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Identification of an orally active opioid receptor-like 1 (ORL1) receptor antagonist 4-{3-[(2R)-2,3-dihydroxypropyl]-2-oxo-2,3-dihydro-1H-benzimidazol-1-yl}-1-[(1S,3S,4R)-spiro[bicyclo[2.2.1]heptane-2,1'-cyclopropan]-3-ylmethyl]piperidine as clinical candidate. [electronic resource] by
- Satoh, Atsushi
- Sagara, Takeshi
- Sakoh, Hiroki
- Hashimoto, Masaya
- Nakashima, Hiroshi
- Kato, Tetsuya
- Goto, Yasuhiro
- Mizutani, Sayaka
- Azuma-Kanoh, Tomoko
- Tani, Takeshi
- Okuda, Shoki
- Okamoto, Osamu
- Ozaki, Satoshi
- Iwasawa, Yoshikazu
- Ohta, Hisashi
- Kawamoto, Hiroshi
Producer: 20090825
In:
Journal of medicinal chemistry vol. 52
Availability: No items available.
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