Results
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21.
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Identification of Imidazo[1,2- [electronic resource] by
- Liu, Chunjian
- Lin, James
- Moslin, Ryan
- Tokarski, John S
- Muckelbauer, Jodi
- Chang, ChiehYing
- Tredup, Jeffrey
- Xie, Dianlin
- Park, Hyunsoo
- Li, Peng
- Wu, Dauh-Rurng
- Strnad, Joann
- Zupa-Fernandez, Adriana
- Cheng, Lihong
- Chaudhry, Charu
- Chen, Jing
- Chen, Cliff
- Sun, Huadong
- Elzinga, Paul
- D'arienzo, Celia
- Gillooly, Kathleen
- Taylor, Tracy L
- McIntyre, Kim W
- Salter-Cid, Luisa
- Lombardo, Louis J
- Carter, Percy H
- Aranibar, Nelly
- Burke, James R
- Weinstein, David S
Publication details: ACS medicinal chemistry letters Mar 2019
In:
ACS medicinal chemistry letters vol. 10
Availability: No items available.
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22.
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Small molecule antagonist of leukocyte function associated antigen-1 (LFA-1): structure-activity relationships leading to the identification of 6-((5S,9R)-9-(4-cyanophenyl)-3-(3,5-dichlorophenyl)-1-methyl-2,4-dioxo-1,3,7-triazaspiro[4.4]nonan-7-yl)nicotinic acid (BMS-688521). [electronic resource] by
- Watterson, Scott H
- Xiao, Zili
- Dodd, Dharmpal S
- Tortolani, David R
- Vaccaro, Wayne
- Potin, Dominique
- Launay, Michele
- Stetsko, Dawn K
- Skala, Stacey
- Davis, Patric M
- Lee, Deborah
- Yang, Xiaoxia
- McIntyre, Kim W
- Balimane, Praveen
- Patel, Karishma
- Yang, Zheng
- Marathe, Punit
- Kadiyala, Pathanjali
- Tebben, Andrew J
- Sheriff, Steven
- Chang, Chiehying Y
- Ziemba, Theresa
- Zhang, Huiping
- Chen, Bang-Chi
- DelMonte, Albert J
- Aranibar, Nelly
- McKinnon, Murray
- Barrish, Joel C
- Suchard, Suzanne J
- Murali Dhar, T G
Producer: 20100611
In:
Journal of medicinal chemistry vol. 53
Availability: No items available.
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23.
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Discovery of a 2,4-disubstituted pyrrolo[1,2-f][1,2,4]triazine inhibitor (BMS-754807) of insulin-like growth factor receptor (IGF-1R) kinase in clinical development. [electronic resource] by
- Wittman, Mark D
- Carboni, Joan M
- Yang, Zheng
- Lee, Francis Y
- Antman, Melissa
- Attar, Ricardo
- Balimane, Praveen
- Chang, Chiehying
- Chen, Cliff
- Discenza, Lorell
- Frennesson, David
- Gottardis, Marco M
- Greer, Ann
- Hurlburt, Warren
- Johnson, Walter
- Langley, David R
- Li, Aixin
- Li, Jianqing
- Liu, Peiying
- Mastalerz, Harold
- Mathur, Arvind
- Menard, Krista
- Patel, Karishma
- Sack, John
- Sang, Xiaopeng
- Saulnier, Mark
- Smith, Daniel
- Stefanski, Kevin
- Trainor, George
- Velaparthi, Upender
- Zhang, Guifen
- Zimmermann, Kurt
- Vyas, Dolatrai M
Producer: 20091231
In:
Journal of medicinal chemistry vol. 52
Availability: No items available.
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24.
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Small Molecule Reversible Inhibitors of Bruton's Tyrosine Kinase (BTK): Structure-Activity Relationships Leading to the Identification of 7-(2-Hydroxypropan-2-yl)-4-[2-methyl-3-(4-oxo-3,4-dihydroquinazolin-3-yl)phenyl]-9H-carbazole-1-carboxamide (BMS-935177). [electronic resource] by
- De Lucca, George V
- Shi, Qing
- Liu, Qingjie
- Batt, Douglas G
- Beaudoin Bertrand, Myra
- Rampulla, Rick
- Mathur, Arvind
- Discenza, Lorell
- D'Arienzo, Celia
- Dai, Jun
- Obermeier, Mary
- Vickery, Rodney
- Zhang, Yingru
- Yang, Zheng
- Marathe, Punit
- Tebben, Andrew J
- Muckelbauer, Jodi K
- Chang, ChiehYing J
- Zhang, Huiping
- Gillooly, Kathleen
- Taylor, Tracy
- Pattoli, Mark A
- Skala, Stacey
- Kukral, Daniel W
- McIntyre, Kim W
- Salter-Cid, Luisa
- Fura, Aberra
- Burke, James R
- Barrish, Joel C
- Carter, Percy H
- Tino, Joseph A
Producer: 20170710
In:
Journal of medicinal chemistry vol. 59
Availability: No items available.
