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Uncialamycin as a novel payload for antibody drug conjugate (ADC) based targeted cancer therapy. [electronic resource] by
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- Wang, Yichong
- Kwok, Eilene
- Passmore, David
- Rangan, Vangipuram S
- Deshpande, Shrikant
- Cardarelli, Pina
- Vite, Gregory
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Producer: 20191209
In:
Bioorganic & medicinal chemistry letters vol. 29
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A Functional Na [electronic resource] by
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- Post-Munson, Debra J
- Watson, John
- Langley, David R
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Producer: 20170830
In:
Molecular pharmacology vol. 92
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Discovery and development of hepatitis C virus NS5A replication complex inhibitors. [electronic resource] by
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- Sun, Jin-Hua
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Producer: 20140515
In:
Journal of medicinal chemistry vol. 57
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Respiratory syncytial virus fusion inhibitors. Part 5: Optimization of benzimidazole substitution patterns towards derivatives with improved activity. [electronic resource] by
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- Roach, Julia
- Li, Zhufang
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Producer: 20071121
In:
Bioorganic & medicinal chemistry letters vol. 17
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25.
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Novel 3',6'-anhydro and N12,N13-bridged glycosylated fluoroindolo[2,3-a]carbazoles as topoisomerase I inhibitors. Fluorine as a leaving group from sp3 carbon. [electronic resource] by
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- Zimmermann, Kurt
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Producer: 20060112
In:
Organic letters vol. 7
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26.
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2-(1H-Imidazol-4-yl)ethanamine and 2-(1H-pyrazol-1-yl)ethanamine side chain variants of the IGF-1R inhibitor BMS-536924. [electronic resource] by
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- Carboni, Joan
- Li, Aixin
- Greer, Ann
- Yang, Zheng
- Balimane, Praveen
- Gottardis, Marco
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Producer: 20080519
In:
Bioorganic & medicinal chemistry letters vol. 18
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27.
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Balancing oral exposure with Cyp3A4 inhibition in benzimidazole-based IGF-IR inhibitors. [electronic resource] by
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- Li, Aixin
- Greer, Ann
- Gottardis, Marco
- Attar, Ricardo M
- Yang, Zheng
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Producer: 20081117
In:
Bioorganic & medicinal chemistry letters vol. 18
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In vivo patterns of resistance to the HIV attachment inhibitor BMS-488043. [electronic resource] by
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- Langley, David R
- Wang, Tao
- Kadow, John
- Grasela, Dennis
- Hanna, George J
- Alexander, Louis
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Producer: 20110519
In:
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29.
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Discovery and initial SAR of 3-(1H-benzo[d]imidazol-2-yl)pyridin-2(1H)-ones as inhibitors of insulin-like growth factor 1-receptor (IGF-1R). [electronic resource] by
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- Attar, Ricardo
- Gottardis, Marco
- Greer, Ann
- Chang, ChiehYing Y
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- Sun, Yax
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Producer: 20070530
In:
Bioorganic & medicinal chemistry letters vol. 17
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30.
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Heterocycle amide isosteres: An approach to overcoming resistance for HIV-1 integrase strand transfer inhibitors. [electronic resource] by
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- Lin, Zeyu
- Samanta, Himadri K
- Zheng, Ming
- Jenkins, Susan
- Dicker, Ira B
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Producer: 20210128
In:
Bioorganic & medicinal chemistry letters vol. 30
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31.
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Discovery of the Human Immunodeficiency Virus Type 1 (HIV-1) Attachment Inhibitor Temsavir and Its Phosphonooxymethyl Prodrug Fostemsavir. [electronic resource] by
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- Parker, Dawn D
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- Gong, Yi-Fei
- Ho, Hsu-Tso
- Colonno, Richard J
- Langley, David R
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Producer: 20190624
In:
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32.
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Characterizations of HCV NS5A replication complex inhibitors. [electronic resource] by
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- Belema, Makonen
- Nguyen, Van N
- Laurent, Denis R St
- Serrano-Wu, Michael
- Snyder, Lawrence B
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Producer: 20131106
In:
Virology vol. 444
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33.
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Biochemical and genetic characterizations of a novel human immunodeficiency virus type 1 inhibitor that blocks gp120-CD4 interactions. [electronic resource] by
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- Fan, Li
- Zhou, Nannan
- Friborg, Jacques
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- Wang, Hwei-Gene Heidi
- Rose, Ronald E
- Fang, Hua
- Scarnati, Helen T
- Langley, David R
- Meanwell, Nicholas A
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Producer: 20031014
In:
Journal of virology vol. 77
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34.
