Results
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21.
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SGC-GAK-1: A Chemical Probe for Cyclin G Associated Kinase (GAK). [electronic resource] by
- Asquith, Christopher R M
- Berger, Benedict-Tilman
- Wan, Jing
- Bennett, James M
- Capuzzi, Stephen J
- Crona, Daniel J
- Drewry, David H
- East, Michael P
- Elkins, Jonathan M
- Fedorov, Oleg
- Godoi, Paulo H
- Hunter, Debra M
- Knapp, Stefan
- Müller, Susanne
- Torrice, Chad D
- Wells, Carrow I
- Earp, H Shelton
- Willson, Timothy M
- Zuercher, William J
Producer: 20200406
In:
Journal of medicinal chemistry vol. 62
Availability: No items available.
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22.
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Discovery and in vivo evaluation of alcohol-containing benzothiazoles as potent dual-targeting bacterial DNA supercoiling inhibitors. [electronic resource] by
- Palmer, James T
- Axford, Lorraine C
- Barker, Stephanie
- Bennett, James M
- Blair, Michael
- Collins, Ian
- Davies, David T
- Ford, Leigh
- Gannon, Carlie T
- Lancett, Paul
- Logan, Alastair
- Lunniss, Christopher J
- Morton, Craig J
- Offermann, Daniel A
- Pitt, Gary R W
- Rao, B Narasinga
- Singh, Amit K
- Shukla, Tarun
- Srivastava, Anil
- Stokes, Neil R
- Thomaides-Brears, Helena B
- Yadav, Anju
- Haydon, David J
Producer: 20150330
In:
Bioorganic & medicinal chemistry letters vol. 24
Availability: No items available.
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23.
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C8-substituted pyrido[3,4-d]pyrimidin-4(3H)-ones: Studies towards the identification of potent, cell penetrant Jumonji C domain containing histone lysine demethylase 4 subfamily (KDM4) inhibitors, compound profiling in cell-based target engagement assays. [electronic resource] by
- Le Bihan, Yann-Vaï
- Lanigan, Rachel M
- Atrash, Butrus
- McLaughlin, Mark G
- Velupillai, Srikannathasan
- Malcolm, Andrew G
- England, Katherine S
- Ruda, Gian Filippo
- Mok, N Yi
- Tumber, Anthony
- Tomlin, Kathy
- Saville, Harry
- Shehu, Erald
- McAndrew, Craig
- Carmichael, LeAnne
- Bennett, James M
- Jeganathan, Fiona
- Eve, Paul
- Donovan, Adam
- Hayes, Angela
- Wood, Francesca
- Raynaud, Florence I
- Fedorov, Oleg
- Brennan, Paul E
- Burke, Rosemary
- van Montfort, Rob L M
- Rossanese, Olivia W
- Blagg, Julian
- Bavetsias, Vassilios
Producer: 20190725
In:
European journal of medicinal chemistry vol. 177
Availability: No items available.
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24.
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Isoform-Selective ATAD2 Chemical Probe with Novel Chemical Structure and Unusual Mode of Action. [electronic resource] by
- Fernández-Montalván, Amaury E
- Berger, Markus
- Kuropka, Benno
- Koo, Seong Joo
- Badock, Volker
- Weiske, Joerg
- Puetter, Vera
- Holton, Simon J
- Stöckigt, Detlef
- Ter Laak, Antonius
- Centrella, Paolo A
- Clark, Matthew A
- Dumelin, Christoph E
- Sigel, Eric A
- Soutter, Holly H
- Troast, Dawn M
- Zhang, Ying
- Cuozzo, John W
- Keefe, Anthony D
- Roche, Didier
- Rodeschini, Vincent
- Chaikuad, Apirat
- Díaz-Sáez, Laura
- Bennett, James M
- Fedorov, Oleg
- Huber, Kilian V M
- Hübner, Jan
- Weinmann, Hilmar
- Hartung, Ingo V
- Gorjánácz, Mátyás
Producer: 20171219
In:
ACS chemical biology vol. 12
Availability: No items available.
