Results
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21.
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Discovery of potent, selective, and orally bioavailable 3H-spiro[isobenzofuran-1,4'-piperidine] based melanocortin subtype-4 receptor agonists. [electronic resource] by
- Guo, Liangqin
- Ye, Zhixiong
- Liu, Jian
- He, Shuwen
- Bakshi, Raman K
- Sebhat, Iyassu K
- Dobbelaar, Peter H
- Hong, Qingmei
- Jian, Tianying
- Dellureficio, James P
- Tsou, Nancy N
- Ball, Richard G
- Weinberg, David H
- MacNeil, Tanya
- Tang, Rui
- Tamvakopoulos, Constantin
- Peng, Qianping
- Chen, Howard Y
- Chen, Airu S
- Martin, William J
- MacIntyre, D Euan
- Strack, Alison M
- Fong, Tung M
- Wyvratt, Matthew J
- Nargund, Ravi P
Producer: 20101110
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
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22.
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Melanin-concentrating hormone 1 receptor-deficient mice are lean, hyperactive, and hyperphagic and have altered metabolism. [electronic resource] by
- Marsh, Donald J
- Weingarth, Drew T
- Novi, Dawn E
- Chen, Howard Y
- Trumbauer, Myrna E
- Chen, Airu S
- Guan, Xiao-Ming
- Jiang, Michael M
- Feng, Yue
- Camacho, Ramon E
- Shen, Zhu
- Frazier, Easter G
- Yu, Hong
- Metzger, Joseph M
- Kuca, Stephanie J
- Shearman, Lauren P
- Gopal-Truter, Shobhna
- MacNeil, Douglas J
- Strack, Alison M
- MacIntyre, D Euan
- Van der Ploeg, Lex H T
- Qian, Su
Producer: 20020426
In:
Proceedings of the National Academy of Sciences of the United States of America vol. 99
Availability: No items available.
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23.
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The target of ezetimibe is Niemann-Pick C1-Like 1 (NPC1L1). [electronic resource] by
- Garcia-Calvo, Margarita
- Lisnock, JeanMarie
- Bull, Herbert G
- Hawes, Brian E
- Burnett, Duane A
- Braun, Matthew P
- Crona, James H
- Davis, Harry R
- Dean, Dennis C
- Detmers, Patricia A
- Graziano, Michael P
- Hughes, Meredith
- Macintyre, D Euan
- Ogawa, Anthony
- O'neill, Kim A
- Iyer, Sai Prasad N
- Shevell, Diane E
- Smith, Marsha M
- Tang, Yui S
- Makarewicz, Amanda M
- Ujjainwalla, Feroze
- Altmann, Scott W
- Chapman, Kevin T
- Thornberry, Nancy A
Producer: 20050727
In:
Proceedings of the National Academy of Sciences of the United States of America vol. 102
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24.
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Discovery of a piperazine urea based compound as a potent, selective, orally bioavailable melanocortin subtype-4 receptor partial agonist. [electronic resource] by
- Hong, Qingmei
- Bakshi, Raman K
- Palucki, Brenda L
- Park, Min K
- Ye, Zhixiong
- He, Shuwen
- Pollard, Patrick G
- Sebhat, Iyassu K
- Liu, Jian
- Guo, Liangqin
- Cashen, Doreen E
- Martin, William J
- Weinberg, David H
- MacNeil, Tanya
- Tang, Rui
- Tamvakopoulos, Constantin
- Peng, Qianping
- Miller, Randy R
- Stearns, Ralph A
- Chen, Howard Y
- Chen, Airu S
- Strack, Alison M
- Fong, Tung M
- MacIntyre, D Euan
- Wyvratt, Matthew J
- Nargund, Ravi P
Producer: 20110719
In:
Bioorganic & medicinal chemistry letters vol. 21
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25.
