Results
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Synthesis and characterization of pyrrolidine derivatives as potent agonists of the human melanocortin-4 receptor. [electronic resource] by
- Jiang, Wanlong
- Tran, Joe A
- Tucci, Fabio C
- Fleck, Beth A
- Hoare, Sam R
- Markison, Stacy
- Wen, Jenny
- Chen, Caroline W
- Marinkovic, Dragan
- Arellano, Melissa
- Foster, Alan C
- Chen, Chen
Producer: 20080303
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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23.
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Pyrrolidinones as potent functional antagonists of the human melanocortin-4 receptor. [electronic resource] by
- Jiang, Wanlong
- Tucci, Fabio C
- Tran, Joe A
- Fleck, Beth A
- Wen, Jenny
- Markison, Stacy
- Marinkovic, Dragan
- Chen, Caroline W
- Arellano, Melissa
- Hoare, Sam R
- Johns, Michael
- Foster, Alan C
- Saunders, John
- Chen, Chen
Producer: 20071212
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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24.
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A potent and selective nonpeptide antagonist of the melanocortin-4 receptor induces food intake in satiated mice. [electronic resource] by
- Pontillo, Joseph
- Tran, Joseph A
- Markison, Stacy
- Joppa, Margaret
- Fleck, Beth A
- Marinkovic, Dragan
- Arellano, Melissa
- Tucci, Fabio C
- Lanier, Marion
- Nelson, Jodie
- Saunders, John
- Hoare, Sam R J
- Foster, Alan C
- Chen, Chen
Producer: 20051011
In:
Bioorganic & medicinal chemistry letters vol. 15
Availability: No items available.
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25.
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Identification and characterization of pyrrolidine diastereoisomers as potent functional agonists and antagonists of the human melanocortin-4 receptor. [electronic resource] by
- Chen, Chen
- Jiang, Wanlong
- Tran, Joe A
- Tucci, Fabio C
- Fleck, Beth A
- Markison, Stacy
- Wen, Jenny
- Madan, Ajay
- Hoare, Sam R
- Foster, Alan C
- Marinkovic, Dragan
- Chen, Caroline W
- Arellano, Melissa
- Saunders, John
Producer: 20080212
In:
Bioorganic & medicinal chemistry letters vol. 18
Availability: No items available.
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26.
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Discovery of NBI-77860/GSK561679, a potent corticotropin-releasing factor (CRF1) receptor antagonist with improved pharmacokinetic properties. [electronic resource] by
- Tellew, John E
- Lanier, Marion
- Moorjani, Manisha
- Lin, Emily
- Luo, Zhiyong
- Slee, Deborah H
- Zhang, Xiaohu
- Hoare, Sam R J
- Grigoriadis, Dimitri E
- St Denis, Yves
- Di Fabio, Romano
- Di Modugno, Enza
- Saunders, John
- Williams, John P
Producer: 20110314
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
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27.
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Discovery of 1-[2-[(1S)-(3-dimethylaminopropionyl)amino-2-methylpropyl]-4-methylphenyl]-4-[(2R)-methyl-3-(4-chlorophenyl)-propionyl]piperazine as an orally active antagonist of the melanocortin-4 receptor for the potential treatment of cachexia. [electronic resource] by
- Chen, Chen
- Jiang, Wanlong
- Tucci, Fabio
- Tran, Joe A
- Fleck, Beth A
- Hoare, Sam R
- Joppa, Margaret
- Markison, Stacy
- Wen, Jenny
- Sai, Yang
- Johns, Michael
- Madan, Ajay
- Chen, Takung
- Chen, Caroline W
- Marinkovic, Dragan
- Arellano, Melissa
- Saunders, John
- Foster, Alan C
Producer: 20071206
In:
Journal of medicinal chemistry vol. 50
Availability: No items available.
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28.
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Pyrrolidinones as orally bioavailable antagonists of the human melanocortin-4 receptor with anti-cachectic activity. [electronic resource] by
- Tran, Joe A
- Tucci, Fabio C
- Jiang, Wanlong
- Marinkovic, Dragan
- Chen, Caroline W
- Arellano, Melissa
- Markison, Stacy
- Fleck, Beth A
- Wen, Jenny
- White, Nicole S
- Pontillo, Joseph
- Saunders, John
- Marks, Daniel
- Hoare, Sam R
- Madan, Ajay
- Foster, Alan C
- Chen, Chen
Producer: 20070906
In:
Bioorganic & medicinal chemistry vol. 15
Availability: No items available.
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29.
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Pharmacological and pharmacokinetic characterization of 2-piperazine-alpha-isopropyl benzylamine derivatives as melanocortin-4 receptor antagonists. [electronic resource] by
- Chen, Chen
- Tucci, Fabio C
- Jiang, Wanlong
- Tran, Joe A
- Fleck, Beth A
- Hoare, Sam R
- Wen, Jenny
- Chen, Takung
- Johns, Michael
- Markison, Stacy
- Foster, Alan C
- Marinkovic, Dragan
- Chen, Caroline W
- Arellano, Melissa
- Harman, John
- Saunders, John
- Bozigian, Haig
- Marks, Daniel
Producer: 20080818
In:
Bioorganic & medicinal chemistry vol. 16
Availability: No items available.
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30.
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Design, synthesis, in vitro, and in vivo characterization of phenylpiperazines and pyridinylpiperazines as potent and selective antagonists of the melanocortin-4 receptor. [electronic resource] by
- Tran, Joe A
- Jiang, Wanlong
- Tucci, Fabio C
- Fleck, Beth A
- Wen, Jenny
- Sai, Yang
- Madan, Ajay
- Chen, Ta Kung
- Markison, Stacy
- Foster, Alan C
- Hoare, Sam R
- Marks, Daniel
- Harman, John
- Chen, Caroline W
- Arellano, Melissa
- Marinkovic, Dragan
- Bozigian, Haig
- Saunders, John
- Chen, Chen
Producer: 20080310
In:
Journal of medicinal chemistry vol. 50
Availability: No items available.
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31.
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Design and synthesis of tricyclic corticotropin-releasing factor-1 antagonists. [electronic resource] by
- Gross, Raymond S
- Guo, Zhiqiang
- Dyck, Brian
- Coon, Tim
- Huang, Charles Q
- Lowe, Richard F
- Marinkovic, Dragan
- Moorjani, Manisha
- Nelson, Jodene
- Zamani-Kord, Said
- Grigoriadis, Dimitri E
- Hoare, Sam R J
- Crowe, Paul D
- Bu, Jane Han
- Haddach, Mustapha
- McCarthy, James
- Saunders, John
- Sullivan, Robert
- Chen, Takung
- Williams, John P
Producer: 20051101
In:
Journal of medicinal chemistry vol. 48
Availability: No items available.
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