 2-carboxyindole scaffold: a study combining structure-activity relationship and X-ray crystallography. [electronic resource] by
- Nazaré, Marc
- Will, David W
- Matter, Hans
- Schreuder, Herman
- Ritter, Kurt
- Urmann, Matthias
- Essrich, Melanie
- Bauer, Armin
- Wagner, Michael
- Czech, Jörg
- Lorenz, Martin
- Laux, Volker
- Wehner, Volkmar
Producer: 20050816
In:
Journal of medicinal chemistry vol. 48
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31.
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Factor Xa inhibitors based on a 2-carboxyindole scaffold: SAR of neutral P1 substituents. [electronic resource] by
- Nazaré, Marc
- Essrich, Melanie
- Will, David W
- Matter, Hans
- Ritter, Kurt
- Urmann, Matthias
- Bauer, Armin
- Schreuder, Herman
- Dudda, Angela
- Czech, Jörg
- Lorenz, Martin
- Laux, Volker
- Wehner, Volkmar
Producer: 20050223
In:
Bioorganic & medicinal chemistry letters vol. 14
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32.
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5-Aryl-2-(naphtha-1-yl)sulfonamido-thiazol-4(5H)-ones as clathrin inhibitors. [electronic resource] by
- Robertson, Mark J
- Horatscheck, André
- Sauer, Samantha
- von Kleist, Lisa
- Baker, Jennifer R
- Stahlschmidt, Wiebke
- Nazaré, Marc
- Whiting, Ainslie
- Chau, Ngoc
- Robinson, Phillip J
- Haucke, Volker
- McCluskey, Adam
Producer: 20180216
In:
Organic & biomolecular chemistry vol. 14
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33.
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A New Highly Thyrotropin Receptor-Selective Small-Molecule Antagonist with Potential for the Treatment of Graves' Orbitopathy. [electronic resource] by
- Marcinkowski, Patrick
- Hoyer, Inna
- Specker, Edgar
- Furkert, Jens
- Rutz, Claudia
- Neuenschwander, Martin
- Sobottka, Sebastian
- Sun, Han
- Nazare, Marc
- Berchner-Pfannschmidt, Utta
- von Kries, Jens Peter
- Eckstein, Anja
- Schülein, Ralf
- Krause, Gerd
Producer: 20191206
In:
Thyroid : official journal of the American Thyroid Association vol. 29
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34.
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Discovery of a Novel Series of Tankyrase Inhibitors by a Hybridization Approach. [electronic resource] by
- Anumala, Upendra Rao
- Waaler, Jo
- Nkizinkiko, Yves
- Ignatev, Alexander
- Lazarow, Katina
- Lindemann, Peter
- Olsen, Petter Angell
- Murthy, Sudarshan
- Obaji, Ezeogo
- Majouga, Alexander G
- Leonov, Sergey
- von Kries, Jens Peter
- Lehtiö, Lari
- Krauss, Stefan
- Nazaré, Marc
Producer: 20190401
In:
Journal of medicinal chemistry vol. 60
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35.
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Temperature dependence of cross-effect dynamic nuclear polarization in rotating solids: advantages of elevated temperatures. [electronic resource] by
- Geiger, Michel-Andreas
- Orwick-Rydmark, Marcella
- Märker, Katharina
- Franks, W Trent
- Akhmetzyanov, Dmitry
- Stöppler, Daniel
- Zinke, Maximilian
- Specker, Edgar
- Nazaré, Marc
- Diehl, Anne
- van Rossum, Barth-Jan
- Aussenac, Fabien
- Prisner, Thomas
- Akbey, Ümit
- Oschkinat, Hartmut
Producer: 20180130
In:
Physical chemistry chemical physics : PCCP vol. 18
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36.