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Characterization of a novel and selective cannabinoid CB1 receptor inverse agonist, Imidazole 24b, in rodents. [electronic resource] by
- Shearman, Lauren P
- Stribling, D Sloan
- Camacho, Ramon E
- Rosko, Kimberly M
- Wang, Junying
- Tong, Sharon
- Feng, Yue
- Marsh, Donald J
- Yu, Hong
- Guan, Xiaoming
- Spann, Stephanie K
- Macneil, Douglas J
- Fong, Tung M
- Metzger, Joseph M
- Goulet, Mark T
- Hagmann, William K
- Plummer, Christopher W
- Finke, Paul E
- Mills, Sander G
- Shah, Shrenik K
- Truong, Quang
- Van der Ploeg, L H T
- Macintyre, D Euan
- Strack, Alison M
Producer: 20080415
In:
European journal of pharmacology vol. 579
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26.
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Design and pharmacology of N-[(3R)-1,2,3,4-tetrahydroisoquinolinium- 3-ylcarbonyl]-(1R)-1-(4-chlorobenzyl)- 2-[4-cyclohexyl-4-(1H-1,2,4-triazol- 1-ylmethyl)piperidin-1-yl]-2-oxoethylamine (1), a potent, selective, melanocortin subtype-4 receptor agonist. [electronic resource] by
- Sebhat, Iyassu K
- Martin, William J
- Ye, Zhixiong
- Barakat, Khaled
- Mosley, Ralph T
- Johnston, David B R
- Bakshi, Raman
- Palucki, Brenda
- Weinberg, David H
- MacNeil, Tanya
- Kalyani, Rubana N
- Tang, Rui
- Stearns, Ralph A
- Miller, Randy R
- Tamvakopoulos, Constantin
- Strack, Alison M
- McGowan, Erin
- Cashen, Doreen E
- Drisko, Jennifer E
- Hom, Gary J
- Howard, Andrew D
- MacIntyre, D Euan
- van der Ploeg, Lex H T
- Patchett, Arthur A
- Nargund, Ravi P
Producer: 20021105
In:
Journal of medicinal chemistry vol. 45
Availability: No items available.
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27.
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Discovery of (2S)-N-[(1R)-2-[4-cyclohexyl-4-[[(1,1-dimethylethyl)amino]carbonyl]-1-piperidinyl]-1-[(4-fluorophenyl)methyl]-2-oxoethyl]-4-methyl-2-piperazinecarboxamide (MB243), a potent and selective melanocortin subtype-4 receptor agonist. [electronic resource] by
- Palucki, Brenda L
- Park, Min K
- Nargund, Ravi P
- Ye, Zhixiong
- Sebhat, Iyassu K
- Pollard, Patrick G
- Kalyani, Rubana N
- Tang, Rui
- Macneil, Tanya
- Weinberg, David H
- Vongs, Aurawan
- Rosenblum, Charles I
- Doss, George A
- Miller, Randall R
- Stearns, Ralph A
- Peng, Qianping
- Tamvakopoulos, Constantin
- McGowan, Erin
- Martin, William J
- Metzger, Joseph M
- Shepherd, Cherrie A
- Strack, Alison M
- Macintyre, D Euan
- Van der Ploeg, Lex H T
- Patchett, Arthur A
Producer: 20050502
In:
Bioorganic & medicinal chemistry letters vol. 15
Availability: No items available.
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28.
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Antiobesity efficacy of a novel cannabinoid-1 receptor inverse agonist, N-[(1S,2S)-3-(4-chlorophenyl)-2-(3-cyanophenyl)-1-methylpropyl]-2-methyl-2-[[5-(trifluoromethyl)pyridin-2-yl]oxy]propanamide (MK-0364), in rodents. [electronic resource] by
- Fong, Tung M
- Guan, Xiao-Ming
- Marsh, Donald J
- Shen, Chun-Pyn
- Stribling, D Sloan
- Rosko, Kim M
- Lao, Julie
- Yu, Hong
- Feng, Yue
- Xiao, Jing C
- Van der Ploeg, Lex H T
- Goulet, Mark T
- Hagmann, Williams K
- Lin, Linus S
- Lanza, Thomas J
- Jewell, James P
- Liu, Ping
- Shah, Shrenik K
- Qi, Hongbo
- Tong, Xinchun
- Wang, Junying
- Xu, Suoyu S
- Francis, Barbara
- Strack, Alison M
- MacIntyre, D Euan
- Shearman, Lauren P
Producer: 20070730
In:
The Journal of pharmacology and experimental therapeutics vol. 321
Availability: No items available.
