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Discovery of (R)-N-(3-(7-methyl-1H-indazol-5-yl)-1-(4-(1-methylpiperidin-4-yl)-1-oxopropan-2-yl)-4-(2-oxo-1,2-dihydroquinolin-3-yl)piperidine-1-carboxamide (BMS-742413): a potent human CGRP antagonist with superior safety profile for the treatment of migraine through intranasal delivery. [electronic resource] by
- Chaturvedula, Prasad V
- Mercer, Stephen E
- Pin, Sokhom S
- Thalody, George
- Xu, Cen
- Conway, Charlie M
- Keavy, Deborah
- Signor, Laura
- Cantor, Glenn H
- Mathias, Neil
- Moench, Paul
- Denton, Rex
- Macci, Robert
- Schartman, Richard
- Whiterock, Valerie
- Davis, Carl
- Macor, John E
- Dubowchik, Gene M
Producer: 20131209
In:
Bioorganic & medicinal chemistry letters vol. 23
Availability: No items available.
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1198.
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CGRP receptor activity in mice with global expression of human receptor activity modifying protein 1. [electronic resource] by
- Bohn, Keegan J
- Li, Baolin
- Huang, Xiaofang
- Mason, Bianca N
- Wattiez, Anne-Sophie
- Kuburas, Adisa
- Walker, Christopher S
- Yang, Peiyi
- Yu, Jianliang
- Heinz, Beverly A
- Johnson, Kirk W
- Russo, Andrew F
Producer: 20180129
In:
British journal of pharmacology vol. 174
Availability: No items available.
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