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Discovery of Isonicotinamides as Highly Selective, Brain Penetrable, and Orally Active Glycogen Synthase Kinase-3 Inhibitors. [electronic resource] by
- Luo, Guanglin
- Chen, Ling
- Burton, Catherine R
- Xiao, Hong
- Sivaprakasam, Prasanna
- Krause, Carol M
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- Liu, Nengyin
- Lippy, Jonathan
- Clarke, Wendy J
- Snow, Kimberly
- Raybon, Joseph
- Arora, Vinod
- Pokross, Matt
- Kish, Kevin
- Lewis, Hal A
- Langley, David R
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- Dubowchik, Gene M
Producer: 20160712
In:
Journal of medicinal chemistry vol. 59
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35.
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A General Amino Acid Synthesis Enabled by Innate Radical Cross-Coupling. [electronic resource] by
- Ni, Shengyang
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- Schmitt, Daniel C
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- Yang, Shouliang
- Collins, Michael R
- Qiao, Jennifer X
- Yeung, Kap-Sun
- Langley, David R
- Poss, Michael A
- Scola, Paul M
- Qin, Tian
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Producer: 20190911
In:
Angewandte Chemie (International ed. in English) vol. 57
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Discovery and Optimization of Novel Pyrazolopyrimidines as Potent and Orally Bioavailable Allosteric HIV-1 Integrase Inhibitors. [electronic resource] by
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- Langley, David R
- Naidu, B Narasimhulu
- Sivaprakasam, Prasanna
- Lewis, Hal
- Kish, Kevin
- Khan, Javed A
- Ng, Alicia
- Trainor, George L
- Cianci, Christopher
- Dicker, Ira B
- Walker, Michael A
- Lin, Zeyu
- Protack, Tricia
- Discotto, Linda
- Jenkins, Susan
- Gerritz, Samuel W
- Pendri, Annapurna
Producer: 20200831
In:
Journal of medicinal chemistry vol. 63
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37.
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Respiratory syncytial virus fusion inhibitors. Part 6: an examination of the effect of structural variation of the benzimidazol-2-one heterocycle moiety. [electronic resource] by
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- Gulgeze, H Belgin
- Thuring, Jan W
- Yu, Kuo-Long
- Civiello, Rita L
- Zhang, Yi
- Pearce, Bradley C
- Yin, Zhiwei
- Langley, David R
- Kadow, Kathleen F
- Cianci, Christopher W
- Li, Zhufang
- Clarke, Junius
- Genovesi, Eugene V
- Medina, Ivette
- Lamb, Lucinda
- Yang, Zheng
- Zadjura, Lisa
- Krystal, Mark
- Meanwell, Nicholas A
Producer: 20071120
In:
Bioorganic & medicinal chemistry letters vol. 17
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38.
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Lattice engineering enables definition of molecular features allowing for potent small-molecule inhibition of HIV-1 entry. [electronic resource] by
- Lai, Yen-Ting
- Wang, Tao
- O'Dell, Sijy
- Louder, Mark K
- Schön, Arne
- Cheung, Crystal S F
- Chuang, Gwo-Yu
- Druz, Aliaksandr
- Lin, Bob
- McKee, Krisha
- Peng, Dongjun
- Yang, Yongping
- Zhang, Baoshan
- Herschhorn, Alon
- Sodroski, Joseph
- Bailer, Robert T
- Doria-Rose, Nicole A
- Mascola, John R
- Langley, David R
- Kwong, Peter D
Producer: 20190219
In:
Nature communications vol. 10
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39.
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Chemical genetics strategy identifies an HCV NS5A inhibitor with a potent clinical effect. [electronic resource] by
- Gao, Min
- Nettles, Richard E
- Belema, Makonen
- Snyder, Lawrence B
- Nguyen, Van N
- Fridell, Robert A
- Serrano-Wu, Michael H
- Langley, David R
- Sun, Jin-Hua
- O'Boyle, Donald R
- Lemm, Julie A
- Wang, Chunfu
- Knipe, Jay O
- Chien, Caly
- Colonno, Richard J
- Grasela, Dennis M
- Meanwell, Nicholas A
- Hamann, Lawrence G
Producer: 20100512
In:
Nature vol. 465
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40.
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Discovery of new acylaminopyridines as GSK-3 inhibitors by a structure guided in-depth exploration of chemical space around a pyrrolopyridinone core. [electronic resource] by
- Sivaprakasam, Prasanna
- Han, Xiaojun
- Civiello, Rita L
- Jacutin-Porte, Swanee
- Kish, Kevin
- Pokross, Matt
- Lewis, Hal A
- Ahmed, Nazia
- Szapiel, Nicolas
- Newitt, John A
- Baldwin, Eric T
- Xiao, Hong
- Krause, Carol M
- Park, Hyunsoo
- Nophsker, Michelle
- Lippy, Jonathan S
- Burton, Catherine R
- Langley, David R
- Macor, John E
- Dubowchik, Gene M
Producer: 20160219
In:
Bioorganic & medicinal chemistry letters vol. 25
Availability: No items available.
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