Results
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21.
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Correction to Noncovalent Mutant Selective Epidermal Growth Factor Receptor Inhibitors: A Lead Optimization Case Study. [electronic resource] by
- Heald, Robert
- Bowman, Krista K
- Bryan, Marian C
- Burdick, Daniel
- Chan, Bryan
- Chan, Emily
- Chen, Yuan
- Clausen, Saundra
- Dominguez-Fernandez, Belen
- Eigenbrot, Charles
- Elliott, Richard
- Hanan, Emily J
- Jackson, Philip
- Knight, Jamie
- La, Hank
- Lainchbury, Michael
- Malek, Shiva
- Mann, Sam
- Merchant, Mark
- Mortara, Kyle
- Purkey, Hans
- Schaefer, Gabriele
- Schmidt, Stephen
- Seward, Eileen
- Sideris, Steve
- Shao, Lily
- Wang, Shumei
- Yeap, Kuen
- Yen, Ivana
- Yu, Christine
- Heffron, Timothy P
Producer: 20160809
In:
Journal of medicinal chemistry vol. 59
Availability: No items available.
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22.
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Noncovalent Mutant Selective Epidermal Growth Factor Receptor Inhibitors: A Lead Optimization Case Study. [electronic resource] by
- Heald, Robert
- Bowman, Krista K
- Bryan, Marian C
- Burdick, Daniel
- Chan, Bryan
- Chan, Emily
- Chen, Yuan
- Clausen, Saundra
- Dominguez-Fernandez, Belen
- Eigenbrot, Charles
- Elliott, Richard
- Hanan, Emily J
- Jackson, Philip
- Knight, Jamie
- La, Hank
- Lainchbury, Michael
- Malek, Shiva
- Mann, Sam
- Merchant, Mark
- Mortara, Kyle
- Purkey, Hans
- Schaefer, Gabriele
- Schmidt, Stephen
- Seward, Eileen
- Sideris, Steve
- Shao, Lily
- Wang, Shumei
- Yeap, Kuen
- Yen, Ivana
- Yu, Christine
- Heffron, Timothy P
Producer: 20160314
In:
Journal of medicinal chemistry vol. 58
Availability: No items available.
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23.
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Ser1292 autophosphorylation is an indicator of LRRK2 kinase activity and contributes to the cellular effects of PD mutations. [electronic resource] by
- Sheng, Zejuan
- Zhang, Shuo
- Bustos, Daisy
- Kleinheinz, Tracy
- Le Pichon, Claire E
- Dominguez, Sara L
- Solanoy, Hilda O
- Drummond, Jason
- Zhang, Xiaolin
- Ding, Xiao
- Cai, Fang
- Song, Qinghua
- Li, Xianting
- Yue, Zhenyu
- van der Brug, Marcel P
- Burdick, Daniel J
- Gunzner-Toste, Janet
- Chen, Huifen
- Liu, Xingrong
- Estrada, Anthony A
- Sweeney, Zachary K
- Scearce-Levie, Kimberly
- Moffat, John G
- Kirkpatrick, Donald S
- Zhu, Haitao
Producer: 20130916
In:
Science translational medicine vol. 4
Availability: No items available.
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24.
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Discovery of a Noncovalent, Mutant-Selective Epidermal Growth Factor Receptor Inhibitor. [electronic resource] by
- Chan, Bryan K
- Hanan, Emily J
- Bowman, Krista K
- Bryan, Marian C
- Burdick, Daniel
- Chan, Emily
- Chen, Yuan
- Clausen, Saundra
- Dela Vega, Trisha
- Dotson, Jennafer
- Eigenbrot, Charles
- Elliott, Richard L
- Heald, Robert A
- Jackson, Philip S
- Knight, Jamie D
- La, Hank
- Lainchbury, Michael D
- Malek, Shiva
- Purkey, Hans E
- Schaefer, Gabriele
- Schmidt, Stephen
- Seward, Eileen M
- Sideris, Steve
- Shao, Lily
- Wang, Shumei
- Yeap, Siew Kuen
- Yen, Ivana
- Yu, Christine
- Heffron, Timothy P
Producer: 20170619
In:
Journal of medicinal chemistry vol. 59
Availability: No items available.
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25.
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GNE-371, a Potent and Selective Chemical Probe for the Second Bromodomains of Human Transcription-Initiation-Factor TFIID Subunit 1 and Transcription-Initiation-Factor TFIID Subunit 1-like. [electronic resource] by
- Wang, Shumei
- Tsui, Vickie
- Crawford, Terry D
- Audia, James E
- Burdick, Daniel J
- Beresini, Maureen H
- Côté, Alexandre
- Cummings, Richard
- Duplessis, Martin
- Flynn, E Megan
- Hewitt, Michael C
- Huang, Hon-Ren
- Jayaram, Hariharan
- Jiang, Ying
- Joshi, Shivangi
- Murray, Jeremy
- Nasveschuk, Christopher G
- Pardo, Eneida
- Poy, Florence
- Romero, F Anthony
- Tang, Yong
- Taylor, Alexander M
- Wang, Jian
- Xu, Zhaowu
- Zawadzke, Laura E
- Zhu, Xiaoyu
- Albrecht, Brian K
- Magnuson, Steven R
- Bellon, Steve
- Cochran, Andrea G
Producer: 20190930
In:
Journal of medicinal chemistry vol. 61
Availability: No items available.
