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Structure based design of macrocyclic factor XIa inhibitors: Discovery of cyclic P1 linker moieties with improved oral bioavailability. [electronic resource] by
- Clark, Charles G
- Rossi, Karen A
- Corte, James R
- Fang, Tianan
- Smallheer, Joanne M
- De Lucca, Indawati
- Nirschl, David S
- Orwat, Michael J
- Pinto, Donald J P
- Hu, Zilun
- Wang, Yufeng
- Yang, Wu
- Jeon, Yoon
- Ewing, William R
- Myers, Joseph E
- Sheriff, Steven
- Lou, Zhen
- Bozarth, Jeffrey M
- Wu, Yiming
- Rendina, Alan
- Harper, Timothy
- Zheng, Joanna
- Xin, Baomin
- Xiang, Qian
- Luettgen, Joseph M
- Seiffert, Dietmar A
- Wexler, Ruth R
- Lam, Patrick Y S
Producer: 20200921
In:
Bioorganic & medicinal chemistry letters vol. 29
Availability: No items available.
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Pyridazine and pyridazinone derivatives as potent and selective factor XIa inhibitors. [electronic resource] by
- Hu, Zilun
- Wang, Cailan
- Han, Wei
- Rossi, Karen A
- Bozarth, Jeffrey M
- Wu, Yiming
- Sheriff, Steven
- Myers, Joseph E
- Luettgen, Joseph M
- Seiffert, Dietmar A
- Wexler, Ruth R
- Quan, Mimi L
Producer: 20180924
In:
Bioorganic & medicinal chemistry letters vol. 28
Availability: No items available.
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Synthesis, Docking, and In Vitro Anticoagulant Activity Assay of Hybrid Derivatives of Pyrrolo[3,2,1- [electronic resource] by
- Novichikhina, Nadezhda
- Ilin, Ivan
- Tashchilova, Anna
- Sulimov, Alexey
- Kutov, Danil
- Ledenyova, Irina
- Krysin, Mikhail
- Shikhaliev, Khidmet
- Gantseva, Anna
- Gantseva, Ekaterina
- Podoplelova, Nadezhda
- Sulimov, Vladimir
Producer: 20210202
In:
Molecules (Basel, Switzerland) vol. 25
Availability: No items available.
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