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25.
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Discovery and Preclinical Evaluation of BMS-711939, an Oxybenzylglycine Based PPARα Selective Agonist. [electronic resource] by
- Shi, Yan
- Li, Jun
- Kennedy, Lawrence J
- Tao, Shiwei
- Hernández, Andrés S
- Lai, Zhi
- Chen, Sean
- Wong, Henry
- Zhu, Juliang
- Trehan, Ashok
- Lim, Ngiap-Kie
- Zhang, Huiping
- Chen, Bang-Chi
- Locke, Kenneth T
- O'Malley, Kevin M
- Zhang, Litao
- Srivastava, Rai Ajit
- Miao, Bowman
- Meyers, Daniel S
- Monshizadegan, Hossain
- Search, Debra
- Grimm, Denise
- Zhang, Rongan
- Harrity, Thomas
- Kunselman, Lori K
- Cap, Michael
- Muckelbauer, Jodi
- Chang, Chiehying
- Krystek, Stanley R
- Li, Yi-Xin
- Hosagrahara, Vinayak
- Zhang, Lisa
- Kadiyala, Pathanjali
- Xu, Carrie
- Blanar, Michael A
- Zahler, Robert
- Mukherjee, Ranjan
- Cheng, Peter T W
- Tino, Joseph A
Producer: 20160621
In:
ACS medicinal chemistry letters vol. 7
Availability: No items available.
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26.
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Discovery of 6-Fluoro-5-(R)-(3-(S)-(8-fluoro-1-methyl-2,4-dioxo-1,2-dihydroquinazolin-3(4H)-yl)-2-methylphenyl)-2-(S)-(2-hydroxypropan-2-yl)-2,3,4,9-tetrahydro-1H-carbazole-8-carboxamide (BMS-986142): A Reversible Inhibitor of Bruton's Tyrosine Kinase (BTK) Conformationally Constrained by Two Locked Atropisomers. [electronic resource] by
- Watterson, Scott H
- De Lucca, George V
- Shi, Qing
- Langevine, Charles M
- Liu, Qingjie
- Batt, Douglas G
- Beaudoin Bertrand, Myra
- Gong, Hua
- Dai, Jun
- Yip, Shiuhang
- Li, Peng
- Sun, Dawn
- Wu, Dauh-Rurng
- Wang, Chunlei
- Zhang, Yingru
- Traeger, Sarah C
- Pattoli, Mark A
- Skala, Stacey
- Cheng, Lihong
- Obermeier, Mary T
- Vickery, Rodney
- Discenza, Lorell N
- D'Arienzo, Celia J
- Zhang, Yifan
- Heimrich, Elizabeth
- Gillooly, Kathleen M
- Taylor, Tracy L
- Pulicicchio, Claudine
- McIntyre, Kim W
- Galella, Michael A
- Tebben, Andy J
- Muckelbauer, Jodi K
- Chang, ChiehYing
- Rampulla, Richard
- Mathur, Arvind
- Salter-Cid, Luisa
- Barrish, Joel C
- Carter, Percy H
- Fura, Aberra
- Burke, James R
- Tino, Joseph A
Producer: 20170619
In:
Journal of medicinal chemistry vol. 59
Availability: No items available.
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27.
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Discovery of an oxybenzylglycine based peroxisome proliferator activated receptor alpha selective agonist 2-((3-((2-(4-chlorophenyl)-5-methyloxazol-4-yl)methoxy)benzyl)(methoxycarbonyl)amino)acetic acid (BMS-687453). [electronic resource] by
- Li, Jun
- Kennedy, Lawrence J
- Shi, Yan
- Tao, Shiwei
- Ye, Xiang-Yang
- Chen, Stephanie Y
- Wang, Ying
- Hernández, Andrés S
- Wang, Wei
- Devasthale, Pratik V
- Chen, Sean
- Lai, Zhi
- Zhang, Hao
- Wu, Shung
- Smirk, Rebecca A
- Bolton, Scott A
- Ryono, Denis E
- Zhang, Huiping
- Lim, Ngiap-Kie
- Chen, Bang-Chi
- Locke, Kenneth T
- O'Malley, Kevin M
- Zhang, Litao
- Srivastava, Rai Ajit
- Miao, Bowman
- Meyers, Daniel S
- Monshizadegan, Hossain
- Search, Debra
- Grimm, Denise
- Zhang, Rongan
- Harrity, Thomas
- Kunselman, Lori K
- Cap, Michael
- Kadiyala, Pathanjali
- Hosagrahara, Vinayak
- Zhang, Lisa
- Xu, Carrie
- Li, Yi-Xin
- Muckelbauer, Jodi K
- Chang, Chiehying
- An, Yongmi
- Krystek, Stanley R
- Blanar, Michael A
- Zahler, Robert
- Mukherjee, Ranjan
- Cheng, Peter T W
- Tino, Joseph A
Producer: 20100510
In:
Journal of medicinal chemistry vol. 53
Availability: No items available.
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