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29.
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Discovery of a spiroindane based compound as a potent, selective, orally bioavailable melanocortin subtype-4 receptor agonist. [electronic resource] by
- He, Shuwen
- Ye, Zhixiong
- Dobbelaar, Peter H
- Sebhat, Iyassu K
- Guo, Liangqin
- Liu, Jian
- Jian, Tianying
- Lai, Yingjie
- Franklin, Christopher L
- Bakshi, Raman K
- Dellureficio, James P
- Hong, Qingmei
- Tsou, Nancy N
- Ball, Richard G
- Cashen, Doreen E
- Martin, William J
- Weinberg, David H
- Macneil, Tanya
- Tang, Rui
- Tamvakopoulos, Constantin
- Peng, Qianping
- Miller, Randy R
- Stearns, Ralph A
- Chen, Howard Y
- Chen, Airu S
- Strack, Alison M
- Fong, Tung M
- Macintyre, D Euan
- Wyvratt, Matthew J
- Nargund, Ravi P
Producer: 20100705
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
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30.
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Discovery and activity of (1R,4S,6R)-N-[(1R)-2-[4-cyclohexyl-4-[[(1,1-dimethylethyl)amino]carbonyl]-1-piperidinyl]-1-[(4-fluorophenyl)methyl]-2-oxoethyl]-2-methyl-2-azabicyclo[2.2.2]octane-6-carboxamide (3, RY764), a potent and selective melanocortin subtype-4 receptor agonist. [electronic resource] by
- Ye, Zhixiong
- Guo, Liangqin
- Barakat, Khaled J
- Pollard, Patrick G
- Palucki, Brenda L
- Sebhat, Iyassu K
- Bakshi, Raman K
- Tang, Rui
- Kalyani, Rubana N
- Vongs, Aurawan
- Chen, Airu S
- Chen, Howard Y
- Rosenblum, Charles I
- MacNeil, Tanya
- Weinberg, David H
- Peng, Qianping
- Tamvakopoulos, Constantin
- Miller, Randy R
- Stearns, Ralph A
- Cashen, Doreen E
- Martin, William J
- Metzger, Joseph M
- Strack, Alison M
- MacIntyre, D Euan
- Van der Ploeg, Lex H T
- Patchett, Arthur A
- Wyvratt, Matthew J
- Nargund, Ravi P
Producer: 20051011
In:
Bioorganic & medicinal chemistry letters vol. 15
Availability: No items available.
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31.
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A role for the melanocortin 4 receptor in sexual function. [electronic resource] by
- Van der Ploeg, Lex H T
- Martin, William J
- Howard, Andrew D
- Nargund, Ravi P
- Austin, Christopher P
- Guan, Xiaoming
- Drisko, Jennifer
- Cashen, Doreen
- Sebhat, Iyassu
- Patchett, Arthur A
- Figueroa, David J
- DiLella, Anthony G
- Connolly, Brett M
- Weinberg, David H
- Tan, Carina P
- Palyha, Oksana C
- Pong, Sheng-Shung
- MacNeil, Tanya
- Rosenblum, Charles
- Vongs, Aurawan
- Tang, Rui
- Yu, Hong
- Sailer, Andreas W
- Fong, Tung Ming
- Huang, Cathy
- Tota, Michael R
- Chang, Ray S
- Stearns, Ralph
- Tamvakopoulos, Constantin
- Christ, George
- Drazen, Deborah L
- Spar, Brian D
- Nelson, Randy J
- MacIntyre, D Euan
Producer: 20020927
In:
Proceedings of the National Academy of Sciences of the United States of America vol. 99
Availability: No items available.
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