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25.
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WNT Activates the AAK1 Kinase to Promote Clathrin-Mediated Endocytosis of LRP6 and Establish a Negative Feedback Loop. [electronic resource] by
- Agajanian, Megan J
- Walker, Matthew P
- Axtman, Alison D
- Ruela-de-Sousa, Roberta R
- Serafin, D Stephen
- Rabinowitz, Alex D
- Graham, David M
- Ryan, Meagan B
- Tamir, Tigist
- Nakamichi, Yuko
- Gammons, Melissa V
- Bennett, James M
- Couñago, Rafael M
- Drewry, David H
- Elkins, Jonathan M
- Gileadi, Carina
- Gileadi, Opher
- Godoi, Paulo H
- Kapadia, Nirav
- Müller, Susanne
- Santiago, André S
- Sorrell, Fiona J
- Wells, Carrow I
- Fedorov, Oleg
- Willson, Timothy M
- Zuercher, William J
- Major, Michael B
Producer: 20200319
In:
Cell reports vol. 26
Availability: No items available.
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26.
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Design, synthesis and biological evaluation of α-substituted isonipecotic acid benzothiazole analogues as potent bacterial type II topoisomerase inhibitors. [electronic resource] by
- Axford, Lorraine C
- Agarwal, Piyush K
- Anderson, Kelly H
- Andrau, Laura N
- Atherall, John
- Barker, Stephanie
- Bennett, James M
- Blair, Michael
- Collins, Ian
- Czaplewski, Lloyd G
- Davies, David T
- Gannon, Carlie T
- Kumar, Dushyant
- Lancett, Paul
- Logan, Alastair
- Lunniss, Christopher J
- Mitchell, Dale R
- Offermann, Daniel A
- Palmer, James T
- Palmer, Nicholas
- Pitt, Gary R W
- Pommier, Stéphanie
- Price, Daniel
- Narasinga Rao, B
- Saxena, Rashmi
- Shukla, Tarun
- Singh, Amit K
- Singh, Mahipal
- Srivastava, Anil
- Steele, Christopher
- Stokes, Neil R
- Thomaides-Brears, Helena B
- Tyndall, Edward M
- Watson, David
- Haydon, David J
Producer: 20140725
In:
Bioorganic & medicinal chemistry letters vol. 23
Availability: No items available.
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27.
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8-Substituted Pyrido[3,4-d]pyrimidin-4(3H)-one Derivatives As Potent, Cell Permeable, KDM4 (JMJD2) and KDM5 (JARID1) Histone Lysine Demethylase Inhibitors. [electronic resource] by
- Bavetsias, Vassilios
- Lanigan, Rachel M
- Ruda, Gian Filippo
- Atrash, Butrus
- McLaughlin, Mark G
- Tumber, Anthony
- Mok, N Yi
- Le Bihan, Yann-Vaï
- Dempster, Sally
- Boxall, Katherine J
- Jeganathan, Fiona
- Hatch, Stephanie B
- Savitsky, Pavel
- Velupillai, Srikannathasan
- Krojer, Tobias
- England, Katherine S
- Sejberg, Jimmy
- Thai, Ching
- Donovan, Adam
- Pal, Akos
- Scozzafava, Giuseppe
- Bennett, James M
- Kawamura, Akane
- Johansson, Catrine
- Szykowska, Aleksandra
- Gileadi, Carina
- Burgess-Brown, Nicola A
- von Delft, Frank
- Oppermann, Udo
- Walters, Zoe
- Shipley, Janet
- Raynaud, Florence I
- Westaway, Susan M
- Prinjha, Rab K
- Fedorov, Oleg
- Burke, Rosemary
- Schofield, Christopher J
- Westwood, Isaac M
- Bountra, Chas
- Müller, Susanne
- van Montfort, Rob L M
- Brennan, Paul E
- Blagg, Julian
Producer: 20160726
In:
Journal of medicinal chemistry vol. 59
Availability: No items available.
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