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26.
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Diving into the Water: Inducible Binding Conformations for BRD4, TAF1(2), BRD9, and CECR2 Bromodomains. [electronic resource] by
- Crawford, Terry D
- Tsui, Vickie
- Flynn, E Megan
- Wang, Shumei
- Taylor, Alexander M
- Côté, Alexandre
- Audia, James E
- Beresini, Maureen H
- Burdick, Daniel J
- Cummings, Richard
- Dakin, Les A
- Duplessis, Martin
- Good, Andrew C
- Hewitt, Michael C
- Huang, Hon-Ren
- Jayaram, Hariharan
- Kiefer, James R
- Jiang, Ying
- Murray, Jeremy
- Nasveschuk, Christopher G
- Pardo, Eneida
- Poy, Florence
- Romero, F Anthony
- Tang, Yong
- Wang, Jian
- Xu, Zhaowu
- Zawadzke, Laura E
- Zhu, Xiaoyu
- Albrecht, Brian K
- Magnuson, Steven R
- Bellon, Steve
- Cochran, Andrea G
Producer: 20170606
In:
Journal of medicinal chemistry vol. 59
Availability: No items available.
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27.
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Discovery of highly potent, selective, and brain-penetrant aminopyrazole leucine-rich repeat kinase 2 (LRRK2) small molecule inhibitors. [electronic resource] by
- Estrada, Anthony A
- Chan, Bryan K
- Baker-Glenn, Charles
- Beresford, Alan
- Burdick, Daniel J
- Chambers, Mark
- Chen, Huifen
- Dominguez, Sara L
- Dotson, Jennafer
- Drummond, Jason
- Flagella, Michael
- Fuji, Reina
- Gill, Andrew
- Halladay, Jason
- Harris, Seth F
- Heffron, Timothy P
- Kleinheinz, Tracy
- Lee, Donna W
- Le Pichon, Claire E
- Liu, Xingrong
- Lyssikatos, Joseph P
- Medhurst, Andrew D
- Moffat, John G
- Nash, Kevin
- Scearce-Levie, Kimberly
- Sheng, Zejuan
- Shore, Daniel G
- Wong, Susan
- Zhang, Shuo
- Zhang, Xiaolin
- Zhu, Haitao
- Sweeney, Zachary K
Producer: 20140415
In:
Journal of medicinal chemistry vol. 57
Availability: No items available.
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28.
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GNE-886: A Potent and Selective Inhibitor of the Cat Eye Syndrome Chromosome Region Candidate 2 Bromodomain (CECR2). [electronic resource] by
- Crawford, Terry D
- Audia, James E
- Bellon, Steve
- Burdick, Daniel J
- Bommi-Reddy, Archana
- Côté, Alexandre
- Cummings, Richard T
- Duplessis, Martin
- Flynn, E Megan
- Hewitt, Michael
- Huang, Hon-Ren
- Jayaram, Hariharan
- Jiang, Ying
- Joshi, Shivangi
- Kiefer, James R
- Murray, Jeremy
- Nasveschuk, Christopher G
- Neiss, Arianne
- Pardo, Eneida
- Romero, F Anthony
- Sandy, Peter
- Sims, Robert J
- Tang, Yong
- Taylor, Alexander M
- Tsui, Vickie
- Wang, Jian
- Wang, Shumei
- Wang, Yongyun
- Xu, Zhaowu
- Zawadzke, Laura
- Zhu, Xiaoqin
- Albrecht, Brian K
- Magnuson, Steven R
- Cochran, Andrea G
Publication details: ACS medicinal chemistry letters Jul 2017
In:
ACS medicinal chemistry letters vol. 8
Availability: No items available.
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29.
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Discovery of highly potent, selective, and brain-penetrable leucine-rich repeat kinase 2 (LRRK2) small molecule inhibitors. [electronic resource] by
- Estrada, Anthony A
- Liu, Xingrong
- Baker-Glenn, Charles
- Beresford, Alan
- Burdick, Daniel J
- Chambers, Mark
- Chan, Bryan K
- Chen, Huifen
- Ding, Xiao
- DiPasquale, Antonio G
- Dominguez, Sara L
- Dotson, Jennafer
- Drummond, Jason
- Flagella, Michael
- Flynn, Sean
- Fuji, Reina
- Gill, Andrew
- Gunzner-Toste, Janet
- Harris, Seth F
- Heffron, Timothy P
- Kleinheinz, Tracy
- Lee, Donna W
- Le Pichon, Claire E
- Lyssikatos, Joseph P
- Medhurst, Andrew D
- Moffat, John G
- Mukund, Susmith
- Nash, Kevin
- Scearce-Levie, Kimberly
- Sheng, Zejuan
- Shore, Daniel G
- Tran, Thuy
- Trivedi, Naimisha
- Wang, Shumei
- Zhang, Shuo
- Zhang, Xiaolin
- Zhao, Guiling
- Zhu, Haitao
- Sweeney, Zachary K
Producer: 20130205
In:
Journal of medicinal chemistry vol. 55
Availability: No items available.
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