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Novel factor Xa inhibitors based on a benzoic acid scaffold and incorporating a neutral P1 ligand. [electronic resource] by
- Nazaré, Marc
- Matter, Hans
- Klingler, Otmar
- Al-Obeidi, Fahad
- Schreuder, Herman
- Zoller, Gerhard
- Czech, Jörg
- Lorenz, Martin
- Dudda, Angela
- Peyman, Anusch
- Nestler, Hans Peter
- Urmann, Matthias
- Bauer, Armin
- Laux, Volker
- Wehner, Volkmar
- Will, David W
Producer: 20050104
In:
Bioorganic & medicinal chemistry letters vol. 14
Availability: No items available.
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37.
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None [electronic resource] by
- Hu, Hai-Yu
- Lim, Ngee-Han
- Juretschke, Hans-Paul
- Ding-Pfennigdorff, Danping
- Florian, Peter
- Kohlmann, Markus
- Kandira, Abdullah
- Peter von Kries, Jens
- Saas, Joachim
- Rudolphi, Karl A
- Wendt, K Ulrich
- Nagase, Hideaki
- Plettenburg, Oliver
- Nazare, Marc
- Schultz, Carsten
Publication details: Chemical science Nov 2015
In:
Chemical science vol. 6
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38.
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N-[6-(4-butanoyl-5-methyl-1H-pyrazol-1-yl)pyridazin-3-yl]-5-chloro-1-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-1H-indole-3-carboxamide (SAR216471), a novel intravenous and oral, reversible, and directly acting P2Y12 antagonist. [electronic resource] by
- Boldron, Christophe
- Besse, Angélina
- Bordes, Marie-Françoise
- Tissandié, Stéphanie
- Yvon, Xavier
- Gau, Benjamin
- Badorc, Alain
- Rousseaux, Tristan
- Barré, Guillaume
- Meneyrol, Jérôme
- Zech, Gernot
- Nazare, Marc
- Fossey, Valérie
- Pflieger, Anne-Marie
- Bonnet-Lignon, Sandrine
- Millet, Laurence
- Briot, Christophe
- Dol, Frédérique
- Hérault, Jean-Pascal
- Savi, Pierre
- Lassalle, Gilbert
- Delesque, Nathalie
- Herbert, Jean-Marc
- Bono, Françoise
Producer: 20141203
In:
Journal of medicinal chemistry vol. 57
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39.
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A pharmacological master key mechanism that unlocks the selectivity filter gate in K [electronic resource] by
- Schewe, Marcus
- Sun, Han
- Mert, Ümit
- Mackenzie, Alexandra
- Pike, Ashley C W
- Schulz, Friederike
- Constantin, Cristina
- Vowinkel, Kirsty S
- Conrad, Linus J
- Kiper, Aytug K
- Gonzalez, Wendy
- Musinszki, Marianne
- Tegtmeier, Marie
- Pryde, David C
- Belabed, Hassane
- Nazare, Marc
- de Groot, Bert L
- Decher, Niels
- Fakler, Bernd
- Carpenter, Elisabeth P
- Tucker, Stephen J
- Baukrowitz, Thomas
Producer: 20190806
In:
Science (New York, N.Y.) vol. 363
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40.
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Mutant KRAS-driven cancers depend on PTPN11/SHP2 phosphatase. [electronic resource] by
- Ruess, Dietrich A
- Heynen, Guus J
- Ciecielski, Katrin J
- Ai, Jiaoyu
- Berninger, Alexandra
- Kabacaoglu, Derya
- Görgülü, Kivanc
- Dantes, Zahra
- Wörmann, Sonja M
- Diakopoulos, Kalliope N
- Karpathaki, Angeliki F
- Kowalska, Marlena
- Kaya-Aksoy, Ezgi
- Song, Liang
- van der Laan, Eveline A Zeeuw
- López-Alberca, María P
- Nazaré, Marc
- Reichert, Maximilian
- Saur, Dieter
- Erkan, Mert M
- Hopt, Ulrich T
- Sainz, Bruno
- Birchmeier, Walter
- Schmid, Roland M
- Lesina, Marina
- Algül, Hana
Producer: 20190510
In:
Nature medicine vol. 24
Availability: No items available.
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