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Activities, crystal structures, and molecular dynamics of dihydro-1H-isoindole derivatives, inhibitors of HIV-1 integrase. [electronic resource] by
- Métifiot, Mathieu
- Maddali, Kasthuraiah
- Johnson, Barry C
- Hare, Stephen
- Smith, Steven J
- Zhao, Xue Zhi
- Marchand, Christophe
- Burke, Terrence R
- Hughes, Stephen H
- Cherepanov, Peter
- Pommier, Yves
Producer: 20130702
In:
ACS chemical biology vol. 8
Availability: No items available.
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28.
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Structure-Guided Optimization of HIV Integrase Strand Transfer Inhibitors. [electronic resource] by
- Zhao, Xue Zhi
- Smith, Steven J
- Maskell, Daniel P
- Métifiot, Mathieu
- Pye, Valerie E
- Fesen, Katherine
- Marchand, Christophe
- Pommier, Yves
- Cherepanov, Peter
- Hughes, Stephen H
- Burke, Terrence R
Producer: 20170926
In:
Journal of medicinal chemistry vol. 60
Availability: No items available.
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29.
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HIV-1 Integrase Strand Transfer Inhibitors with Reduced Susceptibility to Drug Resistant Mutant Integrases. [electronic resource] by
- Zhao, Xue Zhi
- Smith, Steven J
- Maskell, Daniel P
- Metifiot, Mathieu
- Pye, Valerie E
- Fesen, Katherine
- Marchand, Christophe
- Pommier, Yves
- Cherepanov, Peter
- Hughes, Stephen H
- Burke, Terrence R
Producer: 20161213
In:
ACS chemical biology vol. 11
Availability: No items available.
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30.
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6-(1-Benzyl-1H-pyrrol-2-yl)-2,4-dioxo-5-hexenoic acids as dual inhibitors of recombinant HIV-1 integrase and ribonuclease H, synthesized by a parallel synthesis approach. [electronic resource] by
- Costi, Roberta
- Métifiot, Mathieu
- Esposito, Francesca
- Cuzzucoli Crucitti, Giuliana
- Pescatori, Luca
- Messore, Antonella
- Scipione, Luigi
- Tortorella, Silvano
- Zinzula, Luca
- Novellino, Ettore
- Pommier, Yves
- Tramontano, Enzo
- Marchand, Christophe
- Di Santo, Roberto
Producer: 20140318
In:
Journal of medicinal chemistry vol. 56
Availability: No items available.
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31.
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Cell-permeable stapled peptides based on HIV-1 integrase inhibitors derived from HIV-1 gene products. [electronic resource] by
- Nomura, Wataru
- Aikawa, Haruo
- Ohashi, Nami
- Urano, Emiko
- Métifiot, Mathieu
- Fujino, Masayuki
- Maddali, Kasthuraiah
- Ozaki, Taro
- Nozue, Ami
- Narumi, Tetsuo
- Hashimoto, Chie
- Tanaka, Tomohiro
- Pommier, Yves
- Yamamoto, Naoki
- Komano, Jun A
- Murakami, Tsutomu
- Tamamura, Hirokazu
Producer: 20150226
In:
ACS chemical biology vol. 8
Availability: No items available.
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32.
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Structure-activity relationship of pyrrolyl diketo acid derivatives as dual inhibitors of HIV-1 integrase and reverse transcriptase ribonuclease H domain. [electronic resource] by
- Cuzzucoli Crucitti, Giuliana
- Métifiot, Mathieu
- Pescatori, Luca
- Messore, Antonella
- Madia, Valentina Noemi
- Pupo, Giovanni
- Saccoliti, Francesco
- Scipione, Luigi
- Tortorella, Silvano
- Esposito, Francesca
- Corona, Angela
- Cadeddu, Marta
- Marchand, Christophe
- Pommier, Yves
- Tramontano, Enzo
- Costi, Roberta
- Di Santo, Roberto
Producer: 20150507
In:
Journal of medicinal chemistry vol. 58
Availability: No items available.
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33.
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Basic quinolinonyl diketo acid derivatives as inhibitors of HIV integrase and their activity against RNase H function of reverse transcriptase. [electronic resource] by
- Costi, Roberta
- Métifiot, Mathieu
- Chung, Suhman
- Cuzzucoli Crucitti, Giuliana
- Maddali, Kasthuraiah
- Pescatori, Luca
- Messore, Antonella
- Madia, Valentina Noemi
- Pupo, Giovanni
- Scipione, Luigi
- Tortorella, Silvano
- Di Leva, Francesco Saverio
- Cosconati, Sandro
- Marinelli, Luciana
- Novellino, Ettore
- Le Grice, Stuart F J
- Corona, Angela
- Pommier, Yves
- Marchand, Christophe
- Di Santo, Roberto
Producer: 20140706
In:
Journal of medicinal chemistry vol. 57
Availability: No items available.
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34.
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N-Substituted Quinolinonyl Diketo Acid Derivatives as HIV Integrase Strand Transfer Inhibitors and Their Activity against RNase H Function of Reverse Transcriptase. [electronic resource] by
- Pescatori, Luca
- Métifiot, Mathieu
- Chung, Suhman
- Masoaka, Takashi
- Cuzzucoli Crucitti, Giuliana
- Messore, Antonella
- Pupo, Giovanni
- Madia, Valentina Noemi
- Saccoliti, Francesco
- Scipione, Luigi
- Tortorella, Silvano
- Di Leva, Francesco Saverio
- Cosconati, Sandro
- Marinelli, Luciana
- Novellino, Ettore
- Le Grice, Stuart F J
- Pommier, Yves
- Marchand, Christophe
- Costi, Roberta
- Di Santo, Roberto
Producer: 20150928
In:
Journal of medicinal chemistry vol. 58
Availability: